KR100196256B1 - 서방성 약물 제형 - Google Patents
서방성 약물 제형 Download PDFInfo
- Publication number
- KR100196256B1 KR100196256B1 KR1019920702558A KR920702558A KR100196256B1 KR 100196256 B1 KR100196256 B1 KR 100196256B1 KR 1019920702558 A KR1019920702558 A KR 1019920702558A KR 920702558 A KR920702558 A KR 920702558A KR 100196256 B1 KR100196256 B1 KR 100196256B1
- Authority
- KR
- South Korea
- Prior art keywords
- membrane
- drug
- consisting essentially
- colon
- formulation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
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- KRKNYBCHXYNGOX-UHFFFAOYSA-N citric acid Chemical class OC(=O)CC(O)(C(O)=O)CC(O)=O KRKNYBCHXYNGOX-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT20054A/90 | 1990-04-17 | ||
| IT02005490A IT1246382B (it) | 1990-04-17 | 1990-04-17 | Metodo per la cessione mirata e controllata di farmaci nell'intestino e particolarmente nel colon |
| PCT/EP1991/000688 WO1991016042A1 (en) | 1990-04-17 | 1991-04-09 | Controlled release drug formulation |
Publications (2)
| Publication Number | Publication Date |
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| KR930700077A KR930700077A (ko) | 1993-03-13 |
| KR100196256B1 true KR100196256B1 (ko) | 1999-06-15 |
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| KR1019920702558A Expired - Fee Related KR100196256B1 (ko) | 1990-04-17 | 1991-04-09 | 서방성 약물 제형 |
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| EP (2) | EP0453001A1 (https=) |
| JP (2) | JP3194974B2 (https=) |
| KR (1) | KR100196256B1 (https=) |
| AT (1) | ATE144138T1 (https=) |
| AU (1) | AU654277B2 (https=) |
| CA (2) | CA2035155A1 (https=) |
| DE (1) | DE69122751T2 (https=) |
| DK (1) | DK0524989T3 (https=) |
| ES (1) | ES2093097T3 (https=) |
| GR (1) | GR3021847T3 (https=) |
| IE (1) | IE911271A1 (https=) |
| IT (1) | IT1246382B (https=) |
| NZ (1) | NZ237823A (https=) |
| PT (1) | PT97370B (https=) |
| RU (1) | RU2111743C1 (https=) |
| SG (1) | SG46584A1 (https=) |
| TW (1) | TW223022B (https=) |
| WO (1) | WO1991016042A1 (https=) |
| ZA (1) | ZA912792B (https=) |
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| US3473490A (en) * | 1966-01-17 | 1969-10-21 | Camillo Corvi Mora | Producing chronoactive pharmaceutical granules |
| GB1468172A (en) * | 1973-03-28 | 1977-03-23 | Benzon As Alfred | Oral drug preparations |
| FR2471186A1 (fr) * | 1979-12-10 | 1981-06-19 | Roussel Uclaf | Nouveaux comprimes a delitescence colique, ainsi que leur procede de preparation |
| JPS57171428A (en) * | 1981-04-13 | 1982-10-22 | Sankyo Co Ltd | Preparation of coated solid preparation |
| DK58983D0 (da) * | 1983-02-11 | 1983-02-11 | Leo Pharm Prod Ltd | Farmaceutisk praeparat |
| US4503030A (en) * | 1983-06-06 | 1985-03-05 | Alza Corporation | Device for delivering drug to certain pH environments |
| SE457505B (sv) * | 1984-01-10 | 1989-01-09 | Lejus Medical Ab | Laminatbelagd oral farmaceutisk komposition och foerfarande foer dess framstaellning |
| DK62184D0 (da) * | 1984-02-10 | 1984-02-10 | Benzon As Alfred | Diffusionsovertrukket polydepotpraeparat |
| DE3572440D1 (en) * | 1984-06-19 | 1989-09-28 | Basf Ag | Gastro-resistant cylindrical pancreatine-microtablets |
| EP0212745B1 (en) * | 1985-08-16 | 1991-04-10 | The Procter & Gamble Company | Drug particles having constant release |
| JPS6261916A (ja) * | 1985-09-12 | 1987-03-18 | Fujisawa Pharmaceut Co Ltd | 持続性製剤 |
| AU591248B2 (en) * | 1986-03-27 | 1989-11-30 | Kinaform Technology, Inc. | Sustained-release pharaceutical preparation |
| US5238686A (en) * | 1986-03-27 | 1993-08-24 | Kinaform Technology, Inc. | Sustained-release pharmaceutical preparation |
| US4800087A (en) * | 1986-11-24 | 1989-01-24 | Mehta Atul M | Taste-masked pharmaceutical compositions |
| SE460945B (sv) * | 1987-01-15 | 1989-12-11 | Lejus Medical Ab | En multipel-unit-dos komposition av furosemid |
| JPH0768125B2 (ja) * | 1988-05-18 | 1995-07-26 | エーザイ株式会社 | 酸不安定化合物の内服用製剤 |
| US4925676A (en) * | 1989-02-02 | 1990-05-15 | Warner-Lambert Company | Extended release gemfibrozil composition |
| US5026559A (en) * | 1989-04-03 | 1991-06-25 | Kinaform Technology, Inc. | Sustained-release pharmaceutical preparation |
| US4983401A (en) * | 1989-05-22 | 1991-01-08 | Kinaform Technology, Inc. | Sustained release pharmaceutical preparations having pH controlled membrane coatings |
-
1990
- 1990-04-17 IT IT02005490A patent/IT1246382B/it active IP Right Grant
-
1991
- 1991-01-29 EP EP91200173A patent/EP0453001A1/en not_active Withdrawn
- 1991-01-29 CA CA002035155A patent/CA2035155A1/en not_active Abandoned
- 1991-01-30 JP JP02778491A patent/JP3194974B2/ja not_active Expired - Lifetime
- 1991-04-09 AU AU76798/91A patent/AU654277B2/en not_active Ceased
- 1991-04-09 SG SG1996006208A patent/SG46584A1/en unknown
- 1991-04-09 JP JP91506876A patent/JPH05506217A/ja active Pending
- 1991-04-09 AT AT91907396T patent/ATE144138T1/de not_active IP Right Cessation
- 1991-04-09 DK DK91907396.5T patent/DK0524989T3/da active
- 1991-04-09 DE DE69122751T patent/DE69122751T2/de not_active Expired - Fee Related
- 1991-04-09 RU RU92016377A patent/RU2111743C1/ru active
- 1991-04-09 ES ES91907396T patent/ES2093097T3/es not_active Expired - Lifetime
- 1991-04-09 WO PCT/EP1991/000688 patent/WO1991016042A1/en not_active Ceased
- 1991-04-09 EP EP91907396A patent/EP0524989B1/en not_active Expired - Lifetime
- 1991-04-09 KR KR1019920702558A patent/KR100196256B1/ko not_active Expired - Fee Related
- 1991-04-15 CA CA002040471A patent/CA2040471A1/en not_active Abandoned
- 1991-04-15 NZ NZ237823A patent/NZ237823A/en unknown
- 1991-04-15 PT PT97370A patent/PT97370B/pt not_active IP Right Cessation
- 1991-04-15 ZA ZA912792A patent/ZA912792B/xx unknown
- 1991-04-16 TW TW080102920A patent/TW223022B/zh active
- 1991-04-16 IE IE127191A patent/IE911271A1/en unknown
-
1992
- 1992-11-06 US US07/972,660 patent/US5900252A/en not_active Expired - Fee Related
-
1996
- 1996-11-29 GR GR960403247T patent/GR3021847T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DE69122751D1 (de) | 1996-11-21 |
| IE911271A1 (en) | 1991-10-23 |
| NZ237823A (en) | 1992-09-25 |
| ATE144138T1 (de) | 1996-11-15 |
| ES2093097T3 (es) | 1996-12-16 |
| PT97370B (pt) | 1998-08-31 |
| EP0524989B1 (en) | 1996-10-16 |
| CA2035155A1 (en) | 1991-10-18 |
| TW223022B (https=) | 1994-05-01 |
| ZA912792B (en) | 1992-12-30 |
| JPH04224517A (ja) | 1992-08-13 |
| US5900252A (en) | 1999-05-04 |
| IT9020054A0 (it) | 1990-04-17 |
| DE69122751T2 (de) | 1997-02-13 |
| PT97370A (pt) | 1992-01-31 |
| EP0453001A1 (en) | 1991-10-23 |
| CA2040471A1 (en) | 1991-10-18 |
| GR3021847T3 (en) | 1997-02-28 |
| IT1246382B (it) | 1994-11-18 |
| RU2111743C1 (ru) | 1998-05-27 |
| AU654277B2 (en) | 1994-11-03 |
| DK0524989T3 (da) | 1996-11-18 |
| EP0524989A1 (en) | 1993-02-03 |
| KR930700077A (ko) | 1993-03-13 |
| WO1991016042A1 (en) | 1991-10-31 |
| AU7679891A (en) | 1991-11-11 |
| JPH05506217A (ja) | 1993-09-16 |
| IT9020054A1 (https=) | 1991-10-17 |
| JP3194974B2 (ja) | 2001-08-06 |
| SG46584A1 (en) | 1998-02-20 |
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