JP2021098728A5 - - Google Patents
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- JP2021098728A5 JP2021098728A5 JP2021037000A JP2021037000A JP2021098728A5 JP 2021098728 A5 JP2021098728 A5 JP 2021098728A5 JP 2021037000 A JP2021037000 A JP 2021037000A JP 2021037000 A JP2021037000 A JP 2021037000A JP 2021098728 A5 JP2021098728 A5 JP 2021098728A5
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- JP
- Japan
- Prior art keywords
- pharmaceutical composition
- pharmaceutically acceptable
- acceptable salt
- orally administered
- acceptable excipient
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 239000008194 pharmaceutical composition Substances 0.000 claims 10
- 239000000546 pharmaceutical excipient Substances 0.000 claims 3
- 150000003839 salts Chemical class 0.000 claims 3
- 206010028980 Neoplasm Diseases 0.000 claims 2
- 201000011510 cancer Diseases 0.000 claims 2
- 239000002246 antineoplastic agent Substances 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 229940127089 cytotoxic agent Drugs 0.000 claims 1
- 239000003814 drug Substances 0.000 claims 1
- 208000002154 non-small cell lung carcinoma Diseases 0.000 claims 1
- 229940124597 therapeutic agent Drugs 0.000 claims 1
- 230000001225 therapeutic effect Effects 0.000 claims 1
- 208000029729 tumor suppressor gene on chromosome 11 Diseases 0.000 claims 1
Claims (7)
- 患者におけるがんを処置するための、請求項1、2および3に記載の医薬組成物。
- 前記がんが、非小細胞肺がんである、請求項4に記載の医薬組成物。
- さらなる治療化合物と組み合わせて投与されることを特徴とする、請求項1~4に記載の医薬組成物。
- 前記さらなる治療剤が化学療法剤である、請求項6に記載の医薬組成物。
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2023032872A JP2023060145A (ja) | 2018-05-14 | 2023-03-03 | Mcl-1阻害剤 |
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201862671306P | 2018-05-14 | 2018-05-14 | |
US62/671,306 | 2018-05-14 | ||
US201862749918P | 2018-10-24 | 2018-10-24 | |
US62/749,918 | 2018-10-24 | ||
JP2020564228A JP6899975B2 (ja) | 2018-05-14 | 2019-05-13 | Mcl−1阻害剤 |
Related Parent Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2020564228A Division JP6899975B2 (ja) | 2018-05-14 | 2019-05-13 | Mcl−1阻害剤 |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2023032872A Division JP2023060145A (ja) | 2018-05-14 | 2023-03-03 | Mcl-1阻害剤 |
Publications (3)
Publication Number | Publication Date |
---|---|
JP2021098728A JP2021098728A (ja) | 2021-07-01 |
JP2021098728A5 true JP2021098728A5 (ja) | 2022-10-12 |
JP7240431B2 JP7240431B2 (ja) | 2023-03-15 |
Family
ID=66770559
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2020564228A Active JP6899975B2 (ja) | 2018-05-14 | 2019-05-13 | Mcl−1阻害剤 |
JP2021037000A Active JP7240431B2 (ja) | 2018-05-14 | 2021-03-09 | Mcl-1阻害剤 |
JP2023032872A Pending JP2023060145A (ja) | 2018-05-14 | 2023-03-03 | Mcl-1阻害剤 |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2020564228A Active JP6899975B2 (ja) | 2018-05-14 | 2019-05-13 | Mcl−1阻害剤 |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2023032872A Pending JP2023060145A (ja) | 2018-05-14 | 2023-03-03 | Mcl-1阻害剤 |
Country Status (29)
Country | Link |
---|---|
US (4) | US10703733B2 (ja) |
EP (2) | EP3793565B1 (ja) |
JP (3) | JP6899975B2 (ja) |
KR (1) | KR102551319B1 (ja) |
CN (2) | CN112118845B (ja) |
AU (3) | AU2019269391B2 (ja) |
BR (1) | BR112020021648A2 (ja) |
CA (1) | CA3099152C (ja) |
CL (1) | CL2020002919A1 (ja) |
CO (1) | CO2020014009A2 (ja) |
CR (1) | CR20200544A (ja) |
CY (1) | CY1125065T1 (ja) |
DK (1) | DK3793565T3 (ja) |
ES (1) | ES2907923T3 (ja) |
HR (1) | HRP20220215T1 (ja) |
HU (1) | HUE057852T2 (ja) |
IL (2) | IL291430B2 (ja) |
LT (1) | LT3793565T (ja) |
MX (1) | MX2020012137A (ja) |
PE (1) | PE20210004A1 (ja) |
PH (1) | PH12020551881A1 (ja) |
PL (1) | PL3793565T3 (ja) |
PT (1) | PT3793565T (ja) |
SG (1) | SG11202010964VA (ja) |
SI (1) | SI3793565T1 (ja) |
TW (2) | TWI719478B (ja) |
UA (1) | UA125163C2 (ja) |
WO (1) | WO2019222112A1 (ja) |
ZA (1) | ZA202007007B (ja) |
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KR20220085796A (ko) | 2019-10-18 | 2022-06-22 | 포티 세븐, 인코포레이티드 | 골수이형성 증후군 및 급성 골수성 백혈병을 치료하기 위한 조합 치료 |
CN114599392A (zh) | 2019-10-31 | 2022-06-07 | 四十七公司 | 基于抗cd47和抗cd20的血癌治疗 |
TWI778443B (zh) * | 2019-11-12 | 2022-09-21 | 美商基利科學股份有限公司 | Mcl1抑制劑 |
WO2021108254A1 (en) | 2019-11-26 | 2021-06-03 | Gilead Sciences, Inc. | Processes and intermediates for preparing mcl1 inhibitors |
KR20220131918A (ko) | 2019-12-24 | 2022-09-29 | 카나 바이오사이언스, 인코포레이션 | 다이아실글리세롤 키나제 조절 화합물 |
US20230212191A1 (en) * | 2020-04-16 | 2023-07-06 | Prelude Therapeutics, Incorporated | Spiro-sulfonimidamide derivatives as inhibitors of myeloid cell leukemia-1 (mcl-1) protein |
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CN116670141A (zh) | 2020-12-17 | 2023-08-29 | 詹森药业有限公司 | 作为mcl-1抑制剂的大环支化3-氟-丁-3-烯酰胺 |
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2019
- 2019-05-13 CA CA3099152A patent/CA3099152C/en active Active
- 2019-05-13 PE PE2020001829A patent/PE20210004A1/es unknown
- 2019-05-13 WO PCT/US2019/032053 patent/WO2019222112A1/en unknown
- 2019-05-13 JP JP2020564228A patent/JP6899975B2/ja active Active
- 2019-05-13 PT PT197287931T patent/PT3793565T/pt unknown
- 2019-05-13 BR BR112020021648-8A patent/BR112020021648A2/pt unknown
- 2019-05-13 AU AU2019269391A patent/AU2019269391B2/en active Active
- 2019-05-13 EP EP19728793.1A patent/EP3793565B1/en active Active
- 2019-05-13 CN CN201980032695.2A patent/CN112118845B/zh active Active
- 2019-05-13 MX MX2020012137A patent/MX2020012137A/es unknown
- 2019-05-13 ES ES19728793T patent/ES2907923T3/es active Active
- 2019-05-13 HU HUE19728793A patent/HUE057852T2/hu unknown
- 2019-05-13 UA UAA202006695A patent/UA125163C2/uk unknown
- 2019-05-13 LT LTEPPCT/US2019/032053T patent/LT3793565T/lt unknown
- 2019-05-13 US US16/410,457 patent/US10703733B2/en active Active
- 2019-05-13 DK DK19728793.1T patent/DK3793565T3/da active
- 2019-05-13 SG SG11202010964VA patent/SG11202010964VA/en unknown
- 2019-05-13 KR KR1020207035485A patent/KR102551319B1/ko active IP Right Grant
- 2019-05-13 EP EP21218221.6A patent/EP4029868A1/en active Pending
- 2019-05-13 CN CN202310897123.9A patent/CN117304130A/zh active Pending
- 2019-05-13 PL PL19728793T patent/PL3793565T3/pl unknown
- 2019-05-13 CR CR20200544A patent/CR20200544A/es unknown
- 2019-05-13 IL IL291430A patent/IL291430B2/en unknown
- 2019-05-13 SI SI201930181T patent/SI3793565T1/sl unknown
- 2019-05-13 HR HRP20220215TT patent/HRP20220215T1/hr unknown
- 2019-05-14 TW TW108116508A patent/TWI719478B/zh active
- 2019-05-14 TW TW110107128A patent/TWI813957B/zh active
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2020
- 2020-04-23 US US16/857,021 patent/US10988451B2/en active Active
- 2020-10-27 IL IL278336A patent/IL278336B/en unknown
- 2020-11-03 PH PH12020551881A patent/PH12020551881A1/en unknown
- 2020-11-10 CL CL2020002919A patent/CL2020002919A1/es unknown
- 2020-11-10 ZA ZA2020/07007A patent/ZA202007007B/en unknown
- 2020-11-10 CO CONC2020/0014009A patent/CO2020014009A2/es unknown
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2021
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