JP2020505327A5 - - Google Patents
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- JP2020505327A5 JP2020505327A5 JP2019534368A JP2019534368A JP2020505327A5 JP 2020505327 A5 JP2020505327 A5 JP 2020505327A5 JP 2019534368 A JP2019534368 A JP 2019534368A JP 2019534368 A JP2019534368 A JP 2019534368A JP 2020505327 A5 JP2020505327 A5 JP 2020505327A5
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- Japan
- Prior art keywords
- alkyl
- substituted
- optionally substituted
- group
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- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- IYDMGGPKSVWQRT-XZWHSSHBSA-N CC(C)Oc(cc(cc1)OC)c1C(N([C@@H]1c(cc2)ccc2Cl)C(N(CC2)CCN2C(C)=O)=O)=N[C@H]1c(cc1)ccc1Cl Chemical compound CC(C)Oc(cc(cc1)OC)c1C(N([C@@H]1c(cc2)ccc2Cl)C(N(CC2)CCN2C(C)=O)=O)=N[C@H]1c(cc1)ccc1Cl IYDMGGPKSVWQRT-XZWHSSHBSA-N 0.000 description 1
- BDUHCSBCVGXTJM-WUFINQPMSA-N CC(C)Oc(cc(cc1)OC)c1C(N([C@@H]1c(cc2)ccc2Cl)C(N(CCN2)CC2=O)=O)=N[C@H]1c(cc1)ccc1Cl Chemical compound CC(C)Oc(cc(cc1)OC)c1C(N([C@@H]1c(cc2)ccc2Cl)C(N(CCN2)CC2=O)=O)=N[C@H]1c(cc1)ccc1Cl BDUHCSBCVGXTJM-WUFINQPMSA-N 0.000 description 1
- PVRYEWOXWGDQHA-UHFFFAOYSA-N CCOc1cc(OC)ccc1C(N(C1c(cc2)ccc2Br)C(N2CCN(CCO)CC2)=O)=NC1c(cc1)ccc1Br Chemical compound CCOc1cc(OC)ccc1C(N(C1c(cc2)ccc2Br)C(N2CCN(CCO)CC2)=O)=NC1c(cc1)ccc1Br PVRYEWOXWGDQHA-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662438901P | 2016-12-23 | 2016-12-23 | |
| US62/438,901 | 2016-12-23 | ||
| US201762563494P | 2017-09-26 | 2017-09-26 | |
| US62/563,494 | 2017-09-26 | ||
| PCT/US2017/068308 WO2018119441A1 (en) | 2016-12-23 | 2017-12-22 | Egfr proteolysis targeting chimeric molecules and associated methods of use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2020505327A JP2020505327A (ja) | 2020-02-20 |
| JP2020505327A5 true JP2020505327A5 (enExample) | 2021-02-04 |
Family
ID=62627537
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019534368A Pending JP2020505327A (ja) | 2016-12-23 | 2017-12-22 | Ｅｇｆｒタンパク質分解標的化キメラ分子およびその関連する使用方法 |
Country Status (13)
| Country | Link |
|---|---|
| US (3) | US10994015B2 (enExample) |
| EP (1) | EP3559002A4 (enExample) |
| JP (1) | JP2020505327A (enExample) |
| KR (1) | KR20190101406A (enExample) |
| CN (1) | CN110753693A (enExample) |
| AU (1) | AU2017382406A1 (enExample) |
| BR (1) | BR112019012682A2 (enExample) |
| CA (1) | CA3047586A1 (enExample) |
| CO (1) | CO2019007892A2 (enExample) |
| IL (1) | IL267398A (enExample) |
| MX (1) | MX2019007646A (enExample) |
| RU (1) | RU2019121527A (enExample) |
| WO (1) | WO2018119441A1 (enExample) |
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2017
- 2017-12-22 RU RU2019121527A patent/RU2019121527A/ru not_active Application Discontinuation
- 2017-12-22 WO PCT/US2017/068308 patent/WO2018119441A1/en not_active Ceased
- 2017-12-22 EP EP17884473.4A patent/EP3559002A4/en not_active Withdrawn
- 2017-12-22 MX MX2019007646A patent/MX2019007646A/es unknown
- 2017-12-22 CA CA3047586A patent/CA3047586A1/en not_active Abandoned
- 2017-12-22 AU AU2017382406A patent/AU2017382406A1/en not_active Abandoned
- 2017-12-22 JP JP2019534368A patent/JP2020505327A/ja active Pending
- 2017-12-22 US US15/852,854 patent/US10994015B2/en active Active
- 2017-12-22 CN CN201780087264.7A patent/CN110753693A/zh active Pending
- 2017-12-22 KR KR1020197021538A patent/KR20190101406A/ko not_active Ceased
- 2017-12-22 BR BR112019012682A patent/BR112019012682A2/pt not_active Application Discontinuation
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2019
- 2019-06-16 IL IL267398A patent/IL267398A/en unknown
- 2019-07-23 CO CONC2019/0007892A patent/CO2019007892A2/es unknown
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2021
- 2021-03-04 US US17/192,083 patent/US20210220475A1/en not_active Abandoned
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2024
- 2024-04-01 US US18/623,722 patent/US20240382599A1/en active Pending
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