JP4164125B2 - Ｌｈｒｈ拮抗物質ペプチド - Google Patents

Ｌｈｒｈ拮抗物質ペプチド Download PDF

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Publication number
JP4164125B2
JP4164125B2 JP50205097A JP50205097A JP4164125B2 JP 4164125 B2 JP4164125 B2 JP 4164125B2 JP 50205097 A JP50205097 A JP 50205097A JP 50205097 A JP50205097 A JP 50205097A JP 4164125 B2 JP4164125 B2 JP 4164125B2
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Prior art keywords
lhrh
peptide
lys
component
pal
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Japanese (ja)
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JPH11507374A (ja
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ダブリュー． レスキ，ロジャー
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アドバンスド リサーチ アンド テクノロジー インスティテュート
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/13—Luteinizing hormone-releasing hormone; related peptides
JP50205097A 1995-06-07 1996-06-07 Ｌｈｒｈ拮抗物質ペプチド Expired - Fee Related JP4164125B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/480,494 US5843901A (en) 1995-06-07 1995-06-07 LHRH antagonist peptides
US08/480,494 1995-06-07
PCT/US1996/009852 WO1996040757A2 (en) 1995-06-07 1996-06-07 Lhrh antagonist peptides

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2007211155A Division JP2007302695A (ja) 1995-06-07 2007-08-13 Ｌｈｒｈ拮抗物質ペプチド

Publications (2)

Publication Number Publication Date
JPH11507374A JPH11507374A (ja) 1999-06-29
JP4164125B2 true JP4164125B2 (ja) 2008-10-08

Family

ID=23908180

Family Applications (3)

Application Number Title Priority Date Filing Date
JP50205097A Expired - Fee Related JP4164125B2 (ja) 1995-06-07 1996-06-07 Ｌｈｒｈ拮抗物質ペプチド
JP2007211155A Withdrawn JP2007302695A (ja) 1995-06-07 2007-08-13 Ｌｈｒｈ拮抗物質ペプチド
JP2008263288A Withdrawn JP2009040793A (ja) 1995-06-07 2008-10-09 Ｌｈｒｈ拮抗物質ペプチド

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2007211155A Withdrawn JP2007302695A (ja) 1995-06-07 2007-08-13 Ｌｈｒｈ拮抗物質ペプチド
JP2008263288A Withdrawn JP2009040793A (ja) 1995-06-07 2008-10-09 Ｌｈｒｈ拮抗物質ペプチド

Country Status (13)

Country Link
US (4) US5843901A (US07071165-20060704-C00014.png)
EP (2) EP0794961B1 (US07071165-20060704-C00014.png)
JP (3) JP4164125B2 (US07071165-20060704-C00014.png)
AT (2) ATE432941T1 (US07071165-20060704-C00014.png)
AU (1) AU715399B2 (US07071165-20060704-C00014.png)
CA (1) CA2219460C (US07071165-20060704-C00014.png)
DE (4) DE69623254T2 (US07071165-20060704-C00014.png)
DK (2) DK1188768T3 (US07071165-20060704-C00014.png)
ES (2) ES2326861T3 (US07071165-20060704-C00014.png)
HK (1) HK1045161B (US07071165-20060704-C00014.png)
LU (2) LU91225I2 (US07071165-20060704-C00014.png)
PT (2) PT1188768E (US07071165-20060704-C00014.png)
WO (1) WO1996040757A2 (US07071165-20060704-C00014.png)

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DK0794961T3 (da) 2002-10-21
EP0794961B1 (en) 2002-08-28
DE69623254D1 (de) 2002-10-02
DE69623254T2 (de) 2002-12-19
EP1188768A2 (en) 2002-03-20
ATE432941T1 (de) 2009-06-15
CA2219460C (en) 2009-04-14
EP1188768B1 (en) 2009-06-03
ES2177789T3 (es) 2002-12-16
CA2219460A1 (en) 1996-12-19
US20030181385A1 (en) 2003-09-25
US20020115615A1 (en) 2002-08-22
US7071165B2 (en) 2006-07-04
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AU6168096A (en) 1996-12-30
ES2326861T3 (es) 2009-10-21
US6423686B1 (en) 2002-07-23
LU91225I2 (fr) 2006-05-03
AU715399B2 (en) 2000-02-03
US5843901A (en) 1998-12-01
US20030040482A1 (en) 2003-02-27
DE122006000012I2 (de) 2010-02-04
ATE222924T1 (de) 2002-09-15
WO1996040757A3 (en) 1997-02-20
DK1188768T3 (da) 2009-09-21
EP1188768A3 (en) 2002-10-23
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HK1045161B (zh) 2009-12-24
DE69535963D1 (de) 2009-07-16
DE122006000012I1 (de) 2006-06-29
EP0794961A2 (en) 1997-09-17
WO1996040757A2 (en) 1996-12-19
PT794961E (pt) 2003-01-31
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LU91857I2 (fr) 2011-10-24

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