JP2021512894A5 - - Google Patents

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Publication number
JP2021512894A5
JP2021512894A5 JP2020542552A JP2020542552A JP2021512894A5 JP 2021512894 A5 JP2021512894 A5 JP 2021512894A5 JP 2020542552 A JP2020542552 A JP 2020542552A JP 2020542552 A JP2020542552 A JP 2020542552A JP 2021512894 A5 JP2021512894 A5 JP 2021512894A5
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JP
Japan
Prior art keywords
composition
subject
compound according
pharmaceutically acceptable
acceptable salt
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020542552A
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English (en)
Japanese (ja)
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JP2021512894A (ja
JP7397797B2 (ja
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Priority claimed from PCT/US2019/016503 external-priority patent/WO2019156929A1/en
Publication of JP2021512894A publication Critical patent/JP2021512894A/ja
Publication of JP2021512894A5 publication Critical patent/JP2021512894A5/ja
Priority to JP2023203652A priority Critical patent/JP2024023490A/ja
Application granted granted Critical
Publication of JP7397797B2 publication Critical patent/JP7397797B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2020542552A 2018-02-07 2019-02-04 治療用化合物および組成物 Active JP7397797B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023203652A JP2024023490A (ja) 2018-02-07 2023-12-01 治療用化合物および組成物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862627435P 2018-02-07 2018-02-07
US62/627,435 2018-02-07
PCT/US2019/016503 WO2019156929A1 (en) 2018-02-07 2019-02-04 Therapeutic compounds and compositions

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023203652A Division JP2024023490A (ja) 2018-02-07 2023-12-01 治療用化合物および組成物

Publications (3)

Publication Number Publication Date
JP2021512894A JP2021512894A (ja) 2021-05-20
JP2021512894A5 true JP2021512894A5 (https=) 2022-02-14
JP7397797B2 JP7397797B2 (ja) 2023-12-13

Family

ID=67548561

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020542552A Active JP7397797B2 (ja) 2018-02-07 2019-02-04 治療用化合物および組成物
JP2023203652A Pending JP2024023490A (ja) 2018-02-07 2023-12-01 治療用化合物および組成物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023203652A Pending JP2024023490A (ja) 2018-02-07 2023-12-01 治療用化合物および組成物

Country Status (10)

Country Link
US (2) US11691962B2 (https=)
EP (1) EP3749662A4 (https=)
JP (2) JP7397797B2 (https=)
KR (1) KR20200118088A (https=)
CN (1) CN111902404A (https=)
AU (1) AU2019217366B2 (https=)
BR (1) BR112020016123A2 (https=)
CA (1) CA3089970A1 (https=)
IL (2) IL276563B1 (https=)
WO (1) WO2019156929A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2733405C2 (ru) 2014-02-07 2020-10-01 Экзитера Фармасьютикалз Инк. Терапевтические соединения и композиции
CA3089970A1 (en) 2018-02-07 2019-08-15 eXIthera Pharmaceuticals Inc. Therapeutic compounds and compositions

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4595532A (en) 1983-02-02 1986-06-17 University Of Notre Dame Du Lac N-(substituted-methyl)-azetidin-2-ones
JP2002501081A (ja) 1998-01-26 2002-01-15 ビーエーエスエフ アクチェンゲゼルシャフト トロンビンインヒビター
HUP0104308A3 (en) 1998-06-25 2002-06-28 Bristol Myers Squibb Co Amidino and guanidino azetidinone derivatives as tryptase inhibitors, process for their preparation, pharmaceutical compositions thereof and intermediates
US6335324B1 (en) 1998-06-25 2002-01-01 Bristol-Myers Squibb Co. Beta lactam compounds and their use as inhibitors of tryptase
EP1099690A4 (en) 1998-07-23 2001-10-17 Shionogi & Co MONOCYCLIC BETA LACTAM COMPOUNDS AND CHYMASE INHIBITORS THAT CONTAIN THEM
KR20060120601A (ko) 2003-08-22 2006-11-27 데이진 화-마 가부시키가이샤 키마제 저해제를 유효 성분으로서 함유하는 약제
EP1871741A4 (en) 2005-04-04 2012-01-11 Daiamed Inc SUBSTITUTED AZETIDINONE
TW200745084A (en) 2006-03-08 2007-12-16 Astrazeneca Ab Novel compounds
JP5756800B2 (ja) 2009-06-16 2015-07-29 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Cb2受容体を調節するアゼチジン2−カルボキサミド誘導体
NZ602266A (en) 2010-02-11 2014-05-30 Bristol Myers Squibb Co Macrocycles as factor xia inhibitors
JP6033319B2 (ja) 2011-10-14 2016-11-30 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company 第XIa因子阻害剤としての置換テトラヒドロイソキノリン化合物
SG11201406142XA (en) 2012-03-27 2014-10-30 Univ Duke Compositions and methods for the prevention and treatment of mast cell-induced vascular leakage
RU2733405C2 (ru) * 2014-02-07 2020-10-01 Экзитера Фармасьютикалз Инк. Терапевтические соединения и композиции
US20190315711A1 (en) 2016-12-23 2019-10-17 Exithera Pharmaceuticals, Inc. Therapeutic compounds and compositions
CA3089970A1 (en) 2018-02-07 2019-08-15 eXIthera Pharmaceuticals Inc. Therapeutic compounds and compositions
JP2022506110A (ja) 2018-10-30 2022-01-17 エクセセーラ ファーマシューティカルズ インコーポレイテッド 治療用化合物および組成物
CN113056263A (zh) 2018-10-30 2021-06-29 艾克赛特赫拉制药有限责任公司 治疗化合物和组合物
JP2022523712A (ja) 2019-01-29 2022-04-26 エクセセーラ ファーマシューティカルズ インコーポレイテッド 治療用化合物および組成物

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