JP2021528446A5 - - Google Patents

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Publication number
JP2021528446A5
JP2021528446A5 JP2020571690A JP2020571690A JP2021528446A5 JP 2021528446 A5 JP2021528446 A5 JP 2021528446A5 JP 2020571690 A JP2020571690 A JP 2020571690A JP 2020571690 A JP2020571690 A JP 2020571690A JP 2021528446 A5 JP2021528446 A5 JP 2021528446A5
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JP
Japan
Prior art keywords
oxa
azabicyclo
nonane
carboxylate
piperidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020571690A
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English (en)
Japanese (ja)
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JP2021528446A (ja
JP7317054B2 (ja
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Priority claimed from GBGB1810239.2A external-priority patent/GB201810239D0/en
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Publication of JP2021528446A publication Critical patent/JP2021528446A/ja
Publication of JP2021528446A5 publication Critical patent/JP2021528446A5/ja
Application granted granted Critical
Publication of JP7317054B2 publication Critical patent/JP7317054B2/ja
Active legal-status Critical Current
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JP2020571690A 2018-06-22 2019-06-24 ムスカリンm1および/またはm4受容体のアゴニストとしての架橋化合物 Active JP7317054B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB1810239.2 2018-06-22
GBGB1810239.2A GB201810239D0 (en) 2018-06-22 2018-06-22 Pharmaceutical compounds
PCT/GB2019/051780 WO2019243851A1 (en) 2018-06-22 2019-06-24 Bridged compounds as agonists of the muscarinic m1 and/or m4 receptor

Publications (3)

Publication Number Publication Date
JP2021528446A JP2021528446A (ja) 2021-10-21
JP2021528446A5 true JP2021528446A5 (enExample) 2022-06-30
JP7317054B2 JP7317054B2 (ja) 2023-07-28

Family

ID=63042513

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020571690A Active JP7317054B2 (ja) 2018-06-22 2019-06-24 ムスカリンm1および/またはm4受容体のアゴニストとしての架橋化合物

Country Status (10)

Country Link
US (2) US10787447B2 (enExample)
EP (1) EP3810614B1 (enExample)
JP (1) JP7317054B2 (enExample)
CN (1) CN112585143B (enExample)
AU (1) AU2019289217B2 (enExample)
CA (1) CA3104222A1 (enExample)
ES (1) ES2984420T3 (enExample)
GB (1) GB201810239D0 (enExample)
TW (1) TWI822803B (enExample)
WO (1) WO2019243851A1 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
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GB201810239D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) * 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds

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