JP2021534095A5 - - Google Patents

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Publication number
JP2021534095A5
JP2021534095A5 JP2021506575A JP2021506575A JP2021534095A5 JP 2021534095 A5 JP2021534095 A5 JP 2021534095A5 JP 2021506575 A JP2021506575 A JP 2021506575A JP 2021506575 A JP2021506575 A JP 2021506575A JP 2021534095 A5 JP2021534095 A5 JP 2021534095A5
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unsubstituted
substituted
alkyl
halogen
pharmaceutically acceptable
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JP2021506575A
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English (en)
Japanese (ja)
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JP7429988B2 (ja
JP2021534095A (ja
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Priority claimed from EP18290093.6A external-priority patent/EP3608318A1/en
Priority claimed from EP18213635.8A external-priority patent/EP3670512A1/en
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Priority claimed from PCT/EP2019/071370 external-priority patent/WO2020030761A1/en
Publication of JP2021534095A publication Critical patent/JP2021534095A/ja
Publication of JP2021534095A5 publication Critical patent/JP2021534095A5/ja
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JP2021506575A 2018-08-09 2019-08-08 セリンベータ-ラクタマーゼのインヒビターとしてのジアザビシクロオクタノン Active JP7429988B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP18290093.6 2018-08-09
EP18290093.6A EP3608318A1 (en) 2018-08-09 2018-08-09 Diaazabicyclooctanone derivatives as antibacterials
EP18213635.8A EP3670512A1 (en) 2018-12-18 2018-12-18 Diazabicyclooctanones as inhibitors of serine beta-lactamases
EP18213635.8 2018-12-18
PCT/EP2019/071370 WO2020030761A1 (en) 2018-08-09 2019-08-08 Diazabicyclooctanones as inhibitors of serine beta-lactamases

Publications (3)

Publication Number Publication Date
JP2021534095A JP2021534095A (ja) 2021-12-09
JP2021534095A5 true JP2021534095A5 (https=) 2022-08-18
JP7429988B2 JP7429988B2 (ja) 2024-02-09

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JP2021506575A Active JP7429988B2 (ja) 2018-08-09 2019-08-08 セリンベータ-ラクタマーゼのインヒビターとしてのジアザビシクロオクタノン

Country Status (24)

Country Link
US (1) US12378244B2 (https=)
EP (2) EP4272831A3 (https=)
JP (1) JP7429988B2 (https=)
KR (1) KR102790878B1 (https=)
CN (2) CN111954671B (https=)
AU (1) AU2019318115B2 (https=)
BR (1) BR112021002311A2 (https=)
CA (1) CA3110111A1 (https=)
DK (1) DK3833665T3 (https=)
ES (1) ES2960952T3 (https=)
FI (1) FI3833665T3 (https=)
HR (1) HRP20231228T1 (https=)
HU (1) HUE063324T2 (https=)
IL (1) IL280770B2 (https=)
LT (1) LT3833665T (https=)
MX (1) MX2021001564A (https=)
PL (1) PL3833665T3 (https=)
RS (1) RS64679B1 (https=)
SG (1) SG11202101255UA (https=)
SI (1) SI3833665T1 (https=)
SM (1) SMT202300354T1 (https=)
TW (1) TWI764030B (https=)
WO (1) WO2020030761A1 (https=)
ZA (1) ZA202100906B (https=)

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CN111943950B (zh) * 2020-09-10 2022-03-29 山东安信制药有限公司 一种瑞来巴坦的制备方法
US12410166B2 (en) 2021-05-07 2025-09-09 Ningxia Academy Of Agriculture And Forestry Sciences Sulfonylamidine substituted compounds and their use as beta-lactamase inhibitors
CN115448920B (zh) * 2022-10-14 2025-01-03 广州楷石医药有限公司 一种β-内酰胺酶抑制剂及其应用
GB202306833D0 (en) 2023-05-09 2023-06-21 Adjutec Pharma As Therapy
GB202306826D0 (en) 2023-05-09 2023-06-21 Adjutec Pharma As Therapy
CN117700415B (zh) * 2024-02-06 2024-04-30 成都四面体药物研究有限公司 含脲双环化合物、其用途、其制备的药物、其联合用药物及其复方制剂
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