JP2023116503A5 - - Google Patents

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JP2023116503A5
JP2023116503A5 JP2023085024A JP2023085024A JP2023116503A5 JP 2023116503 A5 JP2023116503 A5 JP 2023116503A5 JP 2023085024 A JP2023085024 A JP 2023085024A JP 2023085024 A JP2023085024 A JP 2023085024A JP 2023116503 A5 JP2023116503 A5 JP 2023116503A5
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pharmaceutical composition
composition according
crystalline form
treatment
btk
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JP2023085024A
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JP2023116503A (ja
JP7596441B2 (ja
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JP2023085024A 2018-07-31 2023-05-24 (s)-5-アミノ-3-(4-((5-フルオロ-2-メトキシベンズアミド)メチル)フェニル)-1-(1,1,1-トリフルオロプロパン-2-イル)-1h-ピラゾール-4-カルボキサミドの噴霧乾燥分散体および製剤 Active JP7596441B2 (ja)

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JP2024206520A JP2025037966A (ja) 2018-07-31 2024-11-27 (s)-5-アミノ-3-(4-((5-フルオロ-2-メトキシベンズアミド)メチル)フェニル)-1-(1,1,1-トリフルオロプロパン-2-イル)-1h-ピラゾール-4-カルボキサミドの噴霧乾燥分散体および製剤

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US201862712861P 2018-07-31 2018-07-31
US62/712,861 2018-07-31
US201862729855P 2018-09-11 2018-09-11
US62/729,855 2018-09-11
US201862769308P 2018-11-19 2018-11-19
US62/769,308 2018-11-19
PCT/US2019/043937 WO2020028258A1 (en) 2018-07-31 2019-07-29 Spray-dried dispersions and formulations of (s)-5-amino-3-(4-((5-fluoro-2-methoxybenzamido)methyl)phenyl)-1-(1,1,1-trifluoro propan-2-yl)-1h-pyrazole-4-carboxamide
JP2021505208A JP7286755B2 (ja) 2018-07-31 2019-07-29 (s)-5-アミノ-3-(4-((5-フルオロ-2-メトキシベンズアミド)メチル)フェニル)-1-(1,1,1-トリフルオロプロパン-2-イル)-1h-ピラゾール-4-カルボキサミドの噴霧乾燥分散体および製剤

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JP2021505208A Division JP7286755B2 (ja) 2018-07-31 2019-07-29 (s)-5-アミノ-3-(4-((5-フルオロ-2-メトキシベンズアミド)メチル)フェニル)-1-(1,1,1-トリフルオロプロパン-2-イル)-1h-ピラゾール-4-カルボキサミドの噴霧乾燥分散体および製剤

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JP2024206520A Division JP2025037966A (ja) 2018-07-31 2024-11-27 (s)-5-アミノ-3-(4-((5-フルオロ-2-メトキシベンズアミド)メチル)フェニル)-1-(1,1,1-トリフルオロプロパン-2-イル)-1h-ピラゾール-4-カルボキサミドの噴霧乾燥分散体および製剤

Publications (3)

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JP2023116503A JP2023116503A (ja) 2023-08-22
JP2023116503A5 true JP2023116503A5 (enExample) 2024-02-05
JP7596441B2 JP7596441B2 (ja) 2024-12-09

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JP2021505208A Active JP7286755B2 (ja) 2018-07-31 2019-07-29 (s)-5-アミノ-3-(4-((5-フルオロ-2-メトキシベンズアミド)メチル)フェニル)-1-(1,1,1-トリフルオロプロパン-2-イル)-1h-ピラゾール-4-カルボキサミドの噴霧乾燥分散体および製剤
JP2023085024A Active JP7596441B2 (ja) 2018-07-31 2023-05-24 (s)-5-アミノ-3-(4-((5-フルオロ-2-メトキシベンズアミド)メチル)フェニル)-1-(1,1,1-トリフルオロプロパン-2-イル)-1h-ピラゾール-4-カルボキサミドの噴霧乾燥分散体および製剤
JP2024206520A Pending JP2025037966A (ja) 2018-07-31 2024-11-27 (s)-5-アミノ-3-(4-((5-フルオロ-2-メトキシベンズアミド)メチル)フェニル)-1-(1,1,1-トリフルオロプロパン-2-イル)-1h-ピラゾール-4-カルボキサミドの噴霧乾燥分散体および製剤

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JP2021505208A Active JP7286755B2 (ja) 2018-07-31 2019-07-29 (s)-5-アミノ-3-(4-((5-フルオロ-2-メトキシベンズアミド)メチル)フェニル)-1-(1,1,1-トリフルオロプロパン-2-イル)-1h-ピラゾール-4-カルボキサミドの噴霧乾燥分散体および製剤

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Country Status (8)

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US (3) US12109193B2 (enExample)
EP (1) EP3829543A1 (enExample)
JP (3) JP7286755B2 (enExample)
KR (3) KR102653681B1 (enExample)
CN (3) CN117285467A (enExample)
AU (3) AU2019314302A1 (enExample)
CA (4) CA3224945C (enExample)
WO (1) WO2020028258A1 (enExample)

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KR20220100992A (ko) * 2019-12-06 2022-07-18 록쏘 온콜로지, 인코포레이티드 브루톤 티로신 키나제 억제제의 투여
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AU2022337087A1 (en) * 2021-09-03 2024-03-14 Novartis Ag Lou064 for treating multiple sclerosis
WO2024176164A1 (en) 2023-02-22 2024-08-29 Assia Chemical Industries Ltd. Solid state form of pirtobrutinib
WO2024179558A1 (zh) * 2023-03-02 2024-09-06 苏州科睿思制药有限公司 Pirtobrutinib的晶型及其制备方法和用途
WO2024194890A1 (en) * 2023-03-20 2024-09-26 Dr. Reddy’S Laboratories Limited Solid state forms of pirtobrutinib and process for the preparation of intermediate thereof
WO2025078941A1 (en) * 2023-10-09 2025-04-17 Intas Pharmaceuticals Ltd. Pharmaceutical composition of pirtobrutinib
WO2025083736A1 (en) * 2023-10-20 2025-04-24 Msn Laboratories Private Limited, R&D Center Novel process for the preparation of pirtobrutinib and its intermediates thereof
CN119857081B (zh) * 2025-01-16 2025-10-17 江苏亚邦爱普森药业有限公司 一种乌帕替尼缓释片及其制备方法
CN120591230B (zh) * 2025-07-02 2025-11-25 广东金骏康生物技术有限公司 一种甲基转移酶CicOMT10突变体、制备方法、生物材料和应用

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