JP2021504418A5 - - Google Patents

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Publication number
JP2021504418A5
JP2021504418A5 JP2020529522A JP2020529522A JP2021504418A5 JP 2021504418 A5 JP2021504418 A5 JP 2021504418A5 JP 2020529522 A JP2020529522 A JP 2020529522A JP 2020529522 A JP2020529522 A JP 2020529522A JP 2021504418 A5 JP2021504418 A5 JP 2021504418A5
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JP
Japan
Prior art keywords
formula
methoxyisochroman
ethyl
carboxylate
ethanol
Prior art date
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Granted
Application number
JP2020529522A
Other languages
English (en)
Japanese (ja)
Other versions
JP7339946B2 (ja
JP2021504418A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/FI2018/050864 external-priority patent/WO2019106238A1/en
Publication of JP2021504418A publication Critical patent/JP2021504418A/ja
Publication of JP2021504418A5 publication Critical patent/JP2021504418A5/ja
Application granted granted Critical
Publication of JP7339946B2 publication Critical patent/JP7339946B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2020529522A 2017-12-01 2018-11-30 2-(5-メトキシイソクロマン-1-イル)-4,5-ジヒドロ-1h-イミダゾールおよびその硫酸水素塩の製造方法 Active JP7339946B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FI20176085 2017-12-01
FI20176085 2017-12-01
PCT/FI2018/050864 WO2019106238A1 (en) 2017-12-01 2018-11-30 Process for the preparation of 2-(5-methoxyisochroman-1 -yl)-4,5-dihydro-1 h-imidazole and the hydrogensulfate salt thereof

Publications (3)

Publication Number Publication Date
JP2021504418A JP2021504418A (ja) 2021-02-15
JP2021504418A5 true JP2021504418A5 (enExample) 2023-07-13
JP7339946B2 JP7339946B2 (ja) 2023-09-06

Family

ID=64746580

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020529522A Active JP7339946B2 (ja) 2017-12-01 2018-11-30 2-(5-メトキシイソクロマン-1-イル)-4,5-ジヒドロ-1h-イミダゾールおよびその硫酸水素塩の製造方法

Country Status (19)

Country Link
US (1) US11352346B2 (enExample)
EP (1) EP3717476B1 (enExample)
JP (1) JP7339946B2 (enExample)
KR (1) KR102718536B1 (enExample)
CN (1) CN111630049B (enExample)
AU (1) AU2018376872B2 (enExample)
BR (1) BR112020010617A2 (enExample)
CA (1) CA3083734A1 (enExample)
DK (1) DK3717476T3 (enExample)
ES (1) ES2927193T3 (enExample)
HR (1) HRP20221247T1 (enExample)
HU (1) HUE059849T2 (enExample)
IL (1) IL274931B2 (enExample)
LT (1) LT3717476T (enExample)
PL (1) PL3717476T3 (enExample)
PT (1) PT3717476T (enExample)
SI (1) SI3717476T1 (enExample)
WO (1) WO2019106238A1 (enExample)
ZA (1) ZA202003981B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021020935A1 (ko) 2019-07-31 2021-02-04 현대자동차주식회사 차량 내부 네트워크에 대한 sdn 기반의 침입 대응 방법 및 이를 이용한 시스템
AU2022236605A1 (en) * 2021-03-19 2023-11-02 Orion Corporation Tasipimidine formulations and use thereof
JP2025502480A (ja) 2022-01-24 2025-01-24 オリオン コーポレーション イソクロマン-イミダゾール構造のアルファ-2aアドレナリン受容体アゴニストの新規な硫酸塩形
AU2023215667A1 (en) 2022-02-04 2024-09-12 Orion Corporation Novel salt forms of isochroman-imidazole structured alpha-2a adrenoceptor agonist
JP2025531623A (ja) 2022-09-28 2025-09-22 オリオン コーポレーション タシピミジンおよびcyp2d6阻害薬の併用療法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6410562B1 (en) * 1998-12-18 2002-06-25 Eli Lilly And Company Hypoglycemic imidazoline compounds
AR090557A1 (es) * 2012-04-02 2014-11-19 Orion Corp DERIVADOS IMIDAZOLICOS AGONISTAS ADRENERGICOS a2

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