JP2020510664A5 - - Google Patents
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- JP2020510664A5 JP2020510664A5 JP2019547426A JP2019547426A JP2020510664A5 JP 2020510664 A5 JP2020510664 A5 JP 2020510664A5 JP 2019547426 A JP2019547426 A JP 2019547426A JP 2019547426 A JP2019547426 A JP 2019547426A JP 2020510664 A5 JP2020510664 A5 JP 2020510664A5
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022097012A JP7443425B2 (ja) | 2017-02-28 | 2022-06-16 | αｖβ６インテグリン阻害剤 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762464693P | 2017-02-28 | 2017-02-28 | |
| US62/464,693 | 2017-02-28 | ||
| PCT/US2018/019838 WO2018160521A2 (en) | 2017-02-28 | 2018-02-27 | Inhibitors of (alpha-v)(beta-6) integrin |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022097012A Division JP7443425B2 (ja) | 2017-02-28 | 2022-06-16 | αｖβ６インテグリン阻害剤 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020510664A JP2020510664A (ja) | 2020-04-09 |
| JP2020510664A5 true JP2020510664A5 (https=) | 2021-04-01 |
| JP7092784B2 JP7092784B2 (ja) | 2022-06-28 |
Family
ID=63245635
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019547426A Active JP7092784B2 (ja) | 2017-02-28 | 2018-02-27 | αｖβ６インテグリン阻害剤 |
| JP2022097012A Active JP7443425B2 (ja) | 2017-02-28 | 2022-06-16 | αｖβ６インテグリン阻害剤 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022097012A Active JP7443425B2 (ja) | 2017-02-28 | 2022-06-16 | αｖβ６インテグリン阻害剤 |
Country Status (16)
| Country | Link |
|---|---|
| US (5) | US11040955B2 (https=) |
| EP (2) | EP4159727B1 (https=) |
| JP (2) | JP7092784B2 (https=) |
| KR (2) | KR102605460B1 (https=) |
| CN (2) | CN116283977B (https=) |
| AR (2) | AR111009A1 (https=) |
| AU (4) | AU2018229275B2 (https=) |
| BR (1) | BR112019017929A2 (https=) |
| CA (1) | CA3054604A1 (https=) |
| IL (3) | IL316954A (https=) |
| MA (1) | MA47697A (https=) |
| MX (2) | MX394210B (https=) |
| RU (2) | RU2769702C2 (https=) |
| SG (1) | SG11201907820SA (https=) |
| TW (2) | TWI834321B (https=) |
| WO (1) | WO2018160521A2 (https=) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3509590A4 (en) | 2016-09-07 | 2020-12-02 | Pliant Therapeutics, Inc. | N-ACYL AMINO ACID COMPOUNDS AND METHODS OF USE |
| US10696672B2 (en) | 2016-12-23 | 2020-06-30 | Pliant Therapeutics, Inc. | Amino acid compounds and methods of use |
| MA52117A (fr) | 2017-02-28 | 2022-04-06 | Morphic Therapeutic Inc | Inhibiteurs de l'intégrine (alpha-v) (bêta-6) |
| MX394210B (es) | 2017-02-28 | 2025-03-04 | Morphic Therapeutic Inc | INHIBIDORES DE INTEGRINA AVß6. |
| FI3761980T3 (fi) | 2018-03-07 | 2024-02-21 | Pliant Therapeutics Inc | Aminohappoyhdisteitä ja käyttömenetelmiä |
| TWI841573B (zh) | 2018-06-27 | 2024-05-11 | 美商普萊恩醫療公司 | 具有未分支連接子之胺基酸化合物及使用方法 |
| WO2020047207A1 (en) * | 2018-08-29 | 2020-03-05 | Morphic Therapeutics, Inc. | Inhibitors of (alpha-v)(beta-6) integrin |
| SI3844162T1 (sl) * | 2018-08-29 | 2025-06-30 | Morphic Therapeutic, Inc. | Zaviralci integrina alfa v beta6 |
| WO2020047239A1 (en) | 2018-08-29 | 2020-03-05 | Morphic Therapeutic, Inc. | INHIBITING αV β6 INTEGRIN |
| WO2020047208A1 (en) | 2018-08-29 | 2020-03-05 | Morphic Therapeutic, Inc. | Inhibitors of (alpha-v)(beta-6) integrin |
| TW202028179A (zh) | 2018-10-08 | 2020-08-01 | 美商普萊恩醫療公司 | 胺基酸化合物及使用方法 |
| EP3873605B1 (en) | 2018-10-30 | 2024-10-23 | Gilead Sciences, Inc. | Compounds for inhibition of alpha4beta7 integrin |
| ES3013256T3 (en) | 2018-10-30 | 2025-04-11 | Gilead Sciences Inc | Imidazo[1,2-a]pyridine derivatives as alpha4beta7 integrin inhibitors for the treatment of inflammatory diseases |
| FI3873884T3 (fi) | 2018-10-30 | 2025-02-24 | Gilead Sciences Inc | 3-(kinolin-8-yyli)-1,4-dihydropyrido[3,4-d]pyrimidiini-2,4-dionijohdannaisia alfa-4-beta-7-integriinin estäjinä tulehdussairauksien hoidossa |
| JP7189368B2 (ja) | 2018-10-30 | 2022-12-13 | ギリアード サイエンシーズ， インコーポレイテッド | アルファ４ベータ７インテグリンの阻害のための化合物 |
| CN114173803A (zh) | 2019-04-08 | 2022-03-11 | 普利安特治疗公司 | 氨基酸化合物的剂型和方案 |
| WO2021030438A1 (en) | 2019-08-14 | 2021-02-18 | Gilead Sciences, Inc. | Compounds for inhibition of alpha 4 beta 7 integrin |
| TWI775182B (zh) * | 2019-10-16 | 2022-08-21 | 美商莫菲克醫療股份有限公司 | 抑制人類整合素αβ |
| CN111718250B (zh) * | 2020-06-28 | 2022-04-22 | 万华化学集团股份有限公司 | 一种制备r-香茅醛的方法 |
| EP4247472A4 (en) | 2020-11-19 | 2024-10-09 | Pliant Therapeutics, Inc. | INTEGRIN INHIBITORS AND USES THEREOF |
| JP2026506655A (ja) * | 2023-02-14 | 2026-02-25 | モーフィック セラピューティック，インコーポレイテッド | αｖβ８インテグリンの阻害 |
| JP2026506652A (ja) * | 2023-02-14 | 2026-02-25 | モーフィック セラピューティック，インコーポレイテッド | αｖβ８インテグリンの阻害 |
| WO2025106644A1 (en) * | 2023-11-15 | 2025-05-22 | Morphic Therapeutic, Inc. | Heterocyclic compounds as inhibitors of alpha-v beta-1 integrin |
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| US4522811A (en) | 1982-07-08 | 1985-06-11 | Syntex (U.S.A.) Inc. | Serial injection of muramyldipeptides and liposomes enhances the anti-infective activity of muramyldipeptides |
| DE4134467A1 (de) | 1991-10-18 | 1993-04-22 | Thomae Gmbh Dr K | Heterobiarylderivate, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung |
| TW221996B (https=) * | 1991-11-14 | 1994-04-01 | Glaxo Group Ltd | |
| AU3351293A (en) | 1992-01-21 | 1993-08-03 | Glaxo Group Limited | Piperidineacetic acid derivatives as inhibitors of fibrinogen-dependent blood platelet aggregation |
| DK0623615T3 (da) | 1993-05-01 | 1999-12-13 | Merck Patent Gmbh | Adhæsionsreceptor-antagonister |
| US6069143A (en) | 1994-12-20 | 2000-05-30 | Smithkline Beecham Corporation | Fibrinogen receptor antagonists |
| WO1997024122A1 (en) * | 1995-12-29 | 1997-07-10 | Smithkline Beecham Corporation | Vitronectin receptor antagonists |
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- 2018-02-27 EP EP22205911.5A patent/EP4159727B1/en active Active
- 2018-02-27 CN CN202310349794.1A patent/CN116283977B/zh active Active
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- 2018-02-27 WO PCT/US2018/019838 patent/WO2018160521A2/en not_active Ceased
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- 2018-02-27 EP EP18761396.3A patent/EP3589627A4/en not_active Withdrawn
- 2018-02-27 BR BR112019017929A patent/BR112019017929A2/pt not_active Application Discontinuation
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