KR100317149B1 - 신규한에리트로마이신유도체,그의제조방법및그의의약으로서의용도 - Google Patents

신규한에리트로마이신유도체,그의제조방법및그의의약으로서의용도 Download PDF

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Publication number
KR100317149B1
KR100317149B1 KR1019930023371A KR930023371A KR100317149B1 KR 100317149 B1 KR100317149 B1 KR 100317149B1 KR 1019930023371 A KR1019930023371 A KR 1019930023371A KR 930023371 A KR930023371 A KR 930023371A KR 100317149 B1 KR100317149 B1 KR 100317149B1
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South Korea
Prior art keywords
formula
compound
methyl
group
dideoxy
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
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KR1019930023371A
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English (en)
Korean (ko)
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KR940011474A (ko
Inventor
꽁스땅뗑아구리다
알렝본느프와
쟝-프랑스와샹또
알렉시스데니
오딜르르마르뜨레
Original Assignee
쟝-끌로드 비에이으포스
로우셀-우크라프
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Priority claimed from FR9213320A external-priority patent/FR2697523B1/fr
Priority claimed from FR9308109A external-priority patent/FR2707088B1/fr
Application filed by 쟝-끌로드 비에이으포스, 로우셀-우크라프 filed Critical 쟝-끌로드 비에이으포스
Publication of KR940011474A publication Critical patent/KR940011474A/ko
Application granted granted Critical
Publication of KR100317149B1 publication Critical patent/KR100317149B1/ko
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
KR1019930023371A 1992-11-05 1993-11-05 신규한에리트로마이신유도체,그의제조방법및그의의약으로서의용도 Expired - Lifetime KR100317149B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR9213320A FR2697523B1 (fr) 1992-11-05 1992-11-05 Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR92-13320 1992-11-05
FR93-08109 1993-07-02
FR9308109A FR2707088B1 (fr) 1993-07-02 1993-07-02 Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Publications (2)

Publication Number Publication Date
KR940011474A KR940011474A (ko) 1994-06-21
KR100317149B1 true KR100317149B1 (ko) 2002-06-20

Family

ID=26229842

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019930023371A Expired - Lifetime KR100317149B1 (ko) 1992-11-05 1993-11-05 신규한에리트로마이신유도체,그의제조방법및그의의약으로서의용도

Country Status (16)

Country Link
US (2) US5527780A (enExample)
EP (1) EP0596802B1 (enExample)
JP (2) JP3000022B2 (enExample)
KR (1) KR100317149B1 (enExample)
CN (1) CN1040876C (enExample)
AT (1) ATE135706T1 (enExample)
AU (1) AU670329B2 (enExample)
BR (1) BR9304481A (enExample)
CA (1) CA2102457C (enExample)
DE (1) DE69301897T2 (enExample)
DK (1) DK0596802T3 (enExample)
ES (1) ES2085130T3 (enExample)
GR (1) GR3019385T3 (enExample)
HU (3) HU222113B1 (enExample)
MA (1) MA23018A1 (enExample)
RU (1) RU2126416C1 (enExample)

Families Citing this family (86)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2718450B1 (fr) * 1994-04-08 1997-01-10 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR2719587B1 (fr) * 1994-05-03 1996-07-12 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR2727969B1 (fr) * 1994-12-09 1997-01-17 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2732023B1 (fr) * 1995-03-22 1997-04-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2732684B1 (fr) * 1995-04-06 1997-04-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
US5747466A (en) * 1995-11-08 1998-05-05 Abbott Laboratories 3-deoxy-3-descladinose derivatives of erythromycins A and B
FR2742757B1 (fr) 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2751656B1 (fr) * 1996-07-24 1998-10-16 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
DE69733370T2 (de) * 1996-09-04 2006-02-02 Abbott Laboratories, Abbott Park 6-o-Substituierte Ketoliden mit antibakteriellen Wirkung
UA51730C2 (uk) * 1996-09-04 2002-12-16 Ебботт Лабораторіз 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
FR2757168B1 (fr) * 1996-12-12 1999-06-11 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2760017B1 (fr) * 1997-02-27 1999-04-30 Hoechst Marion Roussel Inc Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments
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US6034069A (en) * 1997-09-30 2000-03-07 Abbott Laboratories 3-'N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity
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Also Published As

Publication number Publication date
GR3019385T3 (en) 1996-06-30
JP3000022B2 (ja) 2000-01-17
BR9304481A (pt) 1994-06-21
ATE135706T1 (de) 1996-04-15
AU5047793A (en) 1994-05-19
KR940011474A (ko) 1994-06-21
CA2102457C (fr) 2002-01-22
JP3151188B2 (ja) 2001-04-03
DE69301897T2 (de) 1996-11-07
ES2085130T3 (es) 1996-05-16
HU221978B1 (hu) 2003-03-28
DK0596802T3 (da) 1996-06-03
JPH11180994A (ja) 1999-07-06
JPH06220082A (ja) 1994-08-09
HU220048B (hu) 2001-10-28
EP0596802A1 (fr) 1994-05-11
HU222113B1 (hu) 2003-04-28
DE69301897D1 (de) 1996-04-25
CN1090581A (zh) 1994-08-10
RU2126416C1 (ru) 1999-02-20
EP0596802B1 (fr) 1996-03-20
US5527780A (en) 1996-06-18
CN1040876C (zh) 1998-11-25
HU0003975D0 (enExample) 2000-12-28
AU670329B2 (en) 1996-07-11
MA23018A1 (fr) 1994-07-01
HUT66446A (en) 1994-11-28
CA2102457A1 (fr) 1994-05-06
US5614614A (en) 1997-03-25

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