DE122006000012I1 - Lhrh antagonistische Peptide - Google Patents
Lhrh antagonistische PeptideInfo
- Publication number
- DE122006000012I1 DE122006000012I1 DE1996623254 DE69623254C DE122006000012I1 DE 122006000012 I1 DE122006000012 I1 DE 122006000012I1 DE 1996623254 DE1996623254 DE 1996623254 DE 69623254 C DE69623254 C DE 69623254C DE 122006000012 I1 DE122006000012 I1 DE 122006000012I1
- Authority
- DE
- Germany
- Prior art keywords
- moiety
- longer
- peptide compound
- antagonistic peptides
- lhrh
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S930/00—Peptide or protein sequence
- Y10S930/01—Peptide or protein sequence
- Y10S930/13—Luteinizing hormone-releasing hormone; related peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Endocrinology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Reproductive Health (AREA)
- Immunology (AREA)
- Molecular Biology (AREA)
- Diabetes (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Gynecology & Obstetrics (AREA)
- Urology & Nephrology (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/480,494 US5843901A (en) | 1995-06-07 | 1995-06-07 | LHRH antagonist peptides |
PCT/US1996/009852 WO1996040757A2 (en) | 1995-06-07 | 1996-06-07 | Lhrh antagonist peptides |
Publications (1)
Publication Number | Publication Date |
---|---|
DE122006000012I1 true DE122006000012I1 (de) | 2006-06-29 |
Family
ID=23908180
Family Applications (4)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE1996623254 Pending DE122006000012I1 (de) | 1995-06-07 | 1996-06-07 | Lhrh antagonistische Peptide |
DE122006000012C Active DE122006000012I2 (de) | 1995-06-07 | 1996-06-07 | Lhrh antagonistische peptide |
DE69535963T Expired - Lifetime DE69535963D1 (de) | 1995-06-07 | 1996-06-07 | LHRH antagonistische Peptide |
DE69623254T Expired - Lifetime DE69623254T2 (de) | 1995-06-07 | 1996-06-07 | Lhrh antagonistische peptide |
Family Applications After (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE122006000012C Active DE122006000012I2 (de) | 1995-06-07 | 1996-06-07 | Lhrh antagonistische peptide |
DE69535963T Expired - Lifetime DE69535963D1 (de) | 1995-06-07 | 1996-06-07 | LHRH antagonistische Peptide |
DE69623254T Expired - Lifetime DE69623254T2 (de) | 1995-06-07 | 1996-06-07 | Lhrh antagonistische peptide |
Country Status (13)
Country | Link |
---|---|
US (4) | US5843901A (de) |
EP (2) | EP0794961B1 (de) |
JP (3) | JP4164125B2 (de) |
AT (2) | ATE432941T1 (de) |
AU (1) | AU715399B2 (de) |
CA (1) | CA2219460C (de) |
DE (4) | DE122006000012I1 (de) |
DK (2) | DK1188768T3 (de) |
ES (2) | ES2326861T3 (de) |
HK (1) | HK1045161B (de) |
LU (2) | LU91225I2 (de) |
PT (2) | PT1188768E (de) |
WO (1) | WO1996040757A2 (de) |
Families Citing this family (109)
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IL117175A (en) * | 1995-02-20 | 2005-11-20 | Sankyo Co | Osteoclastogenesis inhibitory factor protein |
US5843901A (en) * | 1995-06-07 | 1998-12-01 | Advanced Research & Technology Institute | LHRH antagonist peptides |
US5780435A (en) * | 1995-12-15 | 1998-07-14 | Praecis Pharmaceuticals Incorporated | Methods for treating prostate cancer with LHRH-R antagonists |
US5968895A (en) * | 1996-12-11 | 1999-10-19 | Praecis Pharmaceuticals, Inc. | Pharmaceutical formulations for sustained drug delivery |
AU713473B2 (en) | 1996-12-23 | 1999-12-02 | Immunex Corporation | Receptor activator of NF-kappa B, receptor is member of TNF receptor superfamily |
US5925730A (en) * | 1997-04-11 | 1999-07-20 | Ferring Bv | GnRH antagonists |
KR100496063B1 (ko) * | 1997-04-15 | 2005-06-21 | 산쿄 가부시키가이샤 | 신규단백질 및 그 제조방법 |
US6316408B1 (en) * | 1997-04-16 | 2001-11-13 | Amgen Inc. | Methods of use for osetoprotegerin binding protein receptors |
RO128635A2 (ro) | 1997-04-16 | 2013-07-30 | Amgen Inc. | Anticorp sau fragment al acestuia care se leagă la opgbp şi utilizarea acestuia, utilizarea unei forme solubile de odar, şi metodă de identificare a unui compus care descreşte activitatea opgbp |
US6217844B1 (en) * | 1998-04-27 | 2001-04-17 | Praecis Pharmaceuticals, Inc. | Methods for detecting lesions in dense breast tissue using LHRH antagonists |
CA2329941A1 (en) * | 1998-04-27 | 1999-11-04 | Marc B. Garnick | Methods for treating hot flashes and gynaecomastia |
US6191115B1 (en) * | 1998-08-12 | 2001-02-20 | Abbott Laboratories | C-terminus modified heptapeptide LHRH analogs |
US6455499B1 (en) * | 1999-02-23 | 2002-09-24 | Indiana University Foundation | Methods for treating disorders associated with LHRH activity |
US6703367B1 (en) * | 1999-04-27 | 2004-03-09 | Praecis Pharmaceuticals Inc. | Methods for treating hot flashes and gynaecomastia |
MXPA02001349A (es) * | 1999-08-09 | 2002-07-22 | Tripep Ab | Inhibidores de la polimerizacion de proteinas y metodos de uso. |
ATE362374T1 (de) * | 1999-09-03 | 2007-06-15 | Amgen Inc | Verfahren und zusammensetzungen zur prevention oder behandlung von krebs und von krebs assoziertem knochenverlust |
US20030103978A1 (en) | 2000-02-23 | 2003-06-05 | Amgen Inc. | Selective binding agents of osteoprotegerin binding protein |
US7109171B2 (en) * | 2000-02-28 | 2006-09-19 | Praecis Pharmaceuticals Inc. | Methods for treating FSH related conditions with GnRH antagonists |
KR20030021184A (ko) * | 2000-06-30 | 2003-03-12 | 산또리 가부시키가이샤 | 신규 생식선 자극 호르몬 방출 호르몬, 이의 전구체폴리펩티드 및 이들을 코딩하는 유전자 |
US6598784B2 (en) * | 2000-12-20 | 2003-07-29 | Meadwestvaco Packaging Syatens, Llc | Beverage carton with strap type carrying handle |
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ATE359790T1 (de) | 2001-05-16 | 2007-05-15 | Novartis Pharma Gmbh | Kombination von n- 5- 4-(4-methyl-piperazino- methyl)-benzoylamido -2-methylphenyl -4-(3- pyridil)-2pyrimidine-amin mit einem biphosphonat |
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EP1944026B1 (de) | 2002-05-16 | 2013-06-26 | Novartis AG | Verwendung von EDG-Rezeptorbindemitteln bei Krebs |
US6861236B2 (en) | 2002-05-24 | 2005-03-01 | Applied Nanosystems B.V. | Export and modification of (poly)peptides in the lantibiotic way |
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AU2006207325B2 (en) | 2005-01-21 | 2012-08-16 | Astex Therapeutics Limited | Pharmaceutical compounds |
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Family Cites Families (76)
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US3974135A (en) * | 1971-06-24 | 1976-08-10 | Karl Folkers | Synthetic decapeptide having the activity of the luteinizing hormone releasing hormone and method for producing the same |
US3953416A (en) * | 1971-12-20 | 1976-04-27 | Karl Folkers | Synthetic decapeptide having the activity of the luteinizing hormone releasing hormone and method for manufacturing the same |
GB1542703A (en) * | 1975-10-29 | 1979-03-21 | Parke Davis & Co | Nonapeptides and methods for their production |
DE2649114A1 (de) * | 1975-10-29 | 1977-05-12 | Parke Davis & Co | Octapeptide |
DE2617646C2 (de) * | 1976-04-22 | 1986-07-31 | Hoechst Ag, 6230 Frankfurt | Nonapeptid-amide und Decapeptid-amide mit Gonadoliberin-Wirkung, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Präparate |
US4215038A (en) * | 1978-10-16 | 1980-07-29 | The Salk Institute For Biological Studies | Peptides which inhibit gonadal function |
US4307083A (en) * | 1978-10-16 | 1981-12-22 | The Salk Institute For Biological Studies | LRF Antagonists |
US4244946A (en) * | 1979-06-11 | 1981-01-13 | The Salk Institute For Biological Studies | Water-soluble peptides affecting gonadal function |
US4409208A (en) * | 1980-04-15 | 1983-10-11 | The Salk Institute For Biological Studies | GnRH antagonists |
US4292313A (en) * | 1980-04-15 | 1981-09-29 | The Salk Institute For Biological Studies | LRF Antagonists |
US4377574A (en) * | 1980-06-26 | 1983-03-22 | The Salk Institute For Biological Studies | Contraceptive treatment of male mammals |
US4386074A (en) * | 1980-08-29 | 1983-05-31 | The Salk Institute For Biological Studies | LRF Antagonists |
US4341767A (en) * | 1980-10-06 | 1982-07-27 | Syntex Inc. | Nonapeptide and decapeptide analogs of LHRH, useful as LHRH antagonists |
US4419347A (en) * | 1980-10-06 | 1983-12-06 | Syntex (U.S.A.) Inc. | Nonapeptide and decapeptide analogs of LHRH, useful as LHRH antagonists |
US4489061A (en) * | 1981-06-12 | 1984-12-18 | The Salk Institute For Biological Studies | Treatment of male mammals |
US4667014A (en) * | 1983-03-07 | 1987-05-19 | Syntex (U.S.A.) Inc. | Nonapeptide and decapeptide analogs of LHRH, useful as LHRH antagonists |
US4481190A (en) * | 1982-12-21 | 1984-11-06 | Syntex (U.S.A.) Inc. | Nonapeptide and decapeptide analogs of LHRH useful as LHRH antagonists |
US4581169A (en) * | 1982-12-21 | 1986-04-08 | Syntex (U.S.A.) Inc. | Nona-peptide and deca-peptide analogs of LHRH, useful as LHRH antagonists |
US4444759A (en) * | 1982-07-26 | 1984-04-24 | The Salk Institute For Biological Studies | GnRH Antagonists II |
US4619914A (en) * | 1983-03-10 | 1986-10-28 | The Salk Institute For Biological Studies | GNRH antagonists IIIB |
US4504414A (en) * | 1983-03-28 | 1985-03-12 | Board Of Regents, The University Of Texas System | Synthetic pyridyl-alanyl decapeptides having antiovulatory activity |
DE3467173D1 (en) * | 1983-08-16 | 1987-12-10 | Akzo Nv | Lh- rh antagonists |
US4547370A (en) * | 1983-11-29 | 1985-10-15 | The Salk Institute For Biological Studies | GnRH Antagonists |
US4569927A (en) * | 1984-02-23 | 1986-02-11 | The Salk Institute For Biological Studies | GnRH Antagonists IV |
US4652550A (en) * | 1984-05-21 | 1987-03-24 | The Salk Institute For Biological Studies | GnRH antagonists VII |
US4647653A (en) * | 1984-08-23 | 1987-03-03 | Tulane Educational Fund | Therapeutic peptides |
US4565804A (en) * | 1984-09-07 | 1986-01-21 | The Salk Institute For Biological Studies | GnRH Antagonists VI |
US4690916A (en) * | 1984-11-13 | 1987-09-01 | Syntex (U.S.A.) Inc. | Nona and decapeptide analogs of LHRH useful as LHRH antagonists |
US4740500A (en) * | 1985-01-31 | 1988-04-26 | The Salk Institute For Biological Studies | GnRH antagonists VIII |
US4659691A (en) * | 1985-02-08 | 1987-04-21 | Merck & Co., Inc. | Novel cyclic Hexapeptide LHRH antagonists |
US4677193A (en) * | 1985-02-22 | 1987-06-30 | The Salk Institute For Biological Studies | Peptides containing an aliphatic-aromatic ketone side chain |
US5003011A (en) * | 1985-04-09 | 1991-03-26 | The Administrators Of The Tulane Educational Fund | Therapeutic decapeptides |
US4866160A (en) * | 1985-04-09 | 1989-09-12 | The Administrators Of The Tulane Educational Fund | Therapeutic decapeptides |
US5073624A (en) * | 1985-04-09 | 1991-12-17 | Administrators Of The Tulane Educational Fund | Therapeutic decapeptides |
US4656247A (en) * | 1985-04-26 | 1987-04-07 | Board Of Regents, The University Of Texas System | Effective hormonal peptides: D-3-QA1 6-LHRH |
US4642332A (en) * | 1985-04-26 | 1987-02-10 | The Board Of Regents, The University Of Texas System | Effective hormonal peptides: D-3-Pal6 -LHRH |
US4661472A (en) * | 1985-05-09 | 1987-04-28 | The Salk Institute For Biological Studies | GnRH antagonists IX |
US4721775A (en) * | 1985-08-26 | 1988-01-26 | Board Of Regents, The University Of Texas System | Effective peptides related to the luteinizing hormone releasing hormone from L-amino acids |
US4705778A (en) * | 1985-10-22 | 1987-11-10 | Sri International | Orally active LHRH analogs |
US5182205A (en) * | 1986-11-27 | 1993-01-26 | Hoffmann-La Roche Inc. | Nucleotide sequences which are selectively expressed in pre-B cells and probes therefor |
US4801577A (en) * | 1987-02-05 | 1989-01-31 | Syntex (U.S.A.) Inc. | Nonapeptide and decapeptide analogs of LHRH useful as LHRH antagonists |
US4851385A (en) * | 1987-07-15 | 1989-07-25 | Indiana University Foundation | LHRH antagonist analogs having low histamine-release activity |
US4800191A (en) * | 1987-07-17 | 1989-01-24 | Schally Andrew Victor | LHRH antagonists |
US4935491A (en) * | 1987-08-24 | 1990-06-19 | Board Of Regents, The University Of Texas System | Effective antagonists of the luteinizing hormone releasing hormone which release negligible histamine |
ES2108684T3 (es) * | 1988-02-10 | 1998-01-01 | Tap Pharmaceuticals Inc | Analogo de la hormona de liberacion de la hormona luteinizante (lhrh). |
US5300492A (en) * | 1988-02-10 | 1994-04-05 | Tap Pharmaceuticals | LHRH analogs |
US5110904A (en) * | 1989-08-07 | 1992-05-05 | Abbott Laboratories | Lhrh analogs |
US5140009A (en) * | 1988-02-10 | 1992-08-18 | Tap Pharmaceuticals, Inc. | Octapeptide LHRH antagonists |
GB2218102B (en) * | 1988-04-08 | 1992-09-16 | Sandoz Ltd | Calcitonin peptide derivatives |
US4992421A (en) * | 1988-04-19 | 1991-02-12 | Abbott Laboratories | Luteinizing hormone releasing hormone antagonist |
US5258492A (en) * | 1988-10-21 | 1993-11-02 | The Administrators Of The Tulane Educational Fund | LHRH analogues with cytotoxic moieties at the sixth position |
US5171835A (en) * | 1988-10-21 | 1992-12-15 | The Administrators Of The Tulane Educational Fund | LHRH antagonists |
US5296468A (en) * | 1989-10-30 | 1994-03-22 | The Salk Institute For Biological Studies | GnRH analogs |
US5169932A (en) * | 1989-10-30 | 1992-12-08 | The Salk Institute For Biological Studies | Gnrh analogs |
US5352796A (en) * | 1989-10-30 | 1994-10-04 | The Salk Institute For Biological Studies | Amino acids useful in making GnRH analogs |
US5064939A (en) * | 1990-02-06 | 1991-11-12 | The Salk Institute For Biological Studies | Cyclic gnrh antagonists |
US5180711A (en) * | 1990-06-14 | 1993-01-19 | Applied Research Systems Ars Holding N.V. | Combined treatment with gnrh antagonist and gnrh to control gonadotropin levels in mammals |
CN1036343C (zh) * | 1990-11-10 | 1997-11-05 | 天津市计划生育研究所 | 新促黄体生成素释放激素拮抗类似物的制备方法 |
IL101074A (en) * | 1991-03-14 | 1997-09-30 | Salk Inst For Biological Studi | GnRH ANALOGS AND THEIR PREPARATION |
US5340585A (en) * | 1991-04-12 | 1994-08-23 | University Of Southern California | Method and formulations for use in treating benign gynecological disorders |
JP2719233B2 (ja) * | 1991-04-25 | 1998-02-25 | デゲンギ,ロマノ | 黄体形成ホルモン放出ホルモン拮抗ペプチド |
DE4117507A1 (de) * | 1991-05-24 | 1992-11-26 | Schering Ag | Verfahren zur herstellung von n(pfeil hoch)6(pfeil hoch)-substituierten lysin-derivaten |
US5480969A (en) * | 1992-09-15 | 1996-01-02 | The Administrators Of The Tulane Educational Fund | Antagonists of LHRH |
US5371070A (en) * | 1992-11-09 | 1994-12-06 | The Salk Institute For Biological Studies | Bicyclic GnRH antagonists and a method for regulating the secretion of gonadotropins |
JPH08504209A (ja) * | 1992-12-04 | 1996-05-07 | アボツト・ラボラトリーズ | 6位修飾デカペプチドlhrh拮抗薬 |
JP3568952B2 (ja) * | 1992-12-18 | 2004-09-22 | アボット・ラボラトリーズ | 5位及び6位に修飾アミノアシル残基を有するlhrh拮抗薬 |
SG50426A1 (en) * | 1993-05-20 | 1998-07-20 | Biotech Australia Pty Ltd | Lhrh antagonists |
DE4320201A1 (de) * | 1993-06-18 | 1995-01-12 | Asta Medica Ag | Verwendung von Cetrorelix und weiteren Nona- und Dekapeptiden zur Herstellung eines Arzneimittels zur Bekämpfung von Aids und zur Wachstumsstimulation |
US5413990A (en) * | 1993-08-06 | 1995-05-09 | Tap Pharmaceuticals Inc. | N-terminus modified analogs of LHRH |
US5502035A (en) * | 1993-08-06 | 1996-03-26 | Tap Holdings Inc. | N-terminus modified analogs of LHRH |
US5508383A (en) * | 1994-03-09 | 1996-04-16 | Tap Holdings Inc. | Cyclic peptide LHRH antagonists |
US5506207A (en) * | 1994-03-18 | 1996-04-09 | The Salk Institute For Biological Studies | GNRH antagonists XIII |
US5516759A (en) * | 1994-12-08 | 1996-05-14 | Tap Holdings Inc. | LHRH antagonists having lactam groups at the N-terminus |
US5843901A (en) * | 1995-06-07 | 1998-12-01 | Advanced Research & Technology Institute | LHRH antagonist peptides |
US5780435A (en) * | 1995-12-15 | 1998-07-14 | Praecis Pharmaceuticals Incorporated | Methods for treating prostate cancer with LHRH-R antagonists |
-
1995
- 1995-06-07 US US08/480,494 patent/US5843901A/en not_active Expired - Lifetime
-
1996
- 1996-06-07 AT AT01204149T patent/ATE432941T1/de active
- 1996-06-07 US US08/973,378 patent/US6423686B1/en not_active Expired - Lifetime
- 1996-06-07 CA CA002219460A patent/CA2219460C/en not_active Expired - Fee Related
- 1996-06-07 ES ES01204149T patent/ES2326861T3/es not_active Expired - Lifetime
- 1996-06-07 DK DK01204149T patent/DK1188768T3/da active
- 1996-06-07 DE DE1996623254 patent/DE122006000012I1/de active Pending
- 1996-06-07 DE DE122006000012C patent/DE122006000012I2/de active Active
- 1996-06-07 DK DK96919311T patent/DK0794961T3/da active
- 1996-06-07 PT PT01204149T patent/PT1188768E/pt unknown
- 1996-06-07 EP EP96919311A patent/EP0794961B1/de not_active Expired - Lifetime
- 1996-06-07 DE DE69535963T patent/DE69535963D1/de not_active Expired - Lifetime
- 1996-06-07 EP EP01204149A patent/EP1188768B1/de not_active Expired - Lifetime
- 1996-06-07 AU AU61680/96A patent/AU715399B2/en not_active Ceased
- 1996-06-07 WO PCT/US1996/009852 patent/WO1996040757A2/en active Search and Examination
- 1996-06-07 ES ES96919311T patent/ES2177789T3/es not_active Expired - Lifetime
- 1996-06-07 DE DE69623254T patent/DE69623254T2/de not_active Expired - Lifetime
- 1996-06-07 JP JP50205097A patent/JP4164125B2/ja not_active Expired - Fee Related
- 1996-06-07 PT PT96919311T patent/PT794961E/pt unknown
- 1996-06-07 AT AT96919311T patent/ATE222924T1/de active
-
2002
- 2002-04-02 US US10/115,553 patent/US20030040482A1/en not_active Abandoned
- 2002-04-05 US US10/117,364 patent/US7071165B2/en not_active Expired - Fee Related
- 2002-09-11 HK HK02106667.7A patent/HK1045161B/zh not_active IP Right Cessation
-
2006
- 2006-03-03 LU LU91225C patent/LU91225I2/fr unknown
-
2007
- 2007-08-13 JP JP2007211155A patent/JP2007302695A/ja not_active Withdrawn
-
2008
- 2008-10-09 JP JP2008263288A patent/JP2009040793A/ja not_active Withdrawn
-
2011
- 2011-08-22 LU LU91857C patent/LU91857I2/fr unknown
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