KR20160090846A - 치환된 벤즈아마이드 및 이의 이용 방법 - Google Patents
치환된 벤즈아마이드 및 이의 이용 방법 Download PDFInfo
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- KR20160090846A KR20160090846A KR1020167016643A KR20167016643A KR20160090846A KR 20160090846 A KR20160090846 A KR 20160090846A KR 1020167016643 A KR1020167016643 A KR 1020167016643A KR 20167016643 A KR20167016643 A KR 20167016643A KR 20160090846 A KR20160090846 A KR 20160090846A
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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- A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
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| US10370368B2 (en) | 2015-11-30 | 2019-08-06 | Merck Sharp & Dohme Corp. | Aryl acylsulfonamides as BLT1 antagonists |
| EP3390374B1 (en) | 2015-12-18 | 2020-08-26 | Merck Sharp & Dohme Corp. | Hydroxyalkylamine- and hydroxycycloalkylamine-substituted diamine-arylsulfonamide compounds with selective activity in voltage-gated sodium channels |
| KR20180086259A (ko) | 2016-02-03 | 2018-07-30 | 상하이 하이옌 파마슈티컬 테크놀로지 컴퍼니, 리미티드 | 헤테로 고리로 치환된 n-설포닐벤즈아미드 유도체, 이의 제조 방법과 약학적 용도 |
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| HRP20250505T1 (hr) * | 2016-05-20 | 2025-06-20 | Xenon Pharmaceuticals Inc. | Spojevi benzensulfonamida i njihova uporaba za terapijska sredstva |
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| JP2020511511A (ja) | 2017-03-24 | 2020-04-16 | ジェネンテック, インコーポレイテッド | ナトリウムチャネル阻害剤としての4−ピペリジン−n−(ピリミジン−4−イル)クロマン−7−スルホンアミド誘導体 |
| AU2018300980A1 (en) | 2017-07-12 | 2020-01-02 | Vanderbilt University | Antagonists of the muscarinic acetylcholine receptor M4 |
| CN110300745B (zh) * | 2017-07-24 | 2023-03-31 | 上海海雁医药科技有限公司 | 钠离子通道抑制剂及其药学上可接受的盐和多晶型物及其应用 |
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-
2014
- 2014-11-26 CR CR20160296A patent/CR20160296A/es unknown
- 2014-11-26 CA CA2931732A patent/CA2931732A1/en not_active Abandoned
- 2014-11-26 KR KR1020167016643A patent/KR20160090846A/ko not_active Withdrawn
- 2014-11-26 JP JP2016534731A patent/JP6383418B2/ja not_active Expired - Fee Related
- 2014-11-26 EP EP18197734.9A patent/EP3450428A1/en not_active Withdrawn
- 2014-11-26 EP EP14865855.2A patent/EP3074377B1/en active Active
- 2014-11-26 CN CN201480064734.4A patent/CN105793238B/zh not_active Expired - Fee Related
- 2014-11-26 AU AU2014356967A patent/AU2014356967A1/en not_active Abandoned
- 2014-11-26 EA EA201691085A patent/EA201691085A1/ru unknown
- 2014-11-26 MX MX2016006936A patent/MX2016006936A/es unknown
- 2014-11-26 PE PE2016000696A patent/PE20161247A1/es not_active Application Discontinuation
- 2014-11-26 WO PCT/CN2014/092269 patent/WO2015078374A1/en not_active Ceased
- 2014-11-27 TW TW103141262A patent/TWI560180B/zh not_active IP Right Cessation
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2015
- 2015-01-22 US US14/603,273 patent/US9546164B2/en not_active Expired - Fee Related
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- 2016-05-25 IL IL245844A patent/IL245844A0/en unknown
- 2016-05-26 CL CL2016001287A patent/CL2016001287A1/es unknown
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- 2016-09-23 US US15/275,131 patent/US9694002B2/en not_active Expired - Fee Related
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2018
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2019
- 2019-04-22 US US16/390,957 patent/US20200108054A1/en not_active Abandoned
- 2019-11-07 US US16/677,487 patent/US20210093618A1/en not_active Abandoned
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| IL245844A0 (en) | 2016-08-02 |
| HK1223913A1 (zh) | 2017-08-11 |
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| US9546164B2 (en) | 2017-01-17 |
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| TWI560180B (en) | 2016-12-01 |
| US20200108054A1 (en) | 2020-04-09 |
| CN105793238B (zh) | 2019-12-24 |
| JP6383418B2 (ja) | 2018-08-29 |
| PE20161247A1 (es) | 2016-11-30 |
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| CA2931732A1 (en) | 2015-06-04 |
| CR20160296A (es) | 2016-09-20 |
| JP2018188466A (ja) | 2018-11-29 |
| MX2016006936A (es) | 2016-10-05 |
| US20150252038A1 (en) | 2015-09-10 |
| TW201533021A (zh) | 2015-09-01 |
| US9694002B2 (en) | 2017-07-04 |
| JP2017504571A (ja) | 2017-02-09 |
| CN105793238A (zh) | 2016-07-20 |
| EP3074377A4 (en) | 2017-04-19 |
| EP3074377A1 (en) | 2016-10-05 |
| PH12016501007A1 (en) | 2016-07-18 |
| WO2015078374A1 (en) | 2015-06-04 |
| AU2014356967A1 (en) | 2016-07-07 |
| US20170087136A1 (en) | 2017-03-30 |
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