JP2021504418A5 - - Google Patents
Info
- Publication number
- JP2021504418A5 JP2021504418A5 JP2020529522A JP2020529522A JP2021504418A5 JP 2021504418 A5 JP2021504418 A5 JP 2021504418A5 JP 2020529522 A JP2020529522 A JP 2020529522A JP 2020529522 A JP2020529522 A JP 2020529522A JP 2021504418 A5 JP2021504418 A5 JP 2021504418A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- methoxyisochroman
- ethyl
- carboxylate
- ethanol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FI20176085 | 2017-12-01 | ||
| FI20176085 | 2017-12-01 | ||
| PCT/FI2018/050864 WO2019106238A1 (en) | 2017-12-01 | 2018-11-30 | Process for the preparation of 2-(5-methoxyisochroman-1 -yl)-4,5-dihydro-1 h-imidazole and the hydrogensulfate salt thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021504418A JP2021504418A (ja) | 2021-02-15 |
| JP2021504418A5 true JP2021504418A5 (enExample) | 2023-07-13 |
| JP7339946B2 JP7339946B2 (ja) | 2023-09-06 |
Family
ID=64746580
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020529522A Active JP7339946B2 (ja) | 2017-12-01 | 2018-11-30 | 2-(5-メトキシイソクロマン-1-イル)-4,5-ジヒドロ-1h-イミダゾールおよびその硫酸水素塩の製造方法 |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US11352346B2 (enExample) |
| EP (1) | EP3717476B1 (enExample) |
| JP (1) | JP7339946B2 (enExample) |
| KR (1) | KR102718536B1 (enExample) |
| CN (1) | CN111630049B (enExample) |
| AU (1) | AU2018376872B2 (enExample) |
| BR (1) | BR112020010617A2 (enExample) |
| CA (1) | CA3083734A1 (enExample) |
| DK (1) | DK3717476T3 (enExample) |
| ES (1) | ES2927193T3 (enExample) |
| HR (1) | HRP20221247T1 (enExample) |
| HU (1) | HUE059849T2 (enExample) |
| IL (1) | IL274931B2 (enExample) |
| LT (1) | LT3717476T (enExample) |
| PL (1) | PL3717476T3 (enExample) |
| PT (1) | PT3717476T (enExample) |
| SI (1) | SI3717476T1 (enExample) |
| WO (1) | WO2019106238A1 (enExample) |
| ZA (1) | ZA202003981B (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE112020003658T5 (de) | 2019-07-31 | 2022-05-19 | Hyundai Motor Company | Sdn-basiertes eindringungsverhinderungsverfahren für ein fahrzeuginternesnetz und system, das dieses verfahren verwendet |
| KR20230159515A (ko) * | 2021-03-19 | 2023-11-21 | 오리온 코포레이션 | 타시피미딘 제형 및 이의 용도 |
| JP2025502480A (ja) * | 2022-01-24 | 2025-01-24 | オリオン コーポレーション | イソクロマン-イミダゾール構造のアルファ-2aアドレナリン受容体アゴニストの新規な硫酸塩形 |
| WO2023148431A1 (en) | 2022-02-04 | 2023-08-10 | Orion Corporation | Novel salt forms of isochroman-imidazole structured alpha-2a adrenoceptor agonist |
| JP2025531623A (ja) | 2022-09-28 | 2025-09-22 | オリオン コーポレーション | タシピミジンおよびcyp2d6阻害薬の併用療法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6410562B1 (en) * | 1998-12-18 | 2002-06-25 | Eli Lilly And Company | Hypoglycemic imidazoline compounds |
| AR090557A1 (es) * | 2012-04-02 | 2014-11-19 | Orion Corp | DERIVADOS IMIDAZOLICOS AGONISTAS ADRENERGICOS a2 |
-
2018
- 2018-11-30 JP JP2020529522A patent/JP7339946B2/ja active Active
- 2018-11-30 KR KR1020207019100A patent/KR102718536B1/ko active Active
- 2018-11-30 PL PL18822414.1T patent/PL3717476T3/pl unknown
- 2018-11-30 HU HUE18822414A patent/HUE059849T2/hu unknown
- 2018-11-30 CN CN201880076883.0A patent/CN111630049B/zh active Active
- 2018-11-30 WO PCT/FI2018/050864 patent/WO2019106238A1/en not_active Ceased
- 2018-11-30 BR BR112020010617-8A patent/BR112020010617A2/pt unknown
- 2018-11-30 AU AU2018376872A patent/AU2018376872B2/en active Active
- 2018-11-30 SI SI201830738T patent/SI3717476T1/sl unknown
- 2018-11-30 HR HRP20221247TT patent/HRP20221247T1/hr unknown
- 2018-11-30 ES ES18822414T patent/ES2927193T3/es active Active
- 2018-11-30 PT PT188224141T patent/PT3717476T/pt unknown
- 2018-11-30 LT LTEPPCT/FI2018/050864T patent/LT3717476T/lt unknown
- 2018-11-30 DK DK18822414.1T patent/DK3717476T3/da active
- 2018-11-30 EP EP18822414.1A patent/EP3717476B1/en active Active
- 2018-11-30 US US16/768,093 patent/US11352346B2/en active Active
- 2018-11-30 CA CA3083734A patent/CA3083734A1/en active Pending
- 2018-11-30 IL IL274931A patent/IL274931B2/en unknown
-
2020
- 2020-06-30 ZA ZA2020/03981A patent/ZA202003981B/en unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP6625115B2 (ja) | 4−アルコキシ−3−ヒドロキシピコリン酸の製造方法 | |
| JP7339946B2 (ja) | 2-(5-メトキシイソクロマン-1-イル)-4,5-ジヒドロ-1h-イミダゾールおよびその硫酸水素塩の製造方法 | |
| JP6228210B2 (ja) | フルボキサミン遊離塩基の精製方法およびそれを用いた高純度フルボキサミンマレイン酸塩の製造方法 | |
| JP6533798B2 (ja) | ジヒドロイソオキサゾール誘導体の製造方法 | |
| WO2014206254A1 (zh) | 一种4-苄基-1-苯乙基哌嗪-2,6-二酮的制备方法、中间体及其制备方法 | |
| CN109563079A (zh) | 脱氢苯基阿夕斯丁类化合物的多晶型及其制备纯化方法和应用 | |
| CN109485567B (zh) | 一种4-羟甲基噻唑的清洁制备方法及其中间体 | |
| TWI361807B (en) | Process for preparing substituted 4-alkoxycarbonyl-3-aminothiophenes | |
| CN109180564B (zh) | 一种哌啶及其衍生物的制备方法 | |
| CA2930089C (en) | Fingolimod hydrochloride process | |
| TW201900602A (zh) | 1-胺基環丙烷羧酸非水合物之製造方法 | |
| CN104030942A (zh) | 一种L-α-氨基丁酰胺盐酸盐的制备方法 | |
| JP2013517235A (ja) | インダゾール−3−カルボン酸及びn−(s)−1−アザビシクロ[2.2.2]オクタ−3−イル−1h−インダゾール−3−カルボキサミド塩酸塩の調製方法 | |
| JP6802815B2 (ja) | ジクロロキノン誘導体の製造方法 | |
| JP6433809B2 (ja) | 1−(3−ヒドロキシメチルピリジル−2−)−2−フェニル−4−メチルピペラジンの製造方法 | |
| TWI753978B (zh) | 製備4-胺基-3-氯-5-氟-6-(4-氯-2-氟-3-甲氧基苯基)吡啶甲酸甲酯之方法 | |
| CN109761894A (zh) | 一种5-溴-2-吡啶甲酸的制备方法 | |
| JP4399996B2 (ja) | 3−オキソニトリル類の製造法 | |
| JP6219516B2 (ja) | 2−アミノ−6−メチルニコチン酸の製造方法 | |
| JP6660393B2 (ja) | 4−シアノピペリジン塩酸塩を調製する方法 | |
| RU2613559C1 (ru) | Способ получения 2-замещенных 1-гидрокси-1Н-индол-5,6-дикарбоновых кислот | |
| CN106187799A (zh) | 一种制备dl‑赖氨酸盐酸盐的方法 | |
| CN114630820A (zh) | 3-硝基-n-(2,2,2-三氟乙基)-4-吡啶胺的合成 | |
| CN107304170A (zh) | 一种二聚物的制备方法 | |
| IL270542B (en) | Pyrazole amine reactive crystallization |