JP2020510664A5 - - Google Patents
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- JP2020510664A5 JP2020510664A5 JP2019547426A JP2019547426A JP2020510664A5 JP 2020510664 A5 JP2020510664 A5 JP 2020510664A5 JP 2019547426 A JP2019547426 A JP 2019547426A JP 2019547426 A JP2019547426 A JP 2019547426A JP 2020510664 A5 JP2020510664 A5 JP 2020510664A5
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022097012A JP7443425B2 (ja) | 2017-02-28 | 2022-06-16 | αｖβ６インテグリン阻害剤 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762464693P | 2017-02-28 | 2017-02-28 | |
| US62/464,693 | 2017-02-28 | ||
| PCT/US2018/019838 WO2018160521A2 (en) | 2017-02-28 | 2018-02-27 | Inhibitors of (alpha-v)(beta-6) integrin |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022097012A Division JP7443425B2 (ja) | 2017-02-28 | 2022-06-16 | αｖβ６インテグリン阻害剤 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020510664A JP2020510664A (ja) | 2020-04-09 |
| JP2020510664A5 true JP2020510664A5 (enExample) | 2021-04-01 |
| JP7092784B2 JP7092784B2 (ja) | 2022-06-28 |
Family
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Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019547426A Active JP7092784B2 (ja) | 2017-02-28 | 2018-02-27 | αｖβ６インテグリン阻害剤 |
| JP2022097012A Active JP7443425B2 (ja) | 2017-02-28 | 2022-06-16 | αｖβ６インテグリン阻害剤 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022097012A Active JP7443425B2 (ja) | 2017-02-28 | 2022-06-16 | αｖβ６インテグリン阻害剤 |
Country Status (16)
| Country | Link |
|---|---|
| US (5) | US20180244648A1 (enExample) |
| EP (2) | EP3589627A4 (enExample) |
| JP (2) | JP7092784B2 (enExample) |
| KR (2) | KR102891803B1 (enExample) |
| CN (2) | CN110573499B (enExample) |
| AR (2) | AR111009A1 (enExample) |
| AU (3) | AU2018229275B2 (enExample) |
| BR (1) | BR112019017929A2 (enExample) |
| CA (1) | CA3054604A1 (enExample) |
| IL (3) | IL316954A (enExample) |
| MA (1) | MA47697A (enExample) |
| MX (2) | MX394210B (enExample) |
| RU (2) | RU2022108080A (enExample) |
| SG (1) | SG11201907820SA (enExample) |
| TW (2) | TW201835078A (enExample) |
| WO (1) | WO2018160521A2 (enExample) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2018049068A1 (en) | 2016-09-07 | 2018-03-15 | Pliant Therapeutics, Inc. | N-acyl amino acid compounds and methods of use |
| WO2018119087A1 (en) | 2016-12-23 | 2018-06-28 | Pliant Therapeutics, Inc. | Amino acid compounds and methods of use |
| MA52117A (fr) | 2017-02-28 | 2022-04-06 | Morphic Therapeutic Inc | Inhibiteurs de l'intégrine (alpha-v) (bêta-6) |
| TW201835078A (zh) | 2017-02-28 | 2018-10-01 | 美商萊築理公司 | αvβ6整合蛋白之抑制劑 |
| EP4509512A3 (en) | 2018-03-07 | 2025-04-09 | Pliant Therapeutics, Inc. | Amino acid compounds and methods of use |
| TWI841573B (zh) | 2018-06-27 | 2024-05-11 | 美商普萊恩醫療公司 | 具有未分支連接子之胺基酸化合物及使用方法 |
| ES3027421T3 (en) * | 2018-08-29 | 2025-06-13 | Morphic Therapeutic Inc | Inhibitors of (alpha-v)(beta-6) integrin |
| TWI835840B (zh) * | 2018-08-29 | 2024-03-21 | 美商莫菲克醫療股份有限公司 | αvβ6整合素之抑制劑 |
| WO2020047208A1 (en) * | 2018-08-29 | 2020-03-05 | Morphic Therapeutic, Inc. | Inhibitors of (alpha-v)(beta-6) integrin |
| MX2021002181A (es) * | 2018-08-29 | 2021-07-15 | Morphic Therapeutic Inc | Inhibicion de la integrina alfa v beta 6. |
| TW202028179A (zh) | 2018-10-08 | 2020-08-01 | 美商普萊恩醫療公司 | 胺基酸化合物及使用方法 |
| US11179383B2 (en) | 2018-10-30 | 2021-11-23 | Gilead Sciences, Inc. | Compounds for inhibition of α4β7 integrin |
| KR102630416B1 (ko) | 2018-10-30 | 2024-02-01 | 길리애드 사이언시즈, 인코포레이티드 | 알파4베타7 인테그린 억제제로서의 퀴놀린 유도체 |
| JP7189368B2 (ja) | 2018-10-30 | 2022-12-13 | ギリアード サイエンシーズ， インコーポレイテッド | アルファ４ベータ７インテグリンの阻害のための化合物 |
| WO2020092394A1 (en) | 2018-10-30 | 2020-05-07 | Gilead Sciences, Inc. | Imidazopyridine derivatives as alpha4beta7 integrin inhibitors |
| EP3952902A4 (en) | 2019-04-08 | 2022-12-21 | Pliant Therapeutics, Inc. | DOSAGE FORMS AND THERAPY SCHEMES FOR AMINO ACID COMPOUNDS |
| CN114222730B (zh) | 2019-08-14 | 2024-09-10 | 吉利德科学公司 | 用于抑制α4β7整合素的化合物 |
| TWI857592B (zh) * | 2019-10-16 | 2024-10-01 | 美商莫菲克醫療股份有限公司 | 抑制人類整合素α4β7 |
| CN111718250B (zh) * | 2020-06-28 | 2022-04-22 | 万华化学集团股份有限公司 | 一种制备r-香茅醛的方法 |
| MX2023005889A (es) | 2020-11-19 | 2023-06-06 | Pliant Therapeutics Inc | Inhibidor de integrina y usos de este. |
| CN120957721A (zh) * | 2023-02-14 | 2025-11-14 | 莫菲克医疗股份有限公司 | 抑制αvβ8整合素 |
| CN121127468A (zh) * | 2023-02-14 | 2025-12-12 | 莫菲克医疗股份有限公司 | 抑制αvβ8整合素 |
| WO2025106644A1 (en) * | 2023-11-15 | 2025-05-22 | Morphic Therapeutic, Inc. | Heterocyclic compounds as inhibitors of alpha-v beta-1 integrin |
Family Cites Families (97)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US4522811A (en) | 1982-07-08 | 1985-06-11 | Syntex (U.S.A.) Inc. | Serial injection of muramyldipeptides and liposomes enhances the anti-infective activity of muramyldipeptides |
| DE4134467A1 (de) | 1991-10-18 | 1993-04-22 | Thomae Gmbh Dr K | Heterobiarylderivate, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung |
| JPH07501063A (ja) * | 1991-11-14 | 1995-02-02 | グラクソ、グループ、リミテッド | フィブリノーゲン依存性血小板凝集阻害剤としてのピペリジン酢酸誘導体 |
| AU3351293A (en) | 1992-01-21 | 1993-08-03 | Glaxo Group Limited | Piperidineacetic acid derivatives as inhibitors of fibrinogen-dependent blood platelet aggregation |
| ATE181735T1 (de) | 1993-05-01 | 1999-07-15 | Merck Patent Gmbh | Substituierte 1-phenyl-oxazolidin-2-on derivate, deren herstellung und deren verwendung als adhäsionsrezeptor-antagonisten |
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- 2018-02-27 BR BR112019017929A patent/BR112019017929A2/pt not_active Application Discontinuation
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