LU91857I2 - Abarelix, optionnellement sous forme de sel pharmaceutiquement acceptable - Google Patents

Abarelix, optionnellement sous forme de sel pharmaceutiquement acceptable

Info

Publication number
LU91857I2
LU91857I2 LU91857C LU91857C LU91857I2 LU 91857 I2 LU91857 I2 LU 91857I2 LU 91857 C LU91857 C LU 91857C LU 91857 C LU91857 C LU 91857C LU 91857 I2 LU91857 I2 LU 91857I2
Authority
LU
Luxembourg
Prior art keywords
moiety
abarelix
optionally
pharmaceutically acceptable
acceptable salt
Prior art date
Application number
LU91857C
Other languages
English (en)
Original Assignee
Univ Indiana Res & Tech Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Indiana Res & Tech Corp filed Critical Univ Indiana Res & Tech Corp
Publication of LU91857I2 publication Critical patent/LU91857I2/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/13—Luteinizing hormone-releasing hormone; related peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Immunology (AREA)
  • Biochemistry (AREA)
  • Diabetes (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Urology & Nephrology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
LU91857C 1995-06-07 2011-08-22 Abarelix, optionnellement sous forme de sel pharmaceutiquement acceptable LU91857I2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/480,494 US5843901A (en) 1995-06-07 1995-06-07 LHRH antagonist peptides
PCT/US1996/009852 WO1996040757A2 (fr) 1995-06-07 1996-06-07 Peptides antagonistes de la lh-rh

Publications (1)

Publication Number Publication Date
LU91857I2 true LU91857I2 (fr) 2011-10-24

Family

ID=23908180

Family Applications (2)

Application Number Title Priority Date Filing Date
LU91225C LU91225I2 (fr) 1995-06-07 2006-03-03 Plenaxis
LU91857C LU91857I2 (fr) 1995-06-07 2011-08-22 Abarelix, optionnellement sous forme de sel pharmaceutiquement acceptable

Family Applications Before (1)

Application Number Title Priority Date Filing Date
LU91225C LU91225I2 (fr) 1995-06-07 2006-03-03 Plenaxis

Country Status (13)

Country Link
US (4) US5843901A (fr)
EP (2) EP0794961B1 (fr)
JP (3) JP4164125B2 (fr)
AT (2) ATE432941T1 (fr)
AU (1) AU715399B2 (fr)
CA (1) CA2219460C (fr)
DE (4) DE69535963D1 (fr)
DK (2) DK1188768T3 (fr)
ES (2) ES2177789T3 (fr)
HK (1) HK1045161B (fr)
LU (2) LU91225I2 (fr)
PT (2) PT794961E (fr)
WO (1) WO1996040757A2 (fr)

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JP4164125B2 (ja) 2008-10-08
PT1188768E (pt) 2009-08-13
US6423686B1 (en) 2002-07-23
EP1188768A3 (fr) 2002-10-23
EP0794961B1 (fr) 2002-08-28
ATE432941T1 (de) 2009-06-15
DE69623254T2 (de) 2002-12-19
US20030181385A1 (en) 2003-09-25
ES2177789T3 (es) 2002-12-16
WO1996040757A3 (fr) 1997-02-20
DK1188768T3 (da) 2009-09-21
JPH11507374A (ja) 1999-06-29
WO1996040757A2 (fr) 1996-12-19
EP0794961A2 (fr) 1997-09-17
DE122006000012I1 (de) 2006-06-29
LU91225I2 (fr) 2006-05-03
US5843901A (en) 1998-12-01
JP2007302695A (ja) 2007-11-22
US20020115615A1 (en) 2002-08-22
HK1045161B (zh) 2009-12-24
ES2326861T3 (es) 2009-10-21
DK0794961T3 (da) 2002-10-21
DE69535963D1 (de) 2009-07-16
US20030040482A1 (en) 2003-02-27
AU6168096A (en) 1996-12-30
AU715399B2 (en) 2000-02-03
CA2219460A1 (fr) 1996-12-19
EP1188768B1 (fr) 2009-06-03
CA2219460C (fr) 2009-04-14
HK1045161A1 (en) 2002-11-15
DE122006000012I2 (de) 2010-02-04
JP2009040793A (ja) 2009-02-26
US7071165B2 (en) 2006-07-04
ATE222924T1 (de) 2002-09-15
EP1188768A2 (fr) 2002-03-20
DE69623254D1 (de) 2002-10-02
PT794961E (pt) 2003-01-31

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