KR101170925B1 - 암 치료용 키네신 방추 단백질 (ｋｓｐ) 억제제로서의ｎ-(1-(1-벤질-4-페닐-1ｈ-이미다졸-2-일)-2,2-디메틸프로필)벤자미드 유도체 및 관련 화합물 - Google Patents

암 치료용 키네신 방추 단백질 (ｋｓｐ) 억제제로서의ｎ-(1-(1-벤질-4-페닐-1ｈ-이미다졸-2-일)-2,2-디메틸프로필)벤자미드 유도체 및 관련 화합물 Download PDF

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KR101170925B1
KR101170925B1 KR1020077000979A KR20077000979A KR101170925B1 KR 101170925 B1 KR101170925 B1 KR 101170925B1 KR 1020077000979 A KR1020077000979 A KR 1020077000979A KR 20077000979 A KR20077000979 A KR 20077000979A KR 101170925 B1 KR101170925 B1 KR 101170925B1
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imidazol
benzyl
phenyl
propyl
dimethylpropyl
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KR20070106961A (ko
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웨이보 왕
폴 에이. 바르산티
이 시
러스텀 에스. 보이스
사비나 페치
나탄 브래미어
메간 필립스
크리스 멘덴홀
켈리 와이만
리아나 마리 라그니톤
라이언 콘스탄틴
홍 양
엘리자베스 미에울리
사비트리 라무르티
엘리사 자잔
아누 샤르마
자인 라마
샤라드하 사브라마니안
폴 레노웨
케네스 월터 바어
데이빗 듈
아네트 월터
틴야 아브람스
케이 허
에릭 마틴
마크 냅
빈센트 레
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노바티스 백신즈 앤드 다이아그노스틱스 인코포레이티드
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
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    • C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
KR1020077000979A 2004-06-18 2005-06-20 암 치료용 키네신 방추 단백질 (ｋｓｐ) 억제제로서의ｎ-(1-(1-벤질-4-페닐-1ｈ-이미다졸-2-일)-2,2-디메틸프로필)벤자미드 유도체 및 관련 화합물 Expired - Fee Related KR101170925B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US58092704P 2004-06-18 2004-06-18
US60/580,927 2004-06-18
PCT/US2005/022062 WO2006002236A1 (en) 2004-06-18 2005-06-20 N- (1- (1-benzyl -4-phenyl-1h-imidazol-2-yl) -2,2-dymethylpropyl) benzamide derivatives and related compounds as kinesin spindle protein (ksp) inhibitors for the treatment of cancer

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KR20070106961A KR20070106961A (ko) 2007-11-06
KR101170925B1 true KR101170925B1 (ko) 2012-08-07

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US (3) US7576221B2 (enExample)
EP (1) EP1765789B1 (enExample)
JP (2) JP4836280B2 (enExample)
KR (1) KR101170925B1 (enExample)
CN (1) CN1993331A (enExample)
AU (1) AU2005258135B2 (enExample)
BR (1) BRPI0510929A (enExample)
CA (1) CA2571002A1 (enExample)
EC (1) ECSP077183A (enExample)
ES (1) ES2409345T3 (enExample)
IL (1) IL180147A0 (enExample)
MA (1) MA28739B1 (enExample)
MX (1) MXPA06014909A (enExample)
NO (1) NO20070343L (enExample)
NZ (1) NZ552510A (enExample)
RU (1) RU2427572C2 (enExample)
SG (1) SG153851A1 (enExample)
TN (1) TNSN06419A1 (enExample)
TW (1) TW200612958A (enExample)
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KR20070106961A (ko) 2007-11-06
EP1765789A1 (en) 2007-03-28
NO20070343L (no) 2007-03-05
JP4836280B2 (ja) 2011-12-14
BRPI0510929A (pt) 2007-07-17
MA28739B1 (fr) 2007-07-02
AU2005258135B2 (en) 2011-09-22
TW200612958A (en) 2006-05-01
EP1765789B1 (en) 2013-02-27
SG153851A1 (en) 2009-07-29
CA2571002A1 (en) 2006-01-05
ECSP077183A (es) 2007-02-28
IL180147A0 (en) 2007-06-03
US20130017196A1 (en) 2013-01-17
US20060009472A1 (en) 2006-01-12
NZ552510A (en) 2010-12-24
CN1993331A (zh) 2007-07-04
ZA200700481B (en) 2008-10-29
US8735599B2 (en) 2014-05-27
AU2005258135A1 (en) 2006-01-05
RU2007101612A (ru) 2008-08-10
JP2011256197A (ja) 2011-12-22
ES2409345T3 (es) 2013-06-26
US7576221B2 (en) 2009-08-18
JP2008503501A (ja) 2008-02-07
US20090258016A1 (en) 2009-10-15
TNSN06419A1 (en) 2008-02-22
US8318791B2 (en) 2012-11-27
MXPA06014909A (es) 2007-02-28
RU2427572C2 (ru) 2011-08-27

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