KR840000079B1 - 6-β-치환된 페니실란산 유도체의 제조방법 - Google Patents

6-β-치환된 페니실란산 유도체의 제조방법 Download PDF

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Publication number
KR840000079B1
KR840000079B1 KR1019800001920A KR800001920A KR840000079B1 KR 840000079 B1 KR840000079 B1 KR 840000079B1 KR 1019800001920 A KR1019800001920 A KR 1019800001920A KR 800001920 A KR800001920 A KR 800001920A KR 840000079 B1 KR840000079 B1 KR 840000079B1
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KR
South Korea
Prior art keywords
acid
ester
substituted
mixture
formula
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Expired
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KR1019800001920A
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English (en)
Korean (ko)
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KR830002769A (ko
Inventor
에드워드 글라인 켐프 존
Original Assignee
화이자 리미티드
알란 프랑크 임페이
죠오지 알란스미
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Publication of KR830002769A publication Critical patent/KR830002769A/ko
Application granted granted Critical
Publication of KR840000079B1 publication Critical patent/KR840000079B1/ko
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04—Preparation
    • C07D499/10—Modification of an amino radical directly attached in position 6
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1019800001920A 1979-05-19 1980-05-15 6-β-치환된 페니실란산 유도체의 제조방법 Expired KR840000079B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7917505 1979-05-19
GB7917505 1979-05-19

Publications (2)

Publication Number Publication Date
KR830002769A KR830002769A (ko) 1983-05-30
KR840000079B1 true KR840000079B1 (ko) 1984-02-08

Family

ID=10505288

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019800001920A Expired KR840000079B1 (ko) 1979-05-19 1980-05-15 6-β-치환된 페니실란산 유도체의 제조방법

Country Status (28)

Country Link
US (1) US4356122A (enExample)
JP (1) JPS5941994B2 (enExample)
KR (1) KR840000079B1 (enExample)
AR (1) AR225038A1 (enExample)
AT (1) AT366694B (enExample)
AU (1) AU517488B2 (enExample)
BE (1) BE883319A (enExample)
CA (1) CA1140916A (enExample)
CH (1) CH650262A5 (enExample)
CS (1) CS214756B2 (enExample)
DD (1) DD151310A5 (enExample)
DE (1) DE3018847C2 (enExample)
DK (1) DK155180A (enExample)
ES (1) ES491612A0 (enExample)
FI (1) FI71562C (enExample)
FR (1) FR2457293A1 (enExample)
GR (1) GR68461B (enExample)
IE (1) IE49804B1 (enExample)
IL (1) IL60097A (enExample)
IT (1) IT1140946B (enExample)
LU (1) LU82458A1 (enExample)
NL (1) NL180937C (enExample)
NO (1) NO801473L (enExample)
PH (1) PH15033A (enExample)
PL (1) PL224188A1 (enExample)
PT (1) PT71253A (enExample)
SE (1) SE449995B (enExample)
ZA (1) ZA802908B (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA803742B (en) * 1979-07-02 1981-06-24 Beecham Group Ltd Penicillanic acid derivatives, their preparation and use
JPS6034969A (ja) * 1983-08-08 1985-02-22 Toyama Chem Co Ltd 新規なペニシラン酸誘導体およびその塩類
WO2018175927A2 (en) * 2017-03-23 2018-09-27 Trucode Gene Repair, Inc. Peptide nucleic acid (pna) monomers with an orthogonally protected ester moiety

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5749555B2 (enExample) * 1973-04-04 1982-10-22
US4282149A (en) * 1977-03-21 1981-08-04 Massachusetts Institute Of Technology Carbon and oxygen analogs of penicillin
US4265882A (en) * 1977-10-03 1981-05-05 Massachusetts Institute Of Technology Sulphur analogs of penicillins having a nucleophile substituted in the 6 and 7 position, respectively

Also Published As

Publication number Publication date
IT8022104A0 (it) 1980-05-16
JPS5941994B2 (ja) 1984-10-11
LU82458A1 (fr) 1980-10-08
AR225038A1 (es) 1982-02-15
SE449995B (sv) 1987-06-01
CS214756B2 (en) 1982-05-28
FI801581A7 (fi) 1980-11-20
FI71562C (fi) 1987-01-19
PT71253A (en) 1980-06-01
IE801024L (en) 1980-11-19
NL180937B (nl) 1986-12-16
ES8105737A1 (es) 1981-05-16
PL224188A1 (enExample) 1981-02-13
FI71562B (fi) 1986-10-10
AU5846880A (en) 1980-11-27
CH650262A5 (de) 1985-07-15
FR2457293A1 (fr) 1980-12-19
DE3018847C2 (de) 1982-09-30
JPS55157588A (en) 1980-12-08
IE49804B1 (en) 1985-12-25
ATA259780A (de) 1981-09-15
KR830002769A (ko) 1983-05-30
GR68461B (enExample) 1981-12-30
IL60097A0 (en) 1980-07-31
IT1140946B (it) 1986-10-10
IL60097A (en) 1983-02-23
NO801473L (no) 1980-11-20
AT366694B (de) 1982-04-26
AU517488B2 (en) 1981-08-06
DE3018847A1 (de) 1980-12-11
DD151310A5 (de) 1981-10-14
ZA802908B (en) 1981-05-27
FR2457293B1 (enExample) 1983-05-20
PH15033A (en) 1982-05-20
DK155180A (da) 1980-11-20
US4356122A (en) 1982-10-26
CA1140916A (en) 1983-02-08
NL180937C (nl) 1987-05-18
NL8002843A (nl) 1980-11-21
BE883319A (fr) 1980-11-14
ES491612A0 (es) 1981-05-16
SE8003676L (sv) 1980-11-20

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