JP6008849B2 - 置換β−シクロデキストリンにより安定化されたポサコナゾール静脈注射用溶液製剤 - Google Patents

置換β−シクロデキストリンにより安定化されたポサコナゾール静脈注射用溶液製剤 Download PDF

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JP6008849B2
JP6008849B2 JP2013518498A JP2013518498A JP6008849B2 JP 6008849 B2 JP6008849 B2 JP 6008849B2 JP 2013518498 A JP2013518498 A JP 2013518498A JP 2013518498 A JP2013518498 A JP 2013518498A JP 6008849 B2 JP6008849 B2 JP 6008849B2
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pharmaceutical composition
composition according
posaconazole
infection
invasive
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JP2013535422A (ja
JP2013535422A5 (enExample
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ヘイムベシヤー，スーザン・ケイ
モンテイース，デイビツド
ピプキン，ジエイムズ・デイ
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Merck and Co Inc
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Merck and Co Inc
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/40—Cyclodextrins; Derivatives thereof
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2013518498A 2010-06-29 2011-06-24 置換β−シクロデキストリンにより安定化されたポサコナゾール静脈注射用溶液製剤 Active JP6008849B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US35970110P 2010-06-29 2010-06-29
US61/359,701 2010-06-29
PCT/US2011/041715 WO2012005973A1 (en) 2010-06-29 2011-06-24 Posaconazole intravenous solution formulations stabilized by substituted beta-cyclodextrin

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JP2013535422A JP2013535422A (ja) 2013-09-12
JP2013535422A5 JP2013535422A5 (enExample) 2014-07-17
JP6008849B2 true JP6008849B2 (ja) 2016-10-19

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US (2) US9023790B2 (enExample)
EP (3) EP2588116A4 (enExample)
JP (1) JP6008849B2 (enExample)
KR (1) KR101834024B1 (enExample)
CN (2) CN102958528A (enExample)
AU (1) AU2011276680B2 (enExample)
BR (1) BR112012033077B8 (enExample)
CA (1) CA2802929C (enExample)
CY (1) CY1124690T1 (enExample)
DK (1) DK3391890T3 (enExample)
ES (1) ES2893444T3 (enExample)
HR (1) HRP20211686T1 (enExample)
HU (1) HUE056581T2 (enExample)
LT (1) LT3391890T (enExample)
MX (2) MX338685B (enExample)
PL (1) PL3391890T3 (enExample)
PT (1) PT3391890T (enExample)
RS (1) RS62583B1 (enExample)
SI (1) SI3391890T1 (enExample)
WO (1) WO2012005973A1 (enExample)

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CN110022857A (zh) 2016-11-18 2019-07-16 艾库里斯抗感染治疗有限公司 基于改性环糊精和酸化剂的脒取代β-内酰胺化合物的新制剂、其制备及作为抗微生物药物组合物的用途
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CN110711174A (zh) * 2018-07-11 2020-01-21 郑州泰丰制药有限公司 一种泊沙康唑注射液中间体溶液配制方法
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CN115038723A (zh) 2019-11-18 2022-09-09 锡德克斯药物公司 烷基化环糊精组合物及其制备和使用方法
WO2021245703A2 (en) * 2020-06-06 2021-12-09 Inventia Healthcare Limited Stable liquid compositions of posaconazole
US12698348B2 (en) 2020-09-24 2026-08-04 Cydex Pharmaceuticals, Inc. Alkylated cyclodextrin compositions and processes for preparing and using the same
CN115429748A (zh) * 2021-06-02 2022-12-06 江苏奥赛康药业有限公司 一种泊沙康唑注射液的制备方法
WO2023148763A1 (en) * 2022-02-01 2023-08-10 Cipla Limited Injectable pharmaceutical compositions of azole antifungal agents
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BR112012033077B1 (pt) 2020-01-21
RU2013103724A (ru) 2014-08-10
US9358297B2 (en) 2016-06-07
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ES2893444T3 (es) 2022-02-09
WO2012005973A1 (en) 2012-01-12
CN102958528A (zh) 2013-03-06
SI3391890T1 (sl) 2021-11-30
PT3391890T (pt) 2021-10-14
EP3391890B1 (en) 2021-08-25
CA2802929A1 (en) 2012-01-12
EP2588116A1 (en) 2013-05-08
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RS62583B1 (sr) 2021-12-31
US20150265715A1 (en) 2015-09-24
MX346901B (es) 2017-04-04
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BR112012033077A2 (pt) 2016-11-22
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