JP2017506666A - 高インスリン血症に関連した症状の処置 - Google Patents

高インスリン血症に関連した症状の処置 Download PDF

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Publication number
JP2017506666A
JP2017506666A JP2016554661A JP2016554661A JP2017506666A JP 2017506666 A JP2017506666 A JP 2017506666A JP 2016554661 A JP2016554661 A JP 2016554661A JP 2016554661 A JP2016554661 A JP 2016554661A JP 2017506666 A JP2017506666 A JP 2017506666A
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alkyl
alkylene
aryl
heteroaryl
heterocycloalkyl
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JP2017506666A5 (enExample
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ランドー，スティーブン，ビー．
ケーギー，マイケル
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テンシャ セラピューティクス，インコーポレイテッド
テンシャ セラピューティクス，インコーポレイテッド
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
    • A61K31/5517—1,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones

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  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2016554661A 2014-02-28 2015-02-27 高インスリン血症に関連した症状の処置 Withdrawn JP2017506666A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201461946682P 2014-02-28 2014-02-28
US61/946,682 2014-02-28
US201462019777P 2014-07-01 2014-07-01
US62/019,777 2014-07-01
US201462054620P 2014-09-24 2014-09-24
US62/054,620 2014-09-24
PCT/US2015/018118 WO2015131113A1 (en) 2014-02-28 2015-02-27 Treatment of conditions associated with hyperinsulinaemia

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2018222642A Division JP6629947B2 (ja) 2014-02-28 2018-11-28 高インスリン血症に関連した症状の処置

Publications (2)

Publication Number Publication Date
JP2017506666A true JP2017506666A (ja) 2017-03-09
JP2017506666A5 JP2017506666A5 (enExample) 2018-02-22

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JP2016554661A Withdrawn JP2017506666A (ja) 2014-02-28 2015-02-27 高インスリン血症に関連した症状の処置
JP2018222642A Expired - Fee Related JP6629947B2 (ja) 2014-02-28 2018-11-28 高インスリン血症に関連した症状の処置

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Country Status (12)

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US (1) US10925881B2 (enExample)
EP (1) EP3110424A1 (enExample)
JP (2) JP2017506666A (enExample)
KR (1) KR20160130778A (enExample)
CN (1) CN106456653A (enExample)
AU (1) AU2015222805B2 (enExample)
CA (1) CA2940472A1 (enExample)
IL (1) IL247354B (enExample)
MX (1) MX377534B (enExample)
RU (1) RU2722179C2 (enExample)
SG (1) SG11201607108XA (enExample)
WO (1) WO2015131113A1 (enExample)

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JP2017504651A (ja) 2014-01-31 2017-02-09 ダナ−ファーバー キャンサー インスティテュート， インコーポレイテッド ジアゼパン誘導体の使用
KR20160115953A (ko) 2014-01-31 2016-10-06 다나-파버 캔서 인스티튜트 인크. 디아미노피리미딘 벤젠술폰 유도체 및 그의 용도
CN106456653A (zh) 2014-02-28 2017-02-22 腾沙治疗公司 高胰岛素血症相关病症的治疗
SG11201703414VA (en) 2014-10-27 2017-05-30 Tensha Therapeutics Inc Bromodomain inhibitors
MX2017016337A (es) 2015-06-26 2018-11-22 Tensha Therapeutics Inc Tratamiento de carcinoma de linea media nut.
PE20181287A1 (es) 2015-09-11 2018-08-07 Dana Farber Cancer Inst Inc Ciano tienotriazolpirazinas y usos de las mismas
HK1256419A1 (zh) 2015-09-11 2019-09-20 达纳-法伯癌症研究所股份有限公司 乙酰胺噻吩並三唑並二氮雜環庚三烯及其用途
SG10201913450PA (en) 2015-11-25 2020-03-30 Dana Farber Cancer Inst Inc Bivalent bromodomain inhibitors and uses thereof
KR20190092429A (ko) * 2016-12-16 2019-08-07 에프. 호프만-라 로슈 아게 다이아제핀 유도체의 제조 방법
WO2019052980A1 (en) 2017-09-14 2019-03-21 F. Hoffmann-La Roche Ag NOVEL COMPOUND FOR USE IN THE MANUFACTURE OF MEDICAMENTS
CN112312916A (zh) 2018-06-13 2021-02-02 戴布里股份公司 缩合三氮杂卓衍生物的制备及其作为bet抑制剂的用途
CN111253871A (zh) * 2020-03-13 2020-06-09 东莞市永益诚电子有限公司 一种钢化膜及其制备方法

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