LU77530A1 - Procede et composes intermediaires pour la preparation de certaines 2-(piperazin-1-yle 4-substitue)-4-amino-quinazolines - Google Patents

Procede et composes intermediaires pour la preparation de certaines 2-(piperazin-1-yle 4-substitue)-4-amino-quinazolines

Info

Publication number
LU77530A1
LU77530A1 LU77530A LU77530A LU77530A1 LU 77530 A1 LU77530 A1 LU 77530A1 LU 77530 A LU77530 A LU 77530A LU 77530 A LU77530 A LU 77530A LU 77530 A1 LU77530 A1 LU 77530A1
Authority
LU
Luxembourg
Prior art keywords
substitue
yle
quinazolines
piperazin
amino
Prior art date
Application number
LU77530A
Other languages
English (en)
French (fr)
Inventor
P Hammen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of LU77530A1 publication Critical patent/LU77530A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
LU77530A 1976-06-15 1977-06-13 Procede et composes intermediaires pour la preparation de certaines 2-(piperazin-1-yle 4-substitue)-4-amino-quinazolines LU77530A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US69620176A 1976-06-15 1976-06-15

Publications (1)

Publication Number Publication Date
LU77530A1 true LU77530A1 (fr) 1979-03-26

Family

ID=24796111

Family Applications (1)

Application Number Title Priority Date Filing Date
LU77530A LU77530A1 (fr) 1976-06-15 1977-06-13 Procede et composes intermediaires pour la preparation de certaines 2-(piperazin-1-yle 4-substitue)-4-amino-quinazolines

Country Status (34)

Country Link
JP (1) JPS52153985A (ru)
AR (1) AR218251A1 (ru)
AT (1) AT356115B (ru)
BE (1) BE855656A (ru)
BG (3) BG35748A3 (ru)
CA (1) CA1068698A (ru)
CH (3) CH638203A5 (ru)
CS (1) CS202069B2 (ru)
DD (1) DD131021A5 (ru)
DE (1) DE2725019A1 (ru)
DK (1) DK146625C (ru)
EG (1) EG12922A (ru)
ES (1) ES459364A1 (ru)
FI (1) FI66853C (ru)
FR (1) FR2355015A1 (ru)
GB (1) GB1548856A (ru)
GR (1) GR72288B (ru)
HK (1) HK31481A (ru)
HU (1) HU177883B (ru)
IE (1) IE45423B1 (ru)
IL (1) IL52167A (ru)
LU (1) LU77530A1 (ru)
MY (1) MY8100270A (ru)
NL (1) NL172543C (ru)
NO (1) NO147838C (ru)
NZ (1) NZ184168A (ru)
PH (1) PH22196A (ru)
PL (3) PL111221B1 (ru)
PT (1) PT66617B (ru)
RO (3) RO73050A (ru)
SE (2) SE435380B (ru)
SU (2) SU1033002A3 (ru)
YU (1) YU40164B (ru)
ZA (1) ZA773014B (ru)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3346675A1 (de) * 1983-12-23 1985-07-04 Beiersdorf Ag, 2000 Hamburg Substituierte 1-(4-amino-6,7-dialkoxy-chinazolinyl)-4- cyclohexenyl-derivate des piperazins und homopiperazins, verfahren zu ihrer herstellung und ihre verwendung sowie diese verbindungen enthaltende zubereitungen und zwischenprodukte
AT384218B (de) * 1985-12-04 1987-10-12 Gerot Pharmazeutika Verfahren zur herstellung von neuen chinazolin-derivaten
CA2077252C (en) * 1992-08-31 2001-04-10 Khashayar Karimian Methods of making ureas and guanidines, and intermediates therefor
IL112249A (en) 1994-01-25 2001-11-25 Warner Lambert Co Pharmaceutical compositions containing di and tricyclic pyrimidine derivatives for inhibiting tyrosine kinases of the epidermal growth factor receptor family and some new such compounds
US5654307A (en) * 1994-01-25 1997-08-05 Warner-Lambert Company Bicyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family
IL112248A0 (en) 1994-01-25 1995-03-30 Warner Lambert Co Tricyclic heteroaromatic compounds and pharmaceutical compositions containing them
US5932538A (en) * 1996-02-02 1999-08-03 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3511836A (en) 1967-12-13 1970-05-12 Pfizer & Co C 2,4,6,7-tetra substituted quinazolines
US3669968A (en) 1970-05-21 1972-06-13 Pfizer Trialkoxy quinazolines
JPS4966691A (ru) * 1972-10-30 1974-06-27
US3935213A (en) 1973-12-05 1976-01-27 Pfizer Inc. Process for hypotensive 4-amino-2-(piperazin-1-yl) quinazoline derivatives
JPS50126682A (ru) * 1974-03-25 1975-10-04

Also Published As

Publication number Publication date
SU1033002A3 (ru) 1983-07-30
CH638516A5 (en) 1983-09-30
DE2725019A1 (de) 1977-12-22
NO147838C (no) 1983-06-22
IE45423B1 (en) 1982-08-25
FI66853B (fi) 1984-08-31
RO77308A (ro) 1981-08-17
DK240877A (da) 1977-12-16
FI771741A (ru) 1977-12-16
EG12922A (en) 1980-03-31
CA1068698A (en) 1979-12-25
CH638203A5 (en) 1983-09-15
SE450120B (sv) 1987-06-09
CH638517A5 (en) 1983-09-30
IL52167A (en) 1981-01-30
PL105558B1 (pl) 1979-10-31
AU2558377A (en) 1978-09-07
AR218251A1 (es) 1980-05-30
BG35748A3 (en) 1984-06-15
JPS5543465B2 (ru) 1980-11-06
NL7705939A (nl) 1977-12-19
NZ184168A (en) 1979-08-31
BG35594A3 (en) 1984-05-15
NO147838B (no) 1983-03-14
BG35747A3 (en) 1984-06-15
SU946402A3 (ru) 1982-07-23
RO77330A (ro) 1981-06-22
ZA773014B (en) 1978-04-26
DD131021A5 (de) 1978-05-24
ATA386977A (de) 1979-09-15
AT356115B (de) 1980-04-10
HK31481A (en) 1981-07-10
IL52167A0 (en) 1977-07-31
JPS52153985A (en) 1977-12-21
SE8107554L (sv) 1981-12-16
IE45423L (en) 1977-12-15
PL111221B1 (en) 1980-08-30
PT66617A (en) 1977-06-01
CS202069B2 (en) 1980-12-31
DK146625B (da) 1983-11-21
PH22196A (en) 1988-06-28
DK146625C (da) 1984-06-04
HU177883B (en) 1982-01-28
FR2355015A1 (fr) 1978-01-13
PT66617B (en) 1978-10-27
ES459364A1 (es) 1978-03-16
YU40164B (en) 1985-08-31
SE7705745L (sv) 1977-12-16
NL172543C (nl) 1983-09-16
MY8100270A (en) 1981-12-31
FR2355015B1 (ru) 1981-07-24
BE855656A (fr) 1977-12-14
YU132677A (en) 1982-08-31
GB1548856A (en) 1979-07-18
RO73050A (ro) 1981-08-30
NO771919L (no) 1977-12-16
PL113012B1 (en) 1980-11-29
PL198874A1 (pl) 1978-04-10
FI66853C (fi) 1984-12-10
SE435380B (sv) 1984-09-24
NL172543B (nl) 1983-04-18
GR72288B (ru) 1983-10-17

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