KR100583704B1 - 4-아미노-5-페닐-7-시클로부틸-피롤로 (2,3-ｄ) 피리미딘유도체 - Google Patents

4-아미노-5-페닐-7-시클로부틸-피롤로 (2,3-ｄ) 피리미딘유도체 Download PDF

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Publication number
KR100583704B1
KR100583704B1 KR1020037014725A KR20037014725A KR100583704B1 KR 100583704 B1 KR100583704 B1 KR 100583704B1 KR 1020037014725 A KR1020037014725 A KR 1020037014725A KR 20037014725 A KR20037014725 A KR 20037014725A KR 100583704 B1 KR100583704 B1 KR 100583704B1
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South Korea
Prior art keywords
lower alkyl
phenyl
amino
pyrrolo
benzyloxy
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Korean (ko)
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KR20030096386A (ko
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한스-게오르그 카프라로
파스칼 푸레트
카를로스 가르시아-에체베리아
폴 윌리엄 맨리
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노파르티스 아게
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Priority claimed from GB0111764A external-priority patent/GB0111764D0/en
Priority claimed from GB0204752A external-priority patent/GB0204752D0/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020037014725A 2001-05-14 2002-05-13 4-아미노-5-페닐-7-시클로부틸-피롤로 (2,3-ｄ) 피리미딘유도체 Expired - Fee Related KR100583704B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0111764.7 2001-05-14
GB0111764A GB0111764D0 (en) 2001-05-14 2001-05-14 Organic compounds
GB0204752A GB0204752D0 (en) 2002-02-28 2002-02-28 Organic compounds
GB0204752.0 2002-02-28
PCT/EP2002/005239 WO2002092599A1 (en) 2001-05-14 2002-05-13 4-amino-5-phenyl-7-cyclobutyl-pyrrolo (2,3-d) pyrimidine derivatives

Publications (2)

Publication Number Publication Date
KR20030096386A KR20030096386A (ko) 2003-12-24
KR100583704B1 true KR100583704B1 (ko) 2006-05-26

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KR1020037014725A Expired - Fee Related KR100583704B1 (ko) 2001-05-14 2002-05-13 4-아미노-5-페닐-7-시클로부틸-피롤로 (2,3-ｄ) 피리미딘유도체

Country Status (26)

Country Link
US (1) US7326699B2 (https=)
EP (1) EP1390369B1 (https=)
JP (1) JP4099399B2 (https=)
KR (1) KR100583704B1 (https=)
CN (1) CN1264844C (https=)
AR (1) AR035885A1 (https=)
AT (1) ATE309245T1 (https=)
AU (1) AU2002312905B2 (https=)
BR (1) BR0209658A (https=)
CA (1) CA2446435C (https=)
CO (1) CO5540346A2 (https=)
CZ (1) CZ20033067A3 (https=)
DE (1) DE60207241T2 (https=)
ES (1) ES2252465T3 (https=)
HU (1) HUP0304082A3 (https=)
IL (1) IL158697A0 (https=)
MX (1) MXPA03010402A (https=)
MY (1) MY124853A (https=)
NO (1) NO20034929L (https=)
NZ (1) NZ529256A (https=)
PE (1) PE20021096A1 (https=)
PL (1) PL363866A1 (https=)
RU (1) RU2305682C2 (https=)
SK (1) SK14022003A3 (https=)
TW (1) TWI238824B (https=)
WO (1) WO2002092599A1 (https=)

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