JP2014221801A5 - - Google Patents

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Publication number
JP2014221801A5
JP2014221801A5 JP2014142904A JP2014142904A JP2014221801A5 JP 2014221801 A5 JP2014221801 A5 JP 2014221801A5 JP 2014142904 A JP2014142904 A JP 2014142904A JP 2014142904 A JP2014142904 A JP 2014142904A JP 2014221801 A5 JP2014221801 A5 JP 2014221801A5
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JP
Japan
Prior art keywords
polypeptide
helix
enhanced
modified
helix polypeptide
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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JP2014142904A
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English (en)
Japanese (ja)
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JP6067626B2 (ja
JP2014221801A (ja
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Publication of JP2014221801A publication Critical patent/JP2014221801A/ja
Publication of JP2014221801A5 publication Critical patent/JP2014221801A5/ja
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Publication of JP6067626B2 publication Critical patent/JP6067626B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2014142904A 2008-09-22 2014-07-11 ペプチド模倣大環状分子 Expired - Fee Related JP6067626B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US9906308P 2008-09-22 2008-09-22
US61/099,063 2008-09-22

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2011528084A Division JP5711128B2 (ja) 2008-09-22 2009-09-22 ペプチド模倣大環状分子

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2016159624A Division JP2016190882A (ja) 2008-09-22 2016-08-16 ペプチド模倣大環状分子

Publications (3)

Publication Number Publication Date
JP2014221801A JP2014221801A (ja) 2014-11-27
JP2014221801A5 true JP2014221801A5 (enExample) 2015-09-10
JP6067626B2 JP6067626B2 (ja) 2017-01-25

Family

ID=41611441

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2011528084A Expired - Fee Related JP5711128B2 (ja) 2008-09-22 2009-09-22 ペプチド模倣大環状分子
JP2014142904A Expired - Fee Related JP6067626B2 (ja) 2008-09-22 2014-07-11 ペプチド模倣大環状分子
JP2016159624A Pending JP2016190882A (ja) 2008-09-22 2016-08-16 ペプチド模倣大環状分子

Family Applications Before (1)

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JP2011528084A Expired - Fee Related JP5711128B2 (ja) 2008-09-22 2009-09-22 ペプチド模倣大環状分子

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2016159624A Pending JP2016190882A (ja) 2008-09-22 2016-08-16 ペプチド模倣大環状分子

Country Status (10)

Country Link
US (5) US8524653B2 (enExample)
EP (1) EP2342222B1 (enExample)
JP (3) JP5711128B2 (enExample)
CN (1) CN102482336B (enExample)
AU (1) AU2009294877C1 (enExample)
BR (1) BRPI0918948A2 (enExample)
CA (1) CA2737922A1 (enExample)
ES (1) ES2666458T3 (enExample)
IL (1) IL211836A0 (enExample)
WO (1) WO2010034034A1 (enExample)

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NZ627528A (en) 2012-02-15 2016-05-27 Aileron Therapeutics Inc Peptidomimetic macrocycles
US9617309B2 (en) 2012-09-26 2017-04-11 President And Fellows Of Harvard College Proline-locked stapled peptides and uses thereof
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US10286078B2 (en) 2013-09-13 2019-05-14 The California Institute For Biomedical Research Modified therapeutic agents and compositions thereof
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JP2021506814A (ja) 2017-12-15 2021-02-22 デイナ ファーバー キャンサー インスティチュート，インコーポレイテッド 安定化ペプチドによって介在される標的タンパク質の分解
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US9163330B2 (en) 2009-07-13 2015-10-20 President And Fellows Of Harvard College Bifunctional stapled polypeptides and uses thereof
WO2011038049A1 (en) 2009-09-22 2011-03-31 Aileron Therapeutics, Inc. Peptidomimetic macrocycles
US20110223149A1 (en) 2009-10-14 2011-09-15 Aileron Therapeutics, Inc. Peptidomimetic macrocycles
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NZ627528A (en) 2012-02-15 2016-05-27 Aileron Therapeutics Inc Peptidomimetic macrocycles
HK1205454A1 (en) 2012-02-15 2015-12-18 Aileron Therapeutics, Inc. Triazole-crosslinked and thioether-crosslinked peptidomimetic macrocycles
SG11201503052RA (en) 2012-11-01 2015-05-28 Aileron Therapeutics Inc Disubstituted amino acids and methods of preparation and use thereof
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