JP2012503026A5 - - Google Patents

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Publication number
JP2012503026A5
JP2012503026A5 JP2011528084A JP2011528084A JP2012503026A5 JP 2012503026 A5 JP2012503026 A5 JP 2012503026A5 JP 2011528084 A JP2011528084 A JP 2011528084A JP 2011528084 A JP2011528084 A JP 2011528084A JP 2012503026 A5 JP2012503026 A5 JP 2012503026A5
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JP
Japan
Prior art keywords
polypeptide
enhanced
helix
helical
amino acid
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JP2011528084A
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English (en)
Japanese (ja)
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JP2012503026A (ja
JP5711128B2 (ja
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Priority claimed from PCT/US2009/057934 external-priority patent/WO2010034034A1/en
Publication of JP2012503026A publication Critical patent/JP2012503026A/ja
Publication of JP2012503026A5 publication Critical patent/JP2012503026A5/ja
Application granted granted Critical
Publication of JP5711128B2 publication Critical patent/JP5711128B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2011528084A 2008-09-22 2009-09-22 ペプチド模倣大環状分子 Expired - Fee Related JP5711128B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US9906308P 2008-09-22 2008-09-22
US61/099,063 2008-09-22
PCT/US2009/057934 WO2010034034A1 (en) 2008-09-22 2009-09-22 Peptidomimetic macrocycles

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014142904A Division JP6067626B2 (ja) 2008-09-22 2014-07-11 ペプチド模倣大環状分子

Publications (3)

Publication Number Publication Date
JP2012503026A JP2012503026A (ja) 2012-02-02
JP2012503026A5 true JP2012503026A5 (enExample) 2013-05-16
JP5711128B2 JP5711128B2 (ja) 2015-04-30

Family

ID=41611441

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2011528084A Expired - Fee Related JP5711128B2 (ja) 2008-09-22 2009-09-22 ペプチド模倣大環状分子
JP2014142904A Expired - Fee Related JP6067626B2 (ja) 2008-09-22 2014-07-11 ペプチド模倣大環状分子
JP2016159624A Pending JP2016190882A (ja) 2008-09-22 2016-08-16 ペプチド模倣大環状分子

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2014142904A Expired - Fee Related JP6067626B2 (ja) 2008-09-22 2014-07-11 ペプチド模倣大環状分子
JP2016159624A Pending JP2016190882A (ja) 2008-09-22 2016-08-16 ペプチド模倣大環状分子

Country Status (10)

Country Link
US (5) US8524653B2 (enExample)
EP (1) EP2342222B1 (enExample)
JP (3) JP5711128B2 (enExample)
CN (1) CN102482336B (enExample)
AU (1) AU2009294877C1 (enExample)
BR (1) BRPI0918948A2 (enExample)
CA (1) CA2737922A1 (enExample)
ES (1) ES2666458T3 (enExample)
IL (1) IL211836A0 (enExample)
WO (1) WO2010034034A1 (enExample)

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CA2774973A1 (en) 2009-09-22 2011-03-31 Aileron Therapeutics, Inc. Peptidomimetic macrocycles
BR112012008831A2 (pt) 2009-10-14 2019-09-24 Aileron Therapeutics Inc macrociclos de peptideomiméticos aprimorados.
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KR102112373B1 (ko) 2012-02-15 2020-05-18 에일러론 테라퓨틱스 인코포레이티드 펩티드모방체 마크로사이클
HK1205454A1 (en) 2012-02-15 2015-12-18 Aileron Therapeutics, Inc. Triazole-crosslinked and thioether-crosslinked peptidomimetic macrocycles
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