JPWO2020141460A5 - - Google Patents
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- JPWO2020141460A5 JPWO2020141460A5 JP2021538388A JP2021538388A JPWO2020141460A5 JP WO2020141460 A5 JPWO2020141460 A5 JP WO2020141460A5 JP 2021538388 A JP2021538388 A JP 2021538388A JP 2021538388 A JP2021538388 A JP 2021538388A JP WO2020141460 A5 JPWO2020141460 A5 JP WO2020141460A5
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- JP
- Japan
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- integer
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- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024178728A JP2025020144A (ja) | 2019-01-03 | 2024-10-11 | 切断可能なリンカーを含む化合物及びその使用 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962788039P | 2019-01-03 | 2019-01-03 | |
| US62/788,039 | 2019-01-03 | ||
| PCT/IB2020/000019 WO2020141460A2 (en) | 2019-01-03 | 2020-01-02 | Compounds comprising cleavable linker and uses thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024178728A Division JP2025020144A (ja) | 2019-01-03 | 2024-10-11 | 切断可能なリンカーを含む化合物及びその使用 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2022515885A JP2022515885A (ja) | 2022-02-22 |
| JPWO2020141460A5 true JPWO2020141460A5 (https=) | 2023-01-19 |
| JP2022515885A5 JP2022515885A5 (https=) | 2023-01-19 |
| JP7657153B2 JP7657153B2 (ja) | 2025-04-04 |
Family
ID=71407384
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021538388A Active JP7657153B2 (ja) | 2019-01-03 | 2020-01-02 | 切断可能なリンカーを含む化合物及びその使用 |
| JP2024178728A Withdrawn JP2025020144A (ja) | 2019-01-03 | 2024-10-11 | 切断可能なリンカーを含む化合物及びその使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024178728A Withdrawn JP2025020144A (ja) | 2019-01-03 | 2024-10-11 | 切断可能なリンカーを含む化合物及びその使用 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US12551570B2 (https=) |
| EP (1) | EP3906063A4 (https=) |
| JP (2) | JP7657153B2 (https=) |
| KR (1) | KR20210099658A (https=) |
| CN (2) | CN114306635A (https=) |
| EA (1) | EA202191855A1 (https=) |
| WO (1) | WO2020141460A2 (https=) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2019008441A1 (en) | 2017-07-04 | 2019-01-10 | Intocell, Inc. | COMPOUNDS COMPRISING A CLIABABLE BIT AND USES THEREOF |
| WO2020141460A2 (en) | 2019-01-03 | 2020-07-09 | Intocell, Inc. | Compounds comprising cleavable linker and uses thereof |
| IL322315A (en) | 2019-05-14 | 2025-09-01 | Provention Bio Inc | Methods and preparations for preventing type 1 diabetes |
| AU2021287998B2 (en) | 2020-06-11 | 2026-03-12 | Benaroya Research Institute At Virginia Mason | Methods and compositions for preventing type 1 diabetes |
| US12565529B2 (en) | 2021-05-24 | 2026-03-03 | Provention Bio, Inc. | Methods for treating type 1 diabetes |
| CN114874287B (zh) * | 2022-05-20 | 2024-04-02 | 联宁（苏州）生物制药有限公司 | 一种抗体偶联药物-连接子lnd1042的合成方法 |
| WO2025252011A1 (zh) * | 2024-06-03 | 2025-12-11 | 杭州多域生物技术有限公司 | 含Sulfoximine连接子的降解剂及其中间体和应用 |
| CN119462688B (zh) * | 2024-11-08 | 2026-03-10 | 青岛大学 | 一种生物素化氨基酸衍生物的制备方法 |
| CN121494812A (zh) * | 2026-01-14 | 2026-02-10 | 西南林业大学 | 一种基于肉桂酸衍生物的n2h4比率型荧光探针及其合成方法和应用 |
Family Cites Families (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1182232B (de) | 1963-03-08 | 1964-11-26 | Hans J Zimmer Verfahrenstechni | Verfahren zur Herstellung von Trialkylaryloxysilanen |
| CH565791A5 (https=) | 1972-07-11 | 1975-08-29 | Sandoz Ag | |
| US4540828A (en) | 1982-06-01 | 1985-09-10 | Vista Chemical Company | Catalysts for alkoxylation reactions |
| JPS5978171A (ja) | 1982-10-26 | 1984-05-04 | Ikeda Mohandou:Kk | 複素環式化合物 |
| DE3632329A1 (de) | 1986-09-24 | 1988-03-31 | Bayer Ag | Substituierte phenylsulfonamide |
| JP3041736B2 (ja) * | 1991-11-01 | 2000-05-15 | コニカ株式会社 | ハロゲン化銀写真感光材料 |
| JP3061862B2 (ja) | 1994-10-14 | 2000-07-10 | 山之内製薬株式会社 | アゾール誘導体 |
| JP2005291974A (ja) | 2004-03-31 | 2005-10-20 | Kyocera Chemical Corp | フェルダジル基を有する磁性有機粒子、粒子固定方法及びマイクロアレイ |
| EP1867729A1 (en) | 2006-06-14 | 2007-12-19 | Libragen | Water soluble phenolics derivatives with dermocosmetic and therapeutic applications |
| MY168297A (en) | 2011-11-17 | 2018-10-23 | Pfizer | Cytotoxic Peptides and Antibody Drug Conjugates Thereof |
| TWI585115B (zh) | 2011-12-15 | 2017-06-01 | 普利司通股份有限公司 | 經穩定之多價陰離子聚合反應引發劑及其製備方法 |
| PL2872157T3 (pl) | 2012-07-12 | 2020-07-13 | Hangzhou Dac Biotech Co., Ltd | Koniugaty wiążących komórkę cząsteczek ze środkami cytotoksycznymi |
| JP6255038B2 (ja) | 2013-02-26 | 2017-12-27 | トリアクト セラピューティクス，インク． | 癌治療 |
| US9499528B2 (en) | 2013-04-08 | 2016-11-22 | The University Of Akron | Class of near infrared molecular probes for biological applications |
| CN105899539B (zh) * | 2014-01-10 | 2021-11-09 | 博笛生物科技有限公司 | 用于免疫疗法的化合物和组合物 |
| KR101628872B1 (ko) * | 2014-05-28 | 2016-06-09 | 주식회사 레고켐 바이오사이언스 | 자가-희생 기를 포함하는 화합물 |
| WO2016029324A1 (en) | 2014-08-29 | 2016-03-03 | Rsem, Limited Partnership | Azasulfurylpeptide-based cd36 modulators and uses thereof |
| US10035526B2 (en) | 2014-12-03 | 2018-07-31 | New York Air Brake, LLC | Brake piston assembly |
| WO2016118770A1 (en) | 2015-01-21 | 2016-07-28 | The Regents Of The University Of California | Affinity-assisted protein modification and recycling |
| CN107922375B (zh) | 2015-07-30 | 2020-05-22 | 正大天晴药业集团股份有限公司 | 靶向idh2突变的抗肿瘤化合物及其使用方法 |
| WO2017044043A1 (en) | 2015-09-09 | 2017-03-16 | Agency For Science, Technology And Research | Process for direct amidation of amines via rh(i)-catalyzed addition of boroxines |
| KR101766822B1 (ko) | 2015-09-10 | 2017-08-24 | 서울대학교산학협력단 | 디페닐설페이트 유도체 또는 이의 약학적으로 허용가능한 염, 이의 제조방법 및 이를 유효성분으로 포함하는 c형 간염 바이러스 관련 질환의 예방 또는 치료용 약학적 조성물 |
| KR102847350B1 (ko) | 2015-11-25 | 2025-08-19 | 주식회사 리가켐바이오사이언스 | 분지된 링커를 포함하는 항체-약물 접합체 및 이의 제조방법 |
| WO2018053552A2 (en) | 2016-09-19 | 2018-03-22 | Cellerant Therapeutics, Inc. | Isoquinolidinobenzodiazepines |
| WO2018124758A2 (ko) * | 2016-12-28 | 2018-07-05 | 주식회사 인투셀 | 베타-갈락토사이드가 도입된 자가-희생 기를 포함하는 화합물 |
| WO2019008441A1 (en) | 2017-07-04 | 2019-01-10 | Intocell, Inc. | COMPOUNDS COMPRISING A CLIABABLE BIT AND USES THEREOF |
| MX2020012718A (es) | 2018-05-29 | 2021-02-16 | Intocell Inc | Derivados de benzodiazepinas novedosos y usos de los mismos. |
| KR20210068591A (ko) | 2018-10-31 | 2021-06-09 | 주식회사 인투셀 | 융합된 헤테로시클릭 벤조디아제핀 유도체 및 그의 용도 |
| WO2020141460A2 (en) | 2019-01-03 | 2020-07-09 | Intocell, Inc. | Compounds comprising cleavable linker and uses thereof |
| EP3906064A4 (en) | 2019-01-03 | 2023-03-08 | Intocell, Inc. | CLEAVABLE LINKER COMPOUNDS AND USES THEREOF |
-
2020
- 2020-01-02 WO PCT/IB2020/000019 patent/WO2020141460A2/en not_active Ceased
- 2020-01-02 KR KR1020217024209A patent/KR20210099658A/ko not_active Ceased
- 2020-01-02 CN CN202111628316.1A patent/CN114306635A/zh active Pending
- 2020-01-02 EA EA202191855A patent/EA202191855A1/ru unknown
- 2020-01-02 EP EP20735849.0A patent/EP3906063A4/en active Pending
- 2020-01-02 US US17/419,435 patent/US12551570B2/en active Active
- 2020-01-02 CN CN202080007805.2A patent/CN113423431A/zh active Pending
- 2020-01-02 JP JP2021538388A patent/JP7657153B2/ja active Active
-
2024
- 2024-10-11 JP JP2024178728A patent/JP2025020144A/ja not_active Withdrawn
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