JP2010517990A5 - - Google Patents
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- Publication number
- JP2010517990A5 JP2010517990A5 JP2009547778A JP2009547778A JP2010517990A5 JP 2010517990 A5 JP2010517990 A5 JP 2010517990A5 JP 2009547778 A JP2009547778 A JP 2009547778A JP 2009547778 A JP2009547778 A JP 2009547778A JP 2010517990 A5 JP2010517990 A5 JP 2010517990A5
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- JP
- Japan
- Prior art keywords
- condition
- composition
- compound
- composition according
- salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- 150000001875 compounds Chemical class 0.000 claims 6
- 150000003839 salts Chemical class 0.000 claims 3
- 208000024827 Alzheimer disease Diseases 0.000 claims 2
- 201000004624 Dermatitis Diseases 0.000 claims 2
- 102000003676 Glucocorticoid Receptors Human genes 0.000 claims 2
- 108090000079 Glucocorticoid Receptors Proteins 0.000 claims 2
- 208000022559 Inflammatory bowel disease Diseases 0.000 claims 2
- 208000006673 asthma Diseases 0.000 claims 2
- 230000000694 effects Effects 0.000 claims 2
- 208000006545 Chronic Obstructive Pulmonary Disease Diseases 0.000 claims 1
- 206010061218 Inflammation Diseases 0.000 claims 1
- 208000028017 Psychotic disease Diseases 0.000 claims 1
- 206010052779 Transplant rejections Diseases 0.000 claims 1
- 206010046851 Uveitis Diseases 0.000 claims 1
- 159000000007 calcium salts Chemical class 0.000 claims 1
- 230000001684 chronic effect Effects 0.000 claims 1
- 230000004054 inflammatory process Effects 0.000 claims 1
- 208000024714 major depressive disease Diseases 0.000 claims 1
- 230000001404 mediated effect Effects 0.000 claims 1
- 201000006417 multiple sclerosis Diseases 0.000 claims 1
- 201000001119 neuropathy Diseases 0.000 claims 1
- 230000007823 neuropathy Effects 0.000 claims 1
- 208000033808 peripheral neuropathy Diseases 0.000 claims 1
- 206010039073 rheumatoid arthritis Diseases 0.000 claims 1
- 159000000000 sodium salts Chemical class 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US88798107P | 2007-02-02 | 2007-02-02 | |
| PCT/IB2008/000229 WO2008093227A1 (en) | 2007-02-02 | 2008-01-25 | Tricyclic compounds and their use as glucocorticoid receptor modulators |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010517990A JP2010517990A (ja) | 2010-05-27 |
| JP2010517990A5 true JP2010517990A5 (enExample) | 2010-08-12 |
| JP4599462B2 JP4599462B2 (ja) | 2010-12-15 |
Family
ID=39315208
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009547778A Expired - Fee Related JP4599462B2 (ja) | 2007-02-02 | 2008-01-25 | 三環式化合物およびそれらのグルココルチコイド受容体調節剤としての使用 |
Country Status (42)
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE69722426T3 (de) | 1996-07-24 | 2015-05-07 | Warner-Lambert Company LLC (n.Ges. des Staates Delaware) | Isobutylgaba und dessen derivate zur schmerzbehandlung |
| MY153057A (en) * | 2007-02-02 | 2014-12-31 | Pfizer Prod Inc | Tryclic compounds,compositions and methods |
| CN102112446B (zh) * | 2008-07-28 | 2012-10-31 | 美国辉瑞有限公司 | 菲酮化合物、组合物及方法 |
| US8765787B2 (en) * | 2008-11-21 | 2014-07-01 | Bridge Pharma, Inc. | Methods of treatment of xerophthalmia with self-preserving ocular formulations of norketotifen |
| US20100136095A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Systems for modulating inflammation |
| US20100137246A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Anti-inflammatory compositions and methods |
| US20100136094A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Systems for modulating inflammation |
| US20100136096A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Systems for modulating inflammation |
| US20100137844A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Delivery devices for modulating inflammation |
| US20100135983A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Anti-inflammatory compositions and methods |
| US20100136097A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Systems for modulating inflammation |
| AU2011251622A1 (en) | 2010-05-10 | 2012-12-20 | Radikal Therapeutics Inc. | Lipoic acid and nitroxide derivatives and uses thereof |
| BR112013004322A2 (pt) * | 2010-08-27 | 2016-06-21 | Corcept Therapeutics Inc | moduladores de azadecalin fundidos com piridil-aminas |
| US20120238549A1 (en) * | 2011-03-15 | 2012-09-20 | Abbott Laboratories | Nuclear Hormone Receptor Modulators |
| US8545904B1 (en) | 2012-06-05 | 2013-10-01 | Liquid Innovators, LLC | Topical composition containing Carapa (andiroba) oil for psoriasis and other related dermatological disorders |
| US9227901B2 (en) | 2012-07-05 | 2016-01-05 | Abbvie Inc. | Process for preparing bicyclic amine derivatives |
| TW201422590A (zh) | 2012-09-07 | 2014-06-16 | Abbvie Inc | 雜環核激素受體調節劑 |
| WO2014094357A1 (en) | 2012-12-21 | 2014-06-26 | Abbvie Inc. | Heterocyclic nuclear hormone receptor modulators |
| GB2525793B (en) | 2014-05-16 | 2016-11-02 | Liqwd Inc | Keratin treatment formulations and methods |
| US9597284B2 (en) * | 2014-10-20 | 2017-03-21 | Oyster Point Pharma, Inc. | Dry eye treatments |
| CN104591988A (zh) * | 2014-12-29 | 2015-05-06 | 甘肃省化工研究院 | 6-溴-2-萘满酮的合成方法 |
| CN107847480B (zh) | 2015-03-23 | 2021-06-25 | 墨尔本大学 | 呼吸性疾病的治疗 |
| TWI790997B (zh) | 2016-04-07 | 2023-02-01 | 美商奧伊斯特普安生物製藥公司 | 醫療調配物用於治療眼部病狀之用途 |
| WO2020093098A1 (en) | 2018-11-07 | 2020-05-14 | The University Of Melbourne | Novel compounds for the treatment of respiratory diseases |
Family Cites Families (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2576025B1 (fr) | 1985-01-14 | 1987-01-23 | Roussel Uclaf | Nouveaux steroides substitues en position 10, leur procede et les intermediaires de preparation, leur application comme medicaments, les compositions pharmaceutiques les contenant |
| FR2600450B1 (fr) * | 1986-06-19 | 1988-08-26 | Pechiney Aluminium | Procede de marquage individuel des anodes precuites pour la production electrolytique d'aluminium |
| GB9518953D0 (en) | 1995-09-15 | 1995-11-15 | Pfizer Ltd | Pharmaceutical formulations |
| IL122740A (en) | 1997-01-15 | 2003-09-17 | Akzo Nobel Nv | 16-hydroxy-11-(substituted phenyl)-estra-9,4-diene derivatives, their preparation and pharmaceutical compositions containing them |
| EA007483B1 (ru) * | 1999-04-30 | 2006-10-27 | Пфайзер Продактс Инк. | Применение модулятора рецепторов глюкокортикоидов и агониста рецепторов глюкокортикоидов при получении лекарственного средства |
| WO2001005229A1 (en) | 1999-07-15 | 2001-01-25 | The General Hospital Corporation | Non-defective epstein-barr viral vector |
| IL146057A (en) * | 2000-10-27 | 2007-09-20 | Pfizer Prod Inc | A process for the preparation of modulators of a non-steroidal glucocorticoid receptor |
| ATE327974T1 (de) * | 2000-10-28 | 2006-06-15 | Pfizer Prod Inc | Modulatoren des glucocorticoid-rezeptors |
| ES2246292T3 (es) | 2000-10-30 | 2006-02-16 | Pfizer Products Inc. | Moduladores de receptor glucocorticoide. |
| WO2002042995A1 (en) * | 2000-11-20 | 2002-05-30 | Seagate Technology Llc | Rf id tag attachment to a disc drive |
| WO2003000226A2 (en) | 2001-06-22 | 2003-01-03 | Pfizer Products Inc. | Pharmaceutical compositions containing polymer and drug assemblies |
| NZ531477A (en) | 2001-08-31 | 2006-10-27 | Corcept Therapeutics Inc | Use of a glucocorticoid receptor antagonist comprising a steroidal skeleton with at least one phenyl-containing moiety in the 11-beta position of the steroidal skeleton to decrease cognitive deterioration in adults with Down's syndrome |
| RU2309148C2 (ru) | 2001-09-27 | 2007-10-27 | Юниверсите Де Льеж | Производные пиридинсульфонамида, фармацевтическая композиция на их основе и применение |
| DE10164366C1 (de) * | 2001-12-28 | 2003-06-05 | Rehau Ag & Co | Permanentkathode |
| EP1469832B2 (en) | 2002-02-01 | 2016-10-26 | Bend Research, Inc. | Pharmaceutical compositions of amorphous dispersions of drugs and lipophilic microphase-forming materials |
| US8476254B2 (en) | 2002-07-02 | 2013-07-02 | Corcept Therapeutics, Inc. | Methods for treating psychosis associated with interferson-α therapy |
| MXPA05000345A (es) | 2002-07-08 | 2005-03-31 | Pfizer Prod Inc | Moduladores del receptor de glucocorticoides. |
| JP2006508951A (ja) | 2002-11-05 | 2006-03-16 | コーセプト セラピューティクス， インコーポレイテッド | 片頭痛を処置するための方法 |
| CA2514966A1 (en) | 2003-02-04 | 2004-08-19 | Corcept Therapeutics, Inc. | Antiglucocorticoids for the treatment of postpartum psychosis |
| US20050080061A1 (en) | 2003-07-23 | 2005-04-14 | Corcept Therapeutics, Inc. | Antiglucocorticoid therapy for the prevention of neurological damage in premature infants |
| US8097606B2 (en) | 2003-07-23 | 2012-01-17 | Corcept Therapeutics, Inc. | Antiglucocorticoids for the treatment of catatonia |
| TW200512181A (en) | 2003-09-26 | 2005-04-01 | Tanabe Seiyaku Co | Amide-type carboxamide derivatives |
| WO2005047524A2 (en) * | 2003-11-10 | 2005-05-26 | The Scripps Research Institute | Compositions and methods for inducing cell dedifferentiation |
| AU2004289532A1 (en) * | 2003-11-13 | 2005-05-26 | Pfizer Products Inc. | Octahydrophenanthrene hydrazinde derivatives useful as glucocorticoid receptor modulators |
| TWI370129B (en) | 2005-02-14 | 2012-08-11 | Msd Oss Bv | Non steroidal glucocorticoid receptor modulators |
| EP2012796A4 (en) | 2006-05-02 | 2010-08-11 | Corcept Therapeutics Inc | USE OF GLUCOCORTICOID TYPE II RECEPTOR ANTAGONISTS TO TREAT PATIENT DEPRESSION WITH IL-2 |
| MY153057A (en) * | 2007-02-02 | 2014-12-31 | Pfizer Prod Inc | Tryclic compounds,compositions and methods |
| PL2114888T3 (pl) * | 2007-02-02 | 2011-04-29 | Pfizer Prod Inc | Związki trójcykliczne i ich zastosowanie jako modulatorów receptora glukokortykoidowego |
-
2008
- 2008-01-25 MY MYPI20123293 patent/MY153057A/en unknown
- 2008-01-25 GE GEAP200811399A patent/GEP20125404B/en unknown
- 2008-01-25 UA UAA200907728A patent/UA94639C2/ru unknown
- 2008-01-25 MY MYPI20093089A patent/MY146087A/en unknown
- 2008-01-25 HR HR20110702T patent/HRP20110702T1/hr unknown
- 2008-01-25 SI SI200830393T patent/SI2114970T1/sl unknown
- 2008-01-25 RS RS20110429A patent/RS51970B/sr unknown
- 2008-01-25 BR BRPI0808634-6A patent/BRPI0808634A2/pt not_active IP Right Cessation
- 2008-01-25 ES ES08702351T patent/ES2368286T3/es active Active
- 2008-01-25 NZ NZ578638A patent/NZ578638A/en not_active IP Right Cessation
- 2008-01-25 AU AU2008211613A patent/AU2008211613B2/en not_active Ceased
- 2008-01-25 PL PL08702351T patent/PL2114970T3/pl unknown
- 2008-01-25 MX MX2009008284A patent/MX2009008284A/es active IP Right Grant
- 2008-01-25 EA EA200970666A patent/EA016494B1/ru not_active IP Right Cessation
- 2008-01-25 AT AT08702351T patent/ATE518872T1/de active
- 2008-01-25 CN CN2008800052954A patent/CN101616925B/zh not_active Expired - Fee Related
- 2008-01-25 EP EP08702351A patent/EP2114970B1/en active Active
- 2008-01-25 JP JP2009547778A patent/JP4599462B2/ja not_active Expired - Fee Related
- 2008-01-25 PT PT08702351T patent/PT2114970E/pt unknown
- 2008-01-25 KR KR1020097018289A patent/KR101107949B1/ko not_active Expired - Fee Related
- 2008-01-25 AP AP2009004942A patent/AP2455A/xx active
- 2008-01-25 DK DK08702351.1T patent/DK2114970T3/da active
- 2008-01-25 CA CA2676670A patent/CA2676670C/en not_active Expired - Fee Related
- 2008-01-25 WO PCT/IB2008/000229 patent/WO2008093227A1/en not_active Ceased
- 2008-01-28 KR KR1020097018294A patent/KR101114682B1/ko not_active Expired - Fee Related
- 2008-01-28 CN CN2008800056527A patent/CN101616896B/zh not_active Expired - Fee Related
- 2008-01-28 UA UAA200907730A patent/UA95332C2/uk unknown
- 2008-01-28 MY MYPI20093135A patent/MY148780A/en unknown
- 2008-01-28 GE GEAP200811398A patent/GEP20125426B/en unknown
- 2008-01-28 RS RS20110008A patent/RS51646B/sr unknown
- 2008-01-28 PT PT08702358T patent/PT2114888E/pt unknown
- 2008-01-28 ES ES08702358T patent/ES2353822T3/es active Active
- 2008-01-31 PE PE2008000231A patent/PE20081736A1/es not_active Application Discontinuation
- 2008-01-31 US US12/023,362 patent/US7598231B2/en not_active Expired - Fee Related
- 2008-01-31 US US12/023,323 patent/US7547714B2/en not_active Expired - Fee Related
- 2008-02-01 HN HN2008000179A patent/HN2008000179A/es unknown
- 2008-02-01 HN HN2008000178A patent/HN2008000178A/es unknown
- 2008-02-01 PE PE2008000234A patent/PE20090113A1/es not_active Application Discontinuation
- 2008-02-01 TW TW097104089A patent/TWI347842B/zh active
- 2008-02-01 AR ARP080100425A patent/AR065135A1/es active IP Right Grant
- 2008-02-01 CL CL200800330A patent/CL2008000330A1/es unknown
- 2008-02-01 AR ARP080100424A patent/AR065134A1/es active IP Right Grant
- 2008-02-01 CL CL200800329A patent/CL2008000329A1/es unknown
- 2008-02-01 TW TW097104074A patent/TWI373466B/zh not_active IP Right Cessation
-
2009
- 2009-05-08 US US12/437,704 patent/US8158660B2/en not_active Expired - Fee Related
- 2009-07-20 IL IL199972A patent/IL199972A/en active IP Right Grant
- 2009-07-21 US US12/506,825 patent/US7786097B2/en not_active Expired - Fee Related
- 2009-07-23 CR CR10949A patent/CR10949A/es not_active IP Right Cessation
- 2009-07-23 CR CR10948A patent/CR10948A/es not_active IP Right Cessation
- 2009-07-24 CU CU2009000132A patent/CU23848B1/es active IP Right Grant
- 2009-07-24 CU CU20090133A patent/CU20090133A7/es active IP Right Grant
- 2009-07-29 DO DO2009000190A patent/DOP2009000190A/es unknown
- 2009-07-29 NI NI200900149A patent/NI200900149A/es unknown
- 2009-07-29 NI NI200900148A patent/NI200900148A/es unknown
- 2009-07-30 GT GT200900209A patent/GT200900209A/es unknown
- 2009-07-30 GT GT200900210A patent/GT200900210A/es unknown
- 2009-07-30 SV SV2009003346A patent/SV2009003346A/es not_active Application Discontinuation
- 2009-07-31 MA MA32127A patent/MA31117B1/fr unknown
- 2009-07-31 EC EC2009009552A patent/ECSP099552A/es unknown
- 2009-07-31 TN TNP2009000324A patent/TN2009000324A1/fr unknown
- 2009-07-31 MA MA32128A patent/MA31158B1/fr unknown
- 2009-07-31 SV SV2009003349A patent/SV2009003349A/es active IP Right Grant
- 2009-07-31 EC EC2009009553A patent/ECSP099553A/es unknown
- 2009-07-31 CO CO09079796A patent/CO6190603A2/es active IP Right Grant
- 2009-07-31 CO CO09079789A patent/CO6220937A2/es active IP Right Grant
- 2009-09-01 ZA ZA200906064A patent/ZA200906064B/xx unknown
- 2009-09-01 ZA ZA200906060A patent/ZA200906060B/xx unknown
-
2010
- 2010-12-02 CY CY20101101109T patent/CY1110962T1/el unknown
-
2011
- 2011-08-17 CY CY20111100784T patent/CY1111758T1/el unknown
- 2011-12-21 US US13/333,104 patent/US8445520B2/en not_active Expired - Fee Related
-
2013
- 2013-04-16 US US13/863,534 patent/US20140142316A1/en not_active Abandoned
-
2014
- 2014-07-01 US US14/320,674 patent/US8901310B2/en not_active Expired - Fee Related
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