JP2016533379A5 - - Google Patents

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JP2016533379A5
JP2016533379A5 JP2016524432A JP2016524432A JP2016533379A5 JP 2016533379 A5 JP2016533379 A5 JP 2016533379A5 JP 2016524432 A JP2016524432 A JP 2016524432A JP 2016524432 A JP2016524432 A JP 2016524432A JP 2016533379 A5 JP2016533379 A5 JP 2016533379A5
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optionally substituted
alkyl
substituted
composition
hydrogen
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JP2016524432A
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JP6491202B2 (ja
JP2016533379A (ja
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Priority claimed from PCT/US2014/061232 external-priority patent/WO2015058140A1/en
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JP2016524432A 2013-10-18 2014-10-17 サイクリン依存性キナーゼ7(cdk7)の多環阻害剤 Expired - Fee Related JP6491202B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361893005P 2013-10-18 2013-10-18
US61/893,005 2013-10-18
PCT/US2014/061232 WO2015058140A1 (en) 2013-10-18 2014-10-17 Polycyclic inhibitors of cyclin-dependent kinase 7 (cdk7)

Publications (3)

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JP2016533379A JP2016533379A (ja) 2016-10-27
JP2016533379A5 true JP2016533379A5 (OSRAM) 2017-11-24
JP6491202B2 JP6491202B2 (ja) 2019-03-27

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JP2016524432A Expired - Fee Related JP6491202B2 (ja) 2013-10-18 2014-10-17 サイクリン依存性キナーゼ7(cdk7)の多環阻害剤

Country Status (7)

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US (2) US10047070B2 (OSRAM)
EP (1) EP3057956B1 (OSRAM)
JP (1) JP6491202B2 (OSRAM)
CN (1) CN105849099B (OSRAM)
AU (2) AU2014337044A1 (OSRAM)
CA (1) CA2927920A1 (OSRAM)
WO (1) WO2015058140A1 (OSRAM)

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CN108348522A (zh) 2015-08-28 2018-07-31 诺华股份有限公司 含(a)周期素依赖性激酶4/6(cdk4/6)抑制剂lee011(=ribociclib)和(b)表皮生长因子受体(egfr)抑制剂厄洛替尼的药物组合,用于治疗或预防癌症
JP7028766B2 (ja) 2015-09-09 2022-03-02 ダナ-ファーバー キャンサー インスティテュート, インコーポレイテッド サイクリン依存性キナーゼの阻害剤

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