JP6611816B2 - ３−オキソ−３−（アリールアミノ）プロパノエイト、その製造方法、およびピロリジノンの製造におけるその使用 - Google Patents
３−オキソ−３−（アリールアミノ）プロパノエイト、その製造方法、およびピロリジノンの製造におけるその使用 Download PDFInfo
- Publication number
- JP6611816B2 JP6611816B2 JP2017548361A JP2017548361A JP6611816B2 JP 6611816 B2 JP6611816 B2 JP 6611816B2 JP 2017548361 A JP2017548361 A JP 2017548361A JP 2017548361 A JP2017548361 A JP 2017548361A JP 6611816 B2 JP6611816 B2 JP 6611816B2
- Authority
- JP
- Japan
- Prior art keywords
- group
- ring
- independently
- halogen atom
- haloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Links
- 0 **C(C(C(CC1=C)O)C1=O)=O Chemical compound **C(C(C(CC1=C)O)C1=O)=O 0.000 description 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/02—Esters of acyclic saturated monocarboxylic acids having the carboxyl group bound to an acyclic carbon atom or to hydrogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B31/00—Reduction in general
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/02—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
- C07C233/04—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with carbon atoms of carboxamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C233/07—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with carbon atoms of carboxamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/12—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups
- C07C233/15—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by halogen atoms or by nitro or nitroso groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
- C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
- C07D207/27—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
- C07D207/273—2-Pyrrolidones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
- C07D207/277—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462088971P | 2014-12-08 | 2014-12-08 | |
| US62/088,971 | 2014-12-08 | ||
| PCT/US2015/063101 WO2016094117A1 (en) | 2014-12-08 | 2015-12-01 | 3-oxo-3-(arylamino)propanoates, a process for their preparation, and their use in preparing pyrrolidinones |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017538785A JP2017538785A (ja) | 2017-12-28 |
| JP2017538785A5 JP2017538785A5 (cg-RX-API-DMAC7.html) | 2019-01-17 |
| JP6611816B2 true JP6611816B2 (ja) | 2019-11-27 |
Family
ID=54782892
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017548361A Active JP6611816B2 (ja) | 2014-12-08 | 2015-12-01 | ３−オキソ−３−（アリールアミノ）プロパノエイト、その製造方法、およびピロリジノンの製造におけるその使用 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US10227286B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP3230264B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP6611816B2 (cg-RX-API-DMAC7.html) |
| KR (1) | KR102542215B1 (cg-RX-API-DMAC7.html) |
| CN (1) | CN107001260B (cg-RX-API-DMAC7.html) |
| AR (1) | AR102939A1 (cg-RX-API-DMAC7.html) |
| AU (1) | AU2015361018B2 (cg-RX-API-DMAC7.html) |
| BR (1) | BR112017009701B1 (cg-RX-API-DMAC7.html) |
| ES (1) | ES2759267T3 (cg-RX-API-DMAC7.html) |
| HU (1) | HUE047582T2 (cg-RX-API-DMAC7.html) |
| IL (1) | IL252637A (cg-RX-API-DMAC7.html) |
| MX (1) | MX382656B (cg-RX-API-DMAC7.html) |
| PL (1) | PL3230264T3 (cg-RX-API-DMAC7.html) |
| RU (1) | RU2712831C2 (cg-RX-API-DMAC7.html) |
| SG (1) | SG11201702924WA (cg-RX-API-DMAC7.html) |
| TW (1) | TWI694982B (cg-RX-API-DMAC7.html) |
| WO (1) | WO2016094117A1 (cg-RX-API-DMAC7.html) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY195078A (en) | 2013-12-03 | 2023-01-09 | Fmc Corp | Pyrrolidinones As Herbicides |
| US11589583B2 (en) | 2013-12-03 | 2023-02-28 | Fmc Corporation | Pyrrolidinones herbicides |
| BR112016030930B1 (pt) | 2014-07-02 | 2022-03-15 | Fmc Corporation | Compostos, composições herbicidas, mistura herbicida e método para controle do crescimento de vegetação indesejável |
| AU2016246410B2 (en) | 2015-04-10 | 2020-11-05 | Fmc Corporation | Substituted cyclic amides as herbicides |
| AU2016254958B2 (en) | 2015-04-27 | 2020-04-23 | Fmc Corporation | Butyrolactones as herbicides |
| JP7000160B2 (ja) | 2015-05-12 | 2022-01-19 | エフ エム シー コーポレーション | 除草剤としてのアリール置換二環式化合物 |
| CN107690426B (zh) | 2015-05-29 | 2021-07-06 | Fmc公司 | 作为除草剂的取代的环酰胺 |
| EP3303321A1 (en) * | 2015-06-02 | 2018-04-11 | E. I. du Pont de Nemours and Company | Substituted cyclic amides and their use as herbicides |
| BR112018001964B1 (pt) | 2015-07-31 | 2022-05-10 | Fmc Corporation | Composto, composição herbicida, mistura herbicida e método para o controle docrescimento de vegetação indesejada |
| GB201617050D0 (en) | 2016-10-07 | 2016-11-23 | Syngenta Participations Ag | Herbicidal mixtures |
| EP3558962B1 (en) | 2016-12-21 | 2023-07-12 | FMC Corporation | Nitrone herbicides |
| KR102774623B1 (ko) | 2017-03-21 | 2025-03-05 | 에프엠씨 코포레이션 | 피롤리디논 및 이의 제조 방법 |
| MX2019011090A (es) | 2017-03-21 | 2019-11-18 | Fmc Corp | Mezcla herbicida, composición y método. |
| WO2018177837A1 (de) | 2017-03-30 | 2018-10-04 | Bayer Aktiengesellschaft | 4-cyclopentyl- und 4-cyclopropyl-2-oxopyrrolidin-3-carboxami d-derivate und verwandte verbindungen als herbizide pflanzenschutzmittel |
| WO2018177836A1 (de) | 2017-03-30 | 2018-10-04 | Bayer Aktiengesellschaft | N-cyclopropyl-2-oxopyrrolidin-3-carboxamid-derivate und verwandte verbindungen als herbizide pflanzenschutzmittel |
| AR111967A1 (es) | 2017-05-30 | 2019-09-04 | Fmc Corp | Amidas herbicidas |
| AR111839A1 (es) | 2017-05-30 | 2019-08-21 | Fmc Corp | Lactamas 3-sustituidas herbicidas |
| WO2019025156A1 (de) | 2017-08-03 | 2019-02-07 | Bayer Aktiengesellschaft | Substituierte pyrrolidinone sowie deren salze und ihre verwendung als herbizide wirkstoffe |
| GB201819747D0 (en) | 2018-12-04 | 2019-01-16 | Syngenta Participations Ag | Herbicidal compositions |
| US20220125052A1 (en) | 2019-02-15 | 2022-04-28 | Syngenta Crop Protection Ag | Herbicidal Compositions |
| US20250066297A1 (en) | 2021-12-15 | 2025-02-27 | Adama Agan Ltd. | Compounds useful for the preparation of various agrochemicals and markers thereof |
Family Cites Families (42)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1262277B (de) | 1962-12-05 | 1968-03-07 | Basf Ag | Verfahren zur Herstellung von Pyrrolidonen |
| US3741989A (en) | 1970-10-27 | 1973-06-26 | Abbott Lab | Lactonic acetals |
| JPS5356288A (en) | 1976-10-30 | 1978-05-22 | Matsushita Electric Works Ltd | Preparation of phenolic resin |
| JPS5488114A (en) | 1977-12-26 | 1979-07-13 | Fuji Photo Film Co Ltd | Manufacturing device for photograph seal |
| US4594094A (en) | 1983-04-04 | 1986-06-10 | Shell Oil Company | Oxacycloalkane-alpha-(thio)carboxylic acid derivatives and use as plant growth regulators and herbicides |
| US4874422A (en) * | 1988-12-27 | 1989-10-17 | Ici Americas Inc. | 1-Phenyl-3-carboxyamidopyrrolidones and their use as herbicides |
| JP3487669B2 (ja) | 1995-03-28 | 2004-01-19 | 積水化学工業株式会社 | 不飽和ポリエステル樹脂組成物 |
| WO2000009481A1 (en) | 1998-08-11 | 2000-02-24 | Takeda Chemical Industries, Ltd. | Cyclic amide compounds, process for producing the same, intermediates thereof and herbicides |
| AU2002340971B2 (en) | 2001-10-08 | 2007-04-26 | Ucb | Use of 2-oxo-1-pyrrolidine derivatives for the treatment of dyskinesia and movement disorders |
| KR20050038631A (ko) | 2002-08-23 | 2005-04-27 | 카이론 코포레이션 | 글리코겐 신타제 키나제 3의 피롤 기제 억제제 |
| CA2502478A1 (en) * | 2002-10-18 | 2004-05-06 | Basf Aktiengesellschaft | 1-phenylpyrrolidine-2-one-3-carboxamides |
| AU2003277721A1 (en) | 2002-11-15 | 2004-06-15 | In Kwon Chung | Beta-nitrostyrene compound and telomerase inhibitor having an anticancer activity |
| US7205318B2 (en) | 2003-03-18 | 2007-04-17 | Bristol-Myers Squibb Company | Lactam-containing cyclic diamines and derivatives as a factor Xa inhibitors |
| WO2006081562A2 (en) | 2005-01-28 | 2006-08-03 | Irm Llc | Synthesis of aryl pyrrolidones |
| US20070123508A1 (en) | 2005-05-27 | 2007-05-31 | Roger Olsson | PAR2-modulating compounds and their use |
| WO2007066828A1 (ja) | 2005-12-09 | 2007-06-14 | Sumitomo Chemical Company, Limited | 光学活性な４－アミノ－３－置換フェニルブタン酸の製造方法 |
| ES2304220B1 (es) | 2007-03-02 | 2009-09-11 | Universidad De Zaragoza | Composicion para el tratamiento de enfermedades infecciosas. |
| EP2065380A1 (en) | 2007-08-22 | 2009-06-03 | F.Hoffmann-La Roche Ag | Pyridoneamide derivatives as focal adhesion kinase (FAK) inhibitors and their use for the treatment of cancer |
| CN101412711A (zh) | 2007-10-15 | 2009-04-22 | 上海恒瑞医药有限公司 | 氨基甲酸酯类衍生物及其在医药上的应用 |
| CN102137841B (zh) | 2008-09-02 | 2014-05-14 | 日产化学工业株式会社 | 邻位取代卤代烷基磺酰苯胺衍生物及除草剂 |
| JPWO2010053165A1 (ja) | 2008-11-04 | 2012-04-05 | 帝人ファーマ株式会社 | ビタミンｄ３ラクタム誘導体 |
| KR20110117194A (ko) * | 2009-02-23 | 2011-10-26 | 에프. 호프만-라 로슈 아게 | 암 치료를 위한 신규한 오르토-아미노아미드 |
| CN101747252A (zh) * | 2009-12-28 | 2010-06-23 | 嘉兴宜博生物医药科技有限公司 | R构诺普利兰的合成方法 |
| JP5788496B2 (ja) | 2010-08-10 | 2015-09-30 | 武田薬品工業株式会社 | 複素環化合物およびその用途 |
| US8946216B2 (en) | 2010-09-01 | 2015-02-03 | Merck Sharp & Dohme Corp. | Indazole derivatives useful as ERK inhibitors |
| BR112013029201B1 (pt) | 2011-05-13 | 2022-08-09 | Array Biopharma Inc | Compostos de pirrolidinil ureia e pirrolidinil tioureia, seu processo de preparação, seu uso e composições farmacêuticas |
| CN102531918B (zh) | 2012-01-18 | 2013-10-02 | 安阳工学院 | 一种对映纯对称反式二烷基环己胺的合成方法 |
| KR20130142477A (ko) | 2012-06-19 | 2013-12-30 | 순천향대학교 산학협력단 | 키랄 나이트로사이클로프로판 유도체의 제조방법 |
| US20160137639A1 (en) | 2012-10-26 | 2016-05-19 | Japan Tobacco Inc. | Triazole-isoxazole compound and medical use thereof |
| MY195078A (en) | 2013-12-03 | 2023-01-09 | Fmc Corp | Pyrrolidinones As Herbicides |
| GB201321743D0 (en) | 2013-12-09 | 2014-01-22 | Ucb Pharma Sa | Therapeutic agents |
| RU2555370C1 (ru) | 2014-02-12 | 2015-07-10 | Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Самарский государственный технический университет" | Способ энантиоселективного синтеза диэтил[3-метил-(1s)-(нитрометил)бутил]малоната формулы i |
| BR112016030930B1 (pt) | 2014-07-02 | 2022-03-15 | Fmc Corporation | Compostos, composições herbicidas, mistura herbicida e método para controle do crescimento de vegetação indesejável |
| AU2016246410B2 (en) | 2015-04-10 | 2020-11-05 | Fmc Corporation | Substituted cyclic amides as herbicides |
| AU2016254958B2 (en) | 2015-04-27 | 2020-04-23 | Fmc Corporation | Butyrolactones as herbicides |
| JP7000160B2 (ja) | 2015-05-12 | 2022-01-19 | エフ エム シー コーポレーション | 除草剤としてのアリール置換二環式化合物 |
| CN107690426B (zh) | 2015-05-29 | 2021-07-06 | Fmc公司 | 作为除草剂的取代的环酰胺 |
| EP3303321A1 (en) * | 2015-06-02 | 2018-04-11 | E. I. du Pont de Nemours and Company | Substituted cyclic amides and their use as herbicides |
| BR112018001964B1 (pt) | 2015-07-31 | 2022-05-10 | Fmc Corporation | Composto, composição herbicida, mistura herbicida e método para o controle docrescimento de vegetação indesejada |
| EP3558962B1 (en) | 2016-12-21 | 2023-07-12 | FMC Corporation | Nitrone herbicides |
| MX2019011090A (es) | 2017-03-21 | 2019-11-18 | Fmc Corp | Mezcla herbicida, composición y método. |
| KR102774623B1 (ko) | 2017-03-21 | 2025-03-05 | 에프엠씨 코포레이션 | 피롤리디논 및 이의 제조 방법 |
-
2015
- 2015-12-01 WO PCT/US2015/063101 patent/WO2016094117A1/en not_active Ceased
- 2015-12-01 BR BR112017009701-0A patent/BR112017009701B1/pt active IP Right Grant
- 2015-12-01 PL PL15805092T patent/PL3230264T3/pl unknown
- 2015-12-01 AU AU2015361018A patent/AU2015361018B2/en active Active
- 2015-12-01 HU HUE15805092A patent/HUE047582T2/hu unknown
- 2015-12-01 CN CN201580065080.1A patent/CN107001260B/zh active Active
- 2015-12-01 SG SG11201702924WA patent/SG11201702924WA/en unknown
- 2015-12-01 EP EP15805092.2A patent/EP3230264B1/en active Active
- 2015-12-01 MX MX2017007087A patent/MX382656B/es unknown
- 2015-12-01 JP JP2017548361A patent/JP6611816B2/ja active Active
- 2015-12-01 RU RU2017123114A patent/RU2712831C2/ru active
- 2015-12-01 US US15/533,448 patent/US10227286B2/en active Active
- 2015-12-01 KR KR1020177018406A patent/KR102542215B1/ko active Active
- 2015-12-01 ES ES15805092T patent/ES2759267T3/es active Active
- 2015-12-04 AR ARP150103996A patent/AR102939A1/es active IP Right Grant
- 2015-12-04 TW TW104140692A patent/TWI694982B/zh active
-
2017
- 2017-06-04 IL IL252637A patent/IL252637A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| CN107001260B (zh) | 2020-11-10 |
| PL3230264T3 (pl) | 2020-03-31 |
| WO2016094117A1 (en) | 2016-06-16 |
| TWI694982B (zh) | 2020-06-01 |
| MX382656B (es) | 2025-03-13 |
| JP2017538785A (ja) | 2017-12-28 |
| ES2759267T3 (es) | 2020-05-08 |
| BR112017009701A2 (pt) | 2018-02-20 |
| EP3230264A1 (en) | 2017-10-18 |
| US10227286B2 (en) | 2019-03-12 |
| AU2015361018A1 (en) | 2017-04-27 |
| HUE047582T2 (hu) | 2020-05-28 |
| RU2712831C2 (ru) | 2020-02-03 |
| EP3230264B1 (en) | 2019-09-11 |
| RU2017123114A (ru) | 2019-01-11 |
| AU2015361018B2 (en) | 2020-01-16 |
| SG11201702924WA (en) | 2017-05-30 |
| IL252637A (en) | 2017-11-30 |
| BR112017009701B1 (pt) | 2021-09-08 |
| KR20170090491A (ko) | 2017-08-07 |
| IL252637A0 (en) | 2017-07-31 |
| US20180057442A1 (en) | 2018-03-01 |
| CN107001260A (zh) | 2017-08-01 |
| KR102542215B1 (ko) | 2023-06-12 |
| TW201632497A (zh) | 2016-09-16 |
| AR102939A1 (es) | 2017-04-05 |
| RU2017123114A3 (cg-RX-API-DMAC7.html) | 2019-07-17 |
| MX2017007087A (es) | 2017-09-05 |
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