JP2016512243A5 - - Google Patents

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JP2016512243A5
JP2016512243A5 JP2016500154A JP2016500154A JP2016512243A5 JP 2016512243 A5 JP2016512243 A5 JP 2016512243A5 JP 2016500154 A JP2016500154 A JP 2016500154A JP 2016500154 A JP2016500154 A JP 2016500154A JP 2016512243 A5 JP2016512243 A5 JP 2016512243A5
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JP6479749B2 (ja
JP2016512243A (ja
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Priority claimed from PCT/US2014/000058 external-priority patent/WO2014149139A2/en
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JP2016500154A 2013-03-15 2014-03-17 トロンビン阻害剤としてのハロゲノピラゾール Active JP6479749B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361789358P 2013-03-15 2013-03-15
US61/789,358 2013-03-15
US201361899588P 2013-11-04 2013-11-04
US61/899,588 2013-11-04
PCT/US2014/000058 WO2014149139A2 (en) 2013-03-15 2014-03-17 Halogenopyrazoles as inhibitors of thrombin

Related Child Applications (1)

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JP2019019308A Division JP2019081782A (ja) 2013-03-15 2019-02-06 トロンビン阻害剤としてのハロゲノピラゾール

Publications (3)

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JP2016512243A JP2016512243A (ja) 2016-04-25
JP2016512243A5 true JP2016512243A5 (cg-RX-API-DMAC7.html) 2017-04-20
JP6479749B2 JP6479749B2 (ja) 2019-03-06

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ID=51538179

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JP2016500154A Active JP6479749B2 (ja) 2013-03-15 2014-03-17 トロンビン阻害剤としてのハロゲノピラゾール
JP2019019308A Pending JP2019081782A (ja) 2013-03-15 2019-02-06 トロンビン阻害剤としてのハロゲノピラゾール
JP2020103499A Pending JP2020158522A (ja) 2013-03-15 2020-06-16 トロンビン阻害剤としてのハロゲノピラゾール

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JP2019019308A Pending JP2019081782A (ja) 2013-03-15 2019-02-06 トロンビン阻害剤としてのハロゲノピラゾール
JP2020103499A Pending JP2020158522A (ja) 2013-03-15 2020-06-16 トロンビン阻害剤としてのハロゲノピラゾール

Country Status (16)

Country Link
US (2) US9951025B2 (cg-RX-API-DMAC7.html)
EP (1) EP2970141B1 (cg-RX-API-DMAC7.html)
JP (3) JP6479749B2 (cg-RX-API-DMAC7.html)
KR (1) KR20150130405A (cg-RX-API-DMAC7.html)
CN (2) CN105209440B (cg-RX-API-DMAC7.html)
AU (2) AU2014238478B2 (cg-RX-API-DMAC7.html)
BR (1) BR112015023214A8 (cg-RX-API-DMAC7.html)
CA (1) CA2902431A1 (cg-RX-API-DMAC7.html)
ES (1) ES2791749T3 (cg-RX-API-DMAC7.html)
HK (1) HK1214252A1 (cg-RX-API-DMAC7.html)
IL (1) IL240763B (cg-RX-API-DMAC7.html)
MX (1) MX373646B (cg-RX-API-DMAC7.html)
RU (1) RU2015144193A (cg-RX-API-DMAC7.html)
SG (2) SG10201707486XA (cg-RX-API-DMAC7.html)
WO (2) WO2014149139A2 (cg-RX-API-DMAC7.html)
ZA (1) ZA201506440B (cg-RX-API-DMAC7.html)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6479749B2 (ja) 2013-03-15 2019-03-06 ヴァーセオン コーポレイション トロンビン阻害剤としてのハロゲノピラゾール
BR112015022340A2 (pt) 2013-03-15 2017-07-18 Verseon Corp método para tratamento ou prevenção de uma doença ou distúrbio relacionado à calicreína em um sujeito, composto, e, composição farmacêutica
LT3261639T (lt) * 2015-02-27 2022-11-25 Verseon International Corporation Pakaitiniai pirazolo junginiai kaip serino proteazės inhibitoriai
KR20220004083A (ko) 2019-04-11 2022-01-11 앤지온 바이오메디카 코포레이션 (e)-3-[2-(2-티에닐)비닐]-1h-피라졸의 고체 형태
CN112062692A (zh) * 2019-06-11 2020-12-11 太仓市茜泾化工有限公司 一种乙氧甲叉氰基乙酸乙酯的制备方法
CN112986065B (zh) * 2021-02-08 2021-08-31 杭州同创医学检验实验室有限公司 一种用于血细胞分析仪的全血质控品及其制备方法

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