JP2010517990A5 - - Google Patents
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- Publication number
- JP2010517990A5 JP2010517990A5 JP2009547778A JP2009547778A JP2010517990A5 JP 2010517990 A5 JP2010517990 A5 JP 2010517990A5 JP 2009547778 A JP2009547778 A JP 2009547778A JP 2009547778 A JP2009547778 A JP 2009547778A JP 2010517990 A5 JP2010517990 A5 JP 2010517990A5
- Authority
- JP
- Japan
- Prior art keywords
- condition
- composition
- compound
- composition according
- salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
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- 150000001875 compounds Chemical class 0.000 claims 6
- 150000003839 salts Chemical class 0.000 claims 3
- 208000024827 Alzheimer disease Diseases 0.000 claims 2
- 201000004624 Dermatitis Diseases 0.000 claims 2
- 102000003676 Glucocorticoid Receptors Human genes 0.000 claims 2
- 108090000079 Glucocorticoid Receptors Proteins 0.000 claims 2
- 208000022559 Inflammatory bowel disease Diseases 0.000 claims 2
- 208000006673 asthma Diseases 0.000 claims 2
- 230000000694 effects Effects 0.000 claims 2
- 208000006545 Chronic Obstructive Pulmonary Disease Diseases 0.000 claims 1
- 206010061218 Inflammation Diseases 0.000 claims 1
- 208000028017 Psychotic disease Diseases 0.000 claims 1
- 206010052779 Transplant rejections Diseases 0.000 claims 1
- 206010046851 Uveitis Diseases 0.000 claims 1
- 159000000007 calcium salts Chemical class 0.000 claims 1
- 230000001684 chronic effect Effects 0.000 claims 1
- 230000004054 inflammatory process Effects 0.000 claims 1
- 208000024714 major depressive disease Diseases 0.000 claims 1
- 230000001404 mediated effect Effects 0.000 claims 1
- 201000006417 multiple sclerosis Diseases 0.000 claims 1
- 201000001119 neuropathy Diseases 0.000 claims 1
- 230000007823 neuropathy Effects 0.000 claims 1
- 208000033808 peripheral neuropathy Diseases 0.000 claims 1
- 206010039073 rheumatoid arthritis Diseases 0.000 claims 1
- 159000000000 sodium salts Chemical class 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US88798107P | 2007-02-02 | 2007-02-02 | |
| PCT/IB2008/000229 WO2008093227A1 (en) | 2007-02-02 | 2008-01-25 | Tricyclic compounds and their use as glucocorticoid receptor modulators |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2010517990A JP2010517990A (ja) | 2010-05-27 |
| JP2010517990A5 true JP2010517990A5 (enExample) | 2010-08-12 |
| JP4599462B2 JP4599462B2 (ja) | 2010-12-15 |
Family
ID=39315208
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009547778A Expired - Fee Related JP4599462B2 (ja) | 2007-02-02 | 2008-01-25 | 三環式化合物およびそれらのグルココルチコイド受容体調節剤としての使用 |
Country Status (42)
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6001876A (en) | 1996-07-24 | 1999-12-14 | Warner-Lambert Company | Isobutylgaba and its derivatives for the treatment of pain |
| DK2114970T3 (da) | 2007-02-02 | 2011-09-19 | Pfizer Prod Inc | Tricykliske forbindelser og deres anvendelse som glucocorticoidreceptormodulatorer |
| PE20110559A1 (es) * | 2008-07-28 | 2011-08-06 | Pfizer | (4bR,6R,7R,8aS)-4b-BENCIL-6,7-DIHIDROXI-6-METIL-N-(2-METILPIRIDIN-3-IL)-10-OXO-7-FENIL-4b,5,6,7,8,8a,9,10-OCTAHIDROFENANTRENO-2-CARBOXAMIDA COMO MODULADOR DEL RECEPTOR GLUCOCORTICOIDE |
| WO2010059894A1 (en) * | 2008-11-21 | 2010-05-27 | Bridge Pharma, Inc. | Ocular formulations of norketotifen |
| US20100137246A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Anti-inflammatory compositions and methods |
| US20100135983A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Anti-inflammatory compositions and methods |
| US20100136094A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Systems for modulating inflammation |
| US20100137787A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Delivery devices for modulating inflammation |
| US20100136096A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Systems for modulating inflammation |
| US20100136097A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Systems for modulating inflammation |
| US20100136095A1 (en) * | 2008-12-02 | 2010-06-03 | Searete Llc, A Limited Liability Corporation Of The State Of Delaware | Systems for modulating inflammation |
| WO2011141909A2 (en) | 2010-05-10 | 2011-11-17 | Radikal Therapeutics Inc. | Lipoic acid and nitroxide derivatives and uses thereof |
| CA2806900A1 (en) * | 2010-08-27 | 2012-03-01 | Corcept Therapeutics, Inc. | Pyridyl-amine fused azadecalin modulators |
| RU2013145912A (ru) * | 2011-03-15 | 2015-04-20 | Эббви Инк. | Модуляторы ядерных рецепторов гормонов |
| US8545904B1 (en) | 2012-06-05 | 2013-10-01 | Liquid Innovators, LLC | Topical composition containing Carapa (andiroba) oil for psoriasis and other related dermatological disorders |
| US9227901B2 (en) * | 2012-07-05 | 2016-01-05 | Abbvie Inc. | Process for preparing bicyclic amine derivatives |
| TW201422590A (zh) | 2012-09-07 | 2014-06-16 | Abbvie Inc | 雜環核激素受體調節劑 |
| WO2014094357A1 (en) | 2012-12-21 | 2014-06-26 | Abbvie Inc. | Heterocyclic nuclear hormone receptor modulators |
| EP3769749A1 (en) | 2014-05-16 | 2021-01-27 | Olaplex, Inc. | Keratin treatment formulations and methods |
| IL293188B2 (en) | 2014-10-20 | 2025-06-01 | Oyster Point Pharma Inc | The compound varenicline for use as a medicament for treating dry eye, increasing tear production and treating ocular discomfort, and a pharmaceutical formulation comprising varenicline |
| CN104591988A (zh) * | 2014-12-29 | 2015-05-06 | 甘肃省化工研究院 | 6-溴-2-萘满酮的合成方法 |
| US10722513B2 (en) | 2015-03-23 | 2020-07-28 | The University Of Melbourne | Treatment of respiratory diseases |
| US10709707B2 (en) | 2016-04-07 | 2020-07-14 | Oyster Point Pharma, Inc. | Methods of treating ocular conditions |
| AU2019374731B2 (en) | 2018-11-07 | 2025-08-21 | Tianli Biotech Pty Ltd | Compounds and compositions for the treatment of respiratory diseases |
Family Cites Families (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2576025B1 (fr) | 1985-01-14 | 1987-01-23 | Roussel Uclaf | Nouveaux steroides substitues en position 10, leur procede et les intermediaires de preparation, leur application comme medicaments, les compositions pharmaceutiques les contenant |
| FR2600450B1 (fr) * | 1986-06-19 | 1988-08-26 | Pechiney Aluminium | Procede de marquage individuel des anodes precuites pour la production electrolytique d'aluminium |
| GB9518953D0 (en) | 1995-09-15 | 1995-11-15 | Pfizer Ltd | Pharmaceutical formulations |
| IL122740A (en) | 1997-01-15 | 2003-09-17 | Akzo Nobel Nv | 16-hydroxy-11-(substituted phenyl)-estra-9,4-diene derivatives, their preparation and pharmaceutical compositions containing them |
| JP3901945B2 (ja) * | 1999-04-30 | 2007-04-04 | ファイザー・プロダクツ・インク | グルココルチコイド受容体モジュレーター |
| WO2001005229A1 (en) | 1999-07-15 | 2001-01-25 | The General Hospital Corporation | Non-defective epstein-barr viral vector |
| IL146057A (en) * | 2000-10-27 | 2007-09-20 | Pfizer Prod Inc | A process for the preparation of modulators of a non-steroidal glucocorticoid receptor |
| DE60120077T2 (de) | 2000-10-28 | 2006-11-02 | Pfizer Products Inc., Groton | Modulatoren des Glucocorticoid-Rezeptors |
| ATE303369T1 (de) | 2000-10-30 | 2005-09-15 | Pfizer Prod Inc | Glucocorticoid rezeptor modulatoren |
| GB2387468B (en) * | 2000-11-20 | 2005-01-19 | Seagate Technology Llc | RF ID Tag attachment to a disc drive |
| EP1401399A2 (en) | 2001-06-22 | 2004-03-31 | Pfizer Products Inc. | Pharmaceutical compositions containing polymer and drug assemblies |
| DE60229411D1 (de) | 2001-08-31 | 2008-11-27 | Corcept Therapeutics Inc | Verfahren zur hemmung der verschlechterung der kognitiven leistungsfähigkeit bei erwachsenen mit down-syndrom |
| RU2309148C2 (ru) | 2001-09-27 | 2007-10-27 | Юниверсите Де Льеж | Производные пиридинсульфонамида, фармацевтическая композиция на их основе и применение |
| DE10164366C1 (de) * | 2001-12-28 | 2003-06-05 | Rehau Ag & Co | Permanentkathode |
| ATE395044T1 (de) | 2002-02-01 | 2008-05-15 | Pfizer Prod Inc | Pharmazeutische zusammensetzungen amorpher dispersionen von wirkstoffen und lipophiler mikrophasenbildender materialien |
| CN1665515A (zh) | 2002-07-02 | 2005-09-07 | 科塞普特治疗公司 | 治疗与干扰素α治疗相关的精神病的方法 |
| AU2003281355A1 (en) | 2002-07-08 | 2004-01-23 | Pfizer Products Inc. | Modulators of the glucocorticoid receptor |
| EP1567167A4 (en) | 2002-11-05 | 2007-09-12 | Corcept Therapeutics Inc | METHODS FOR TREATING GASTRO-OESOPHAGEAL REFLUX PATHOLOGICAL |
| AU2004208842B2 (en) | 2003-02-04 | 2009-05-28 | Corcept Therapeutics, Inc. | Antiglucocorticoids for the treatment of postpartum psychosis |
| US20050080061A1 (en) | 2003-07-23 | 2005-04-14 | Corcept Therapeutics, Inc. | Antiglucocorticoid therapy for the prevention of neurological damage in premature infants |
| US8097606B2 (en) | 2003-07-23 | 2012-01-17 | Corcept Therapeutics, Inc. | Antiglucocorticoids for the treatment of catatonia |
| TW200512181A (en) | 2003-09-26 | 2005-04-01 | Tanabe Seiyaku Co | Amide-type carboxamide derivatives |
| ES2398239T3 (es) * | 2003-11-10 | 2013-03-14 | The Scripps Research Institute | Composiciones y procedimientos para inducir la desdiferenciación celular |
| CA2545020A1 (en) * | 2003-11-13 | 2005-05-26 | Pfizer Products Inc. | Octahydrophenanthrene hydrazinde derivatives useful as glucocorticoid receptor modulators |
| TWI370129B (en) | 2005-02-14 | 2012-08-11 | Msd Oss Bv | Non steroidal glucocorticoid receptor modulators |
| JP2009535430A (ja) | 2006-05-02 | 2009-10-01 | コーセプト セラピューティクス， インコーポレイテッド | Ｉｌ−２を摂取している患者における抑うつを処置するためのグルココルチコイドレセプターｉｉアンタゴニストの使用 |
| SI2114888T1 (sl) * | 2007-02-02 | 2011-02-28 | Pfizer Prod Inc | Triciklične spojine in njihova uporaba kot modulatorji glukokortikoidnega receptorja |
| DK2114970T3 (da) | 2007-02-02 | 2011-09-19 | Pfizer Prod Inc | Tricykliske forbindelser og deres anvendelse som glucocorticoidreceptormodulatorer |
-
2008
- 2008-01-25 DK DK08702351.1T patent/DK2114970T3/da active
- 2008-01-25 SI SI200830393T patent/SI2114970T1/sl unknown
- 2008-01-25 KR KR1020097018289A patent/KR101107949B1/ko not_active Expired - Fee Related
- 2008-01-25 EA EA200970666A patent/EA016494B1/ru not_active IP Right Cessation
- 2008-01-25 GE GEAP200811399A patent/GEP20125404B/en unknown
- 2008-01-25 PT PT08702351T patent/PT2114970E/pt unknown
- 2008-01-25 PL PL08702351T patent/PL2114970T3/pl unknown
- 2008-01-25 AU AU2008211613A patent/AU2008211613B2/en not_active Ceased
- 2008-01-25 MY MYPI20093089A patent/MY146087A/en unknown
- 2008-01-25 BR BRPI0808634-6A patent/BRPI0808634A2/pt not_active IP Right Cessation
- 2008-01-25 AT AT08702351T patent/ATE518872T1/de active
- 2008-01-25 JP JP2009547778A patent/JP4599462B2/ja not_active Expired - Fee Related
- 2008-01-25 CA CA2676670A patent/CA2676670C/en not_active Expired - Fee Related
- 2008-01-25 AP AP2009004942A patent/AP2455A/xx active
- 2008-01-25 EP EP08702351A patent/EP2114970B1/en active Active
- 2008-01-25 WO PCT/IB2008/000229 patent/WO2008093227A1/en not_active Ceased
- 2008-01-25 MX MX2009008284A patent/MX2009008284A/es active IP Right Grant
- 2008-01-25 RS RS20110429A patent/RS51970B/sr unknown
- 2008-01-25 CN CN2008800052954A patent/CN101616925B/zh not_active Expired - Fee Related
- 2008-01-25 HR HR20110702T patent/HRP20110702T1/hr unknown
- 2008-01-25 NZ NZ578638A patent/NZ578638A/en not_active IP Right Cessation
- 2008-01-25 MY MYPI20123293 patent/MY153057A/en unknown
- 2008-01-25 UA UAA200907728A patent/UA94639C2/ru unknown
- 2008-01-25 ES ES08702351T patent/ES2368286T3/es active Active
- 2008-01-28 ES ES08702358T patent/ES2353822T3/es active Active
- 2008-01-28 RS RS20110008A patent/RS51646B/sr unknown
- 2008-01-28 MY MYPI20093135A patent/MY148780A/en unknown
- 2008-01-28 PT PT08702358T patent/PT2114888E/pt unknown
- 2008-01-28 GE GEAP200811398A patent/GEP20125426B/en unknown
- 2008-01-28 UA UAA200907730A patent/UA95332C2/uk unknown
- 2008-01-28 KR KR1020097018294A patent/KR101114682B1/ko not_active Expired - Fee Related
- 2008-01-28 CN CN2008800056527A patent/CN101616896B/zh not_active Expired - Fee Related
- 2008-01-31 US US12/023,323 patent/US7547714B2/en not_active Expired - Fee Related
- 2008-01-31 PE PE2008000231A patent/PE20081736A1/es not_active Application Discontinuation
- 2008-01-31 US US12/023,362 patent/US7598231B2/en not_active Expired - Fee Related
- 2008-02-01 HN HN2008000179A patent/HN2008000179A/es unknown
- 2008-02-01 CL CL200800329A patent/CL2008000329A1/es unknown
- 2008-02-01 PE PE2008000234A patent/PE20090113A1/es not_active Application Discontinuation
- 2008-02-01 CL CL200800330A patent/CL2008000330A1/es unknown
- 2008-02-01 TW TW097104089A patent/TWI347842B/zh active
- 2008-02-01 AR ARP080100424A patent/AR065134A1/es active IP Right Grant
- 2008-02-01 TW TW097104074A patent/TWI373466B/zh not_active IP Right Cessation
- 2008-02-01 HN HN2008000178A patent/HN2008000178A/es unknown
- 2008-02-01 AR ARP080100425A patent/AR065135A1/es active IP Right Grant
-
2009
- 2009-05-08 US US12/437,704 patent/US8158660B2/en not_active Expired - Fee Related
- 2009-07-20 IL IL199972A patent/IL199972A/en active IP Right Grant
- 2009-07-21 US US12/506,825 patent/US7786097B2/en not_active Expired - Fee Related
- 2009-07-23 CR CR10949A patent/CR10949A/es not_active IP Right Cessation
- 2009-07-23 CR CR10948A patent/CR10948A/es not_active IP Right Cessation
- 2009-07-24 CU CU2009000132A patent/CU23848B1/es active IP Right Grant
- 2009-07-24 CU CU20090133A patent/CU23824A3/es active IP Right Grant
- 2009-07-29 NI NI200900148A patent/NI200900148A/es unknown
- 2009-07-29 NI NI200900149A patent/NI200900149A/es unknown
- 2009-07-29 DO DO2009000190A patent/DOP2009000190A/es unknown
- 2009-07-30 GT GT200900209A patent/GT200900209A/es unknown
- 2009-07-30 SV SV2009003346A patent/SV2009003346A/es not_active Application Discontinuation
- 2009-07-30 GT GT200900210A patent/GT200900210A/es unknown
- 2009-07-31 MA MA32127A patent/MA31117B1/fr unknown
- 2009-07-31 EC EC2009009553A patent/ECSP099553A/es unknown
- 2009-07-31 SV SV2009003349A patent/SV2009003349A/es active IP Right Grant
- 2009-07-31 EC EC2009009552A patent/ECSP099552A/es unknown
- 2009-07-31 MA MA32128A patent/MA31158B1/fr unknown
- 2009-07-31 CO CO09079796A patent/CO6190603A2/es active IP Right Grant
- 2009-07-31 TN TNP2009000324A patent/TN2009000324A1/fr unknown
- 2009-07-31 CO CO09079789A patent/CO6220937A2/es active IP Right Grant
- 2009-09-01 ZA ZA200906064A patent/ZA200906064B/xx unknown
- 2009-09-01 ZA ZA200906060A patent/ZA200906060B/xx unknown
-
2010
- 2010-12-02 CY CY20101101109T patent/CY1110962T1/el unknown
-
2011
- 2011-08-17 CY CY20111100784T patent/CY1111758T1/el unknown
- 2011-12-21 US US13/333,104 patent/US8445520B2/en not_active Expired - Fee Related
-
2013
- 2013-04-16 US US13/863,534 patent/US20140142316A1/en not_active Abandoned
-
2014
- 2014-07-01 US US14/320,674 patent/US8901310B2/en not_active Expired - Fee Related
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