ATE305787T1 - 3,4-dihydro-(1h)chinazolin-2-on-verbindungen als csbp/p39-kinase-inhibitoren - Google Patents

3,4-dihydro-(1h)chinazolin-2-on-verbindungen als csbp/p39-kinase-inhibitoren

Info

Publication number
ATE305787T1
ATE305787T1 AT00980576T AT00980576T ATE305787T1 AT E305787 T1 ATE305787 T1 AT E305787T1 AT 00980576 T AT00980576 T AT 00980576T AT 00980576 T AT00980576 T AT 00980576T AT E305787 T1 ATE305787 T1 AT E305787T1
Authority
AT
Austria
Prior art keywords
csbp
kinase inhibitors
compounds
chinazoline
dihydro
Prior art date
Application number
AT00980576T
Other languages
English (en)
Inventor
Jerry L Adams
Michael J Bower
Jeffrey Charles Boehm
Don E Griswold
David C Underwood
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Application granted granted Critical
Publication of ATE305787T1 publication Critical patent/ATE305787T1/de

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/78—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/80—Oxygen atoms
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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AT00980576T 1999-11-23 2000-11-21 3,4-dihydro-(1h)chinazolin-2-on-verbindungen als csbp/p39-kinase-inhibitoren ATE305787T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US16697299P 1999-11-23 1999-11-23
PCT/US2000/031874 WO2001038313A1 (en) 1999-11-23 2000-11-21 3,4-DIHYDRO-(1H)QUINAZOLIN-2-ONE COMPOUNDS AS CSBP/p39 kINASE INHIBITORS

Publications (1)

Publication Number Publication Date
ATE305787T1 true ATE305787T1 (de) 2005-10-15

Family

ID=22605414

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00980576T ATE305787T1 (de) 1999-11-23 2000-11-21 3,4-dihydro-(1h)chinazolin-2-on-verbindungen als csbp/p39-kinase-inhibitoren

Country Status (8)

Country Link
US (1) US6982270B1 (de)
EP (1) EP1233950B1 (de)
JP (1) JP2003528043A (de)
AT (1) ATE305787T1 (de)
AU (1) AU1782301A (de)
DE (1) DE60023025T2 (de)
ES (1) ES2249309T3 (de)
WO (1) WO2001038313A1 (de)

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WO2006137421A1 (ja) * 2005-06-21 2006-12-28 Kyowa Hakko Kogyo Co., Ltd. 局所投与剤
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WO2008114119A2 (en) * 2007-03-20 2008-09-25 Cadila Pharmaceuticals Limited P38 inhibitors
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US20190060286A1 (en) 2016-02-29 2019-02-28 University Of Florida Research Foundation, Incorpo Chemotherapeutic Methods
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US6982270B1 (en) 2006-01-03
EP1233950A1 (de) 2002-08-28
DE60023025D1 (de) 2006-02-16
WO2001038313A1 (en) 2001-05-31
DE60023025T2 (de) 2006-07-13
ES2249309T3 (es) 2006-04-01

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