LV10181B - A nicotine containing stimulant unit - Google Patents

A nicotine containing stimulant unit Download PDF

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Publication number
LV10181B
LV10181B LVP-92-552A LV920552A LV10181B LV 10181 B LV10181 B LV 10181B LV 920552 A LV920552 A LV 920552A LV 10181 B LV10181 B LV 10181B
Authority
LV
Latvia
Prior art keywords
nicotine
water
composition according
mixture
stimulant
Prior art date
Application number
LVP-92-552A
Other languages
English (en)
Other versions
LV10181A (lv
Inventor
Anders Dam
Original Assignee
Anders Dam
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DK556089A external-priority patent/DK556089D0/da
Application filed by Anders Dam filed Critical Anders Dam
Publication of LV10181A publication Critical patent/LV10181A/lv
Publication of LV10181B publication Critical patent/LV10181B/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23GCOCOA; COCOA PRODUCTS, e.g. CHOCOLATE; SUBSTITUTES FOR COCOA OR COCOA PRODUCTS; CONFECTIONERY; CHEWING GUM; ICE-CREAM; PREPARATION THEREOF
    • A23G3/00Sweetmeats; Confectionery; Marzipan; Coated or filled products
    • A23G3/34Sweetmeats, confectionery or marzipan; Processes for the preparation thereof
    • A23G3/36Sweetmeats, confectionery or marzipan; Processes for the preparation thereof characterised by the composition containing organic or inorganic compounds
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23GCOCOA; COCOA PRODUCTS, e.g. CHOCOLATE; SUBSTITUTES FOR COCOA OR COCOA PRODUCTS; CONFECTIONERY; CHEWING GUM; ICE-CREAM; PREPARATION THEREOF
    • A23G3/00Sweetmeats; Confectionery; Marzipan; Coated or filled products
    • A23G3/34Sweetmeats, confectionery or marzipan; Processes for the preparation thereof
    • A23G3/36Sweetmeats, confectionery or marzipan; Processes for the preparation thereof characterised by the composition containing organic or inorganic compounds
    • A23G3/364Sweetmeats, confectionery or marzipan; Processes for the preparation thereof characterised by the composition containing organic or inorganic compounds containing microorganisms or enzymes; containing paramedical or dietetical agents, e.g. vitamins
    • A23G3/368Sweetmeats, confectionery or marzipan; Processes for the preparation thereof characterised by the composition containing organic or inorganic compounds containing microorganisms or enzymes; containing paramedical or dietetical agents, e.g. vitamins containing vitamins, antibiotics
    • AHUMAN NECESSITIES
    • A24TOBACCO; CIGARS; CIGARETTES; SIMULATED SMOKING DEVICES; SMOKERS' REQUISITES
    • A24BMANUFACTURE OR PREPARATION OF TOBACCO FOR SMOKING OR CHEWING; TOBACCO; SNUFF
    • A24B15/00Chemical features or treatment of tobacco; Tobacco substitutes, e.g. in liquid form
    • A24B15/10Chemical features of tobacco products or tobacco substitutes
    • A24B15/16Chemical features of tobacco products or tobacco substitutes of tobacco substitutes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/465Nicotine; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34Tobacco-abuse

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nutrition Science (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Food Science & Technology (AREA)
  • Inorganic Chemistry (AREA)
  • Polymers & Plastics (AREA)
  • Addiction (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • Microbiology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Zoology (AREA)
  • Physiology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Confectionery (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrane Compounds (AREA)
  • Manufacture Of Tobacco Products (AREA)

Claims (15)

  1. LV 10181 NIKOTĪNU SATUROŠS STIMULĒJOŠS SASTĀVS 5 PATENTA FORMULA 1. Siekalās šķīstošs stimulējošs sastāvs, kas satur aktīvu ingredientu un, pēc izvēles, ingredientus, kas satur gēlā ieslēgtas garšas un smaržas piedevas, kas iegūtas ar ūdeni saistošu gēlu 10 veidojošu aģentu, kurā aktīvais ingredients satur nikotīnu vai citus alkaloīdus ar tieši tādu pašu aktivitāti, minētam sastāvam ir i) tekstūras profils, kas noteikts ar tekstūras profila analīzi ar parametru rādītājiem sekojošās robežās : 15 a) izturība, t. i. modulis, lielāks kā 100 N/cm^; b) cietība, t. i. maksimālais spēks, kas pielikts pirmā saspiešanas ciklā, lielāks kā 5N/cm2; c) trauslums, t. i. deformācija procentos, kas vajadzīga, lai sagrautu gēlu, vismaz 30 %; 20 d) adhēzijas spēja, t. i. attiecība starp negatīvā pīķa laukumu starp diviem saspiešanas cikliem un pirmā pīķa laukumu, no 0 līdz 70 %; e) elastība, t. i. attiecība 100 x (D - d) / D, kur D ir parauga augstums (cm) pirms pirmā saspiešanas cikla, 25 un d ir parauga paliekošā deformācija (cm) pirms otra saspiešanas cikla, robežās no 25 līdz 100 %; f) kohēzijas spēja, t. i. kopējā darba attiecība starp pirmo un otro saspiešanas ciklu, robežās no 25 līdz 100 %; 30 ii) dezintegrācijas laiks, kas noteikts pie 37 °C, izmantojot dezintegrācijas testa aparātus atbilstoši Ph. Eur. otram izdevumam, robežās 5-60 minūtes; un 2 iii) nikotīna saturs no 0.5 līdz 10 mg vai tāda paša alkaloīda atbilstošs saturs.
  2. 2. Stimulējošs sastāvs, saskaņā ar 1. punktu, atšķirīgs ar to, 5 ka tekstūras profilam ir parametru rādītāji sekojošās robežās : a) izturība lielāka kā 200 N/cm^; b) cietība lielāka kā 25 N/cm^; c) trauslums vismaz 30 %; d) adhēzijas spēja no 0 līdz 40%; 10 e) elastība robežās no 50 līdz 100 %; f) kohēzijas spēja robežās no 40 līdz 100 %; un, ka dezintegrācijas laiks ir robežās 6 - 45 minūtes.
  3. 3. Stimulējošs sastāvs, saskaņā ar 1. un 2. punktiem, 15 atšķirīgs ar to, ka tekstūras profilam ir parametru rādītāji sekojošās robežās: a) izturība lielāka kā 400 N/cm^; b) cietība no 80 līdz 300 N/cm^; c) trauslums vismaz 30 %; 20 d) adhēzijas spēja no 0 līdz 20 %; e) elastība robežās no 80 līdz' 100 %; 0 kohēzijas spēja robežās no 40 līdz 100 %; un, ka dezintegrācijas laiks ir robežās 15 - 40 minūtes.
  4. 4. Stimulējošs sastāvs, saskaņā ar jebkuru no 1. - 3. punktiem, atšķirīgs ar to, ka gēlu veidojošais aģents satur želatīnu vai vienu vai vairākus sintētiskus vai dabīgus polisaharidus, labāk polisaharīdus, ko izmanto konditorejas produktu ražošanā.
  5. 5. Stimulējošs sastāvs, saskaņā ar jebkuru no 1. - 3. punktiem, atšķirīgs ar to, ka gēlu veidojošais aģents ir izvēlēts no grupas, kas satur agaru, algīnu, karagēnu (carrageenan), guāra (guar) sveķus, gumiarābiku, gata (ghatti) sveķus, astragāla (tragacanth) sveķus, karaija (karaya) sveķus, robinījas (locust) 35 sēklu sveķus, pektīnu, ksantāna (xanthan) sveķus, šajā gadījuma gumiarabiku un karagēnu (carrageenan), labāk gumiarābiku.
  6. 6. Stimulējošs sastāvs, saskaņā ar jebkuru no 1. - 5. punktiem, atšķirīgs ar to, ka garšas un smaržas piedevas satur vienu vai vairākus sintētiskus vai dabīgus garšas aģentus, kas izvēlēti no ēteriskām eļļām, esencēm, augļu sulām, un pulveriem, miltiem vai sasmalcināta augu materiāla, ieskaitot tabaku, kafiju, tēju un piparmētru.
  7. 7. Stimulējošs sastāvs saskaņā ar jebkuru no 1. - 6. punktiem, atšķirīgs ar to, ka piedevas satur vienu vai vairākus vitamīnus vai minerālus.
  8. 8. Stimulējošs sastāvs saskaņā ar jebkuru no 1. - 7. punktiem, atšķirīgs ar to, ka piedevas satur fizioloģiski saderīgu bufervielu vai aģentu.
  9. 9. Stimulējošs sastāvs saskaņā ar 8. punktu, atšķirīgs ar to, ka bufervielu vai aģentu un tā daudzumu izvēlas, lai, dezintegrējot sastāvu, nodrošinātu siekalās pH 8 -10.
  10. 10. Stimulējošs sastāvs saskaņā ar jebkuru no 8. - 9. punktiem, atšķirīgs ar to, ka bufervielas vai aģenta daudzums sastāvā ir no 5 mg līdz 50 mg.
  11. 11. Stimulējošs sastāvs, saskaņā ar jebkuru no 8. -10. punktiem, atšķirīgs ar to, ka buferviela vai aģents ietver sārmu metālu karbonātus, bikarbonātus, fosfātus, un/vai hidrogenfosfatus.
  12. 12. Stimulējošs sastāvs, saskaņā ar jebkuru no 1. -11. punktiem, atšķirīgs ar to, ka tas satur nikotīna daudzumu, kas izvēlēts robežās no 0,5 līdz 5.0 mg nikotīna, labāk robežās no 1.0 līdz 1.5 mg, no 1.5 līdz 2.5 mg, vai no 2.5 līdz 3.0 mg nikotīna, lai nodrošinātu vajadzīgo nikotīna stimulēšanu. 4
  13. 13. Stimulējošs sastāvs, saskaņā ar jebkuru no 1. -12. punktiem, atšķirīgs ar to, ka būtībā stabila nikotīna izdalīšana ir nodrošināta ar vienmērīgu nikotīna sadalījumu sastāvā. 5
  14. 14. Stimulējošs sastāvs, saskaņā ar jebkuru no 1. -12. punktiem, atšķirīgs ar to, ka izdalīšanās, kas ietver sākuma un uzturošu izdalīšanos, pakāpeniska izmainīšanās ir nodrošināta ar nikotīna strukturāli neviendabīgu sadalījumu daudzslāņainā 10 sastāvā.
  15. 15. Stimulējošs sastāvs, saskaņā ar jebkuru no 1. -14. punktiem, atšķirīgs ar to, ka tas ir noformēts tādā veidā, kas ir piemērots, lai pieliptu pie aukslējām.
LVP-92-552A 1989-11-07 1992-12-29 A nicotine containing stimulant unit LV10181B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DK556089A DK556089D0 (da) 1989-11-07 1989-11-07 Ryge supplement eller rygeerstatningsprodukt
DK615689A DK615689A (da) 1989-11-07 1989-12-04 Rygesupplement eller rygeerstatningsprodukt
PCT/DK1990/000280 WO1991006288A1 (en) 1989-11-07 1990-11-06 A nicotine containing stimulant unit

Publications (2)

Publication Number Publication Date
LV10181A LV10181A (lv) 1994-10-20
LV10181B true LV10181B (en) 1995-04-20

Family

ID=26067888

Family Applications (1)

Application Number Title Priority Date Filing Date
LVP-92-552A LV10181B (en) 1989-11-07 1992-12-29 A nicotine containing stimulant unit

Country Status (18)

Country Link
EP (1) EP0500658B1 (lv)
JP (2) JP2958663B2 (lv)
KR (1) KR0154341B1 (lv)
AT (1) ATE100707T1 (lv)
AU (1) AU648522B2 (lv)
BR (1) BR9007821A (lv)
CA (1) CA2073055C (lv)
DE (1) DE69006363T2 (lv)
DK (2) DK615689A (lv)
ES (1) ES2048510T3 (lv)
FI (1) FI101599B (lv)
HU (2) HUT62783A (lv)
IE (1) IE62388B1 (lv)
LV (1) LV10181B (lv)
NO (1) NO177082C (lv)
NZ (1) NZ235988A (lv)
PT (1) PT95813B (lv)
WO (1) WO1991006288A1 (lv)

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GB2299756A (en) * 1995-03-29 1996-10-16 Gilbert Falkingham Clayton Gelatinous pastille containing nicotine
US6082370A (en) * 1998-02-09 2000-07-04 Rousseau Research, Inc. Cigarette with dry powered Vitamin E
SE0103211D0 (sv) * 2001-09-27 2001-09-27 Pharmacia Ab New formulations and use thereof
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SI1578422T1 (sl) 2002-12-20 2007-12-31 Niconovum Ab Fizikalno in kemiäśno stabilni nikotin in mikrokristal na celulozo vsebujoäś material iz trdnih delcev
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CA2576344C (en) * 2004-08-11 2010-10-05 Cadbury Adams Usa Llc Warming compositions and delivery systems therefor
SE527323C2 (sv) * 2004-11-11 2006-02-07 Mahmood Valadi Cigarett
GB0501655D0 (en) * 2005-01-26 2005-03-02 Veritron Ltd Therapeutic use
WO2007104573A2 (en) 2006-03-16 2007-09-20 Niconovum Ab Improved snuff composition
US9032971B2 (en) 2006-11-15 2015-05-19 Philip Morris Usa Inc. Moist tobacco product and method of making
WO2010044736A1 (en) * 2008-10-14 2010-04-22 Mcneil Ab Multi portion intra-oral dosage form and use thereof
US9687023B2 (en) 2009-10-09 2017-06-27 Philip Morris Usa Inc. Moist smokeless tobacco product for oral usage having on a portion of the outer surface at least one friction reducing strip that provides texture during use
KR20130008535A (ko) * 2010-02-18 2013-01-22 자틴 바산트 타카르 니코틴을 함유하는 소프트 젤라틴 알약
US9775376B2 (en) * 2010-12-01 2017-10-03 R.J. Reynolds Tobacco Company Smokeless tobacco pastille and moulding process for forming smokeless tobacco products
WO2012116491A1 (zh) * 2011-03-02 2012-09-07 深圳市如烟生物科技有限公司 凝胶态水溶性烟用香精制备方法
US9629392B2 (en) 2011-09-22 2017-04-25 R.J. Reynolds Tobacco Company Translucent smokeless tobacco product
US20130078307A1 (en) 2011-09-22 2013-03-28 Niconovum Usa, Inc. Nicotine-containing pharmaceutical composition
US9084439B2 (en) 2011-09-22 2015-07-21 R.J. Reynolds Tobacco Company Translucent smokeless tobacco product
US9474303B2 (en) 2011-09-22 2016-10-25 R.J. Reynolds Tobacco Company Translucent smokeless tobacco product
GB2542192A (en) * 2015-09-11 2017-03-15 Revolymer (Uk) Ltd Chewable medicament
US20180199617A1 (en) * 2017-01-18 2018-07-19 Bianca Iodice Tobacco Free Hookah Smoking Gel
CN108693029A (zh) * 2018-04-09 2018-10-23 上海烟草集团有限责任公司 一种利用物性测试仪测试再造烟叶弹性的方法
US20210169784A1 (en) * 2019-12-09 2021-06-10 Nicoventures Trading Limited Buffered oral compositions
CN113197327B (zh) * 2021-05-13 2022-11-04 云南中烟工业有限责任公司 基于长链烷基二元脂肪酸尼古丁盐胶凝剂的凝胶
EP4371421A1 (en) 2022-11-18 2024-05-22 JT International SA A nicotine pouch product container, and a method of consuming nicotine pouch products therein

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Also Published As

Publication number Publication date
FI922066A (fi) 1992-05-07
DK615689A (da) 1991-05-08
NO921791D0 (no) 1992-05-06
DK615689D0 (da) 1989-12-04
IE903995A1 (en) 1991-05-08
NO177082B (no) 1995-04-10
EP0500658A1 (en) 1992-09-02
KR0154341B1 (ko) 1998-11-16
CA2073055C (en) 2000-01-25
NZ235988A (en) 1993-04-28
FI101599B1 (fi) 1998-07-31
NO177082C (no) 1995-07-19
EP0500658B1 (en) 1994-01-26
DK0500658T3 (da) 1994-05-09
DE69006363T2 (de) 1994-08-18
JPH05501880A (ja) 1993-04-08
AU648522B2 (en) 1994-04-28
WO1991006288A1 (en) 1991-05-16
PT95813A (pt) 1991-09-13
HUT62783A (en) 1993-06-28
HU9201521D0 (en) 1992-09-28
LV10181A (lv) 1994-10-20
NO921791L (no) 1992-07-03
JP2958663B2 (ja) 1999-10-06
IE62388B1 (en) 1995-01-25
JPH11315023A (ja) 1999-11-16
DE69006363D1 (de) 1994-03-10
ES2048510T3 (es) 1994-03-16
BR9007821A (pt) 1992-09-29
CA2073055A1 (en) 1991-05-08
ATE100707T1 (de) 1994-02-15
JP3357618B2 (ja) 2002-12-16
KR920703019A (ko) 1992-12-17
FI922066A0 (fi) 1992-05-07
FI101599B (fi) 1998-07-31
PT95813B (pt) 1997-11-28
AU6725490A (en) 1991-05-31

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