JP2022507957A5 - - Google Patents

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Publication number
JP2022507957A5
JP2022507957A5 JP2021529266A JP2021529266A JP2022507957A5 JP 2022507957 A5 JP2022507957 A5 JP 2022507957A5 JP 2021529266 A JP2021529266 A JP 2021529266A JP 2021529266 A JP2021529266 A JP 2021529266A JP 2022507957 A5 JP2022507957 A5 JP 2022507957A5
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JP
Japan
Prior art keywords
methyl
chlorobenzyl
imidazole
tetraone
phenoxy
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JP2021529266A
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English (en)
Japanese (ja)
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JP7577656B2 (ja
JP2022507957A (ja
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Priority claimed from PCT/IB2019/060201 external-priority patent/WO2020110009A1/en
Publication of JP2022507957A publication Critical patent/JP2022507957A/ja
Publication of JP2022507957A5 publication Critical patent/JP2022507957A5/ja
Application granted granted Critical
Publication of JP7577656B2 publication Critical patent/JP7577656B2/ja
Active legal-status Critical Current
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JP2021529266A 2018-11-27 2019-11-26 代謝障害の治療用のプロタンパク質転換酵素サブチリシン/ケキシン9型(pcsk9)阻害薬としての環状四量体化合物 Active JP7577656B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862772030P 2018-11-27 2018-11-27
US62/772,030 2018-11-27
US201962924828P 2019-10-23 2019-10-23
US62/924,828 2019-10-23
PCT/IB2019/060201 WO2020110009A1 (en) 2018-11-27 2019-11-26 Cyclic tetramer compounds as proprotein convertase subtilisin/kexin type 9 (pcsk9) inhibitors for the treatment of metabolic disorders

Publications (3)

Publication Number Publication Date
JP2022507957A JP2022507957A (ja) 2022-01-18
JP2022507957A5 true JP2022507957A5 (https=) 2022-12-05
JP7577656B2 JP7577656B2 (ja) 2024-11-05

Family

ID=68808460

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021529266A Active JP7577656B2 (ja) 2018-11-27 2019-11-26 代謝障害の治療用のプロタンパク質転換酵素サブチリシン/ケキシン9型(pcsk9)阻害薬としての環状四量体化合物

Country Status (25)

Country Link
US (2) US11026993B2 (https=)
EP (1) EP3887365A1 (https=)
JP (1) JP7577656B2 (https=)
KR (1) KR20210096154A (https=)
CN (1) CN113166114B (https=)
AU (1) AU2019387294B2 (https=)
BR (1) BR112021009857A2 (https=)
CA (1) CA3115960A1 (https=)
CL (1) CL2021001365A1 (https=)
CO (1) CO2021006895A2 (https=)
CR (1) CR20210267A (https=)
CU (1) CU20210043A7 (https=)
DO (1) DOP2021000100A (https=)
EC (1) ECSP21036194A (https=)
IL (1) IL283374A (https=)
JO (1) JOP20210120A1 (https=)
MA (1) MA54284A (https=)
MX (1) MX2021006069A (https=)
PE (1) PE20211658A1 (https=)
PH (1) PH12021551049A1 (https=)
PY (1) PY1998404A (https=)
SG (1) SG11202103807WA (https=)
TW (1) TW202038990A (https=)
UY (1) UY38485A (https=)
WO (1) WO2020110009A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11882610B2 (en) * 2020-08-13 2024-01-23 Qualcomm Incorporated Establishing connections using multiple subscriber identity modules via a single communication link
CN114163343A (zh) * 2021-12-10 2022-03-11 许昌学院 含氟氨基酸及衍生物含氟多肽的制备方法以及应用

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