JP2010507565A - メタスチン誘導体およびその用途 - Google Patents

メタスチン誘導体およびその用途 Download PDF

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Publication number
JP2010507565A
JP2010507565A JP2009518179A JP2009518179A JP2010507565A JP 2010507565 A JP2010507565 A JP 2010507565A JP 2009518179 A JP2009518179 A JP 2009518179A JP 2009518179 A JP2009518179 A JP 2009518179A JP 2010507565 A JP2010507565 A JP 2010507565A
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JP2010507565A5 (https=
Inventor
泰司 浅見
直城 西澤
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Takeda Pharmaceutical Co Ltd
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Takeda Pharmaceutical Co Ltd
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • C07K14/4701Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
    • C07K14/4702Regulators; Modulating activity
    • C07K14/4703Inhibitors; Suppressors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
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    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/1703Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • A61K38/1709Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
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  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Endocrinology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Reproductive Health (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Zoology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Toxicology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Oncology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
JP2009518179A 2006-10-25 2007-10-24 メタスチン誘導体およびその用途 Pending JP2010507565A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2006290536 2006-10-25
JP2007021387 2007-01-31
JP2007221911 2007-08-28
PCT/JP2007/071169 WO2008050897A1 (en) 2006-10-25 2007-10-24 Metastin derivatives and use thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013004011A Division JP5686825B2 (ja) 2006-10-25 2013-01-11 メタスチン誘導体およびその用途

Publications (2)

Publication Number Publication Date
JP2010507565A true JP2010507565A (ja) 2010-03-11
JP2010507565A5 JP2010507565A5 (https=) 2010-12-09

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ID=38925530

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2009518179A Pending JP2010507565A (ja) 2006-10-25 2007-10-24 メタスチン誘導体およびその用途
JP2013004011A Expired - Fee Related JP5686825B2 (ja) 2006-10-25 2013-01-11 メタスチン誘導体およびその用途

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2013004011A Expired - Fee Related JP5686825B2 (ja) 2006-10-25 2013-01-11 メタスチン誘導体およびその用途

Country Status (33)

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US (2) US8765909B2 (https=)
EP (1) EP2081955B1 (https=)
JP (2) JP2010507565A (https=)
KR (1) KR101424306B1 (https=)
AR (1) AR063367A1 (https=)
AU (1) AU2007309969B2 (https=)
BR (1) BRPI0717441B8 (https=)
CA (1) CA2667537C (https=)
CL (1) CL2007003053A1 (https=)
CR (1) CR10799A (https=)
CY (1) CY1116627T1 (https=)
DK (1) DK2081955T3 (https=)
EC (1) ECSP099279A (https=)
ES (1) ES2539430T3 (https=)
GE (1) GEP20125568B (https=)
HR (1) HRP20150819T1 (https=)
HU (1) HUE025291T2 (https=)
IL (1) IL198046A (https=)
JO (1) JO3048B1 (https=)
MA (1) MA30887B1 (https=)
ME (1) ME00786B (https=)
MX (1) MX2009004148A (https=)
MY (1) MY145975A (https=)
NO (1) NO341584B1 (https=)
NZ (1) NZ576375A (https=)
PE (1) PE20081469A1 (https=)
PL (1) PL2081955T3 (https=)
PT (1) PT2081955E (https=)
RS (1) RS54083B1 (https=)
SI (1) SI2081955T1 (https=)
TN (1) TN2009000140A1 (https=)
TW (1) TWI404726B (https=)
WO (1) WO2008050897A1 (https=)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2016523238A (ja) * 2013-06-12 2016-08-08 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung 関節症の処置のためのヒドロキシエチレン誘導体
JP2020525534A (ja) * 2017-07-05 2020-08-27 エックスディーシーエクスプローラー (シャンハイ) カンパニー リミテッド ペプチド類化合物、その使用及びそれを含む組成物
JP2023521388A (ja) * 2020-04-08 2023-05-24 ラトガース,ザ ステート ユニバーシティ オブ ニュー ジャージー 脂肪肝疾患に対する修飾キスペプチン受容体作用薬

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1761680A (zh) 2002-12-26 2006-04-19 武田药品工业株式会社 肿瘤迁移抑制素衍生物及其用途
CA2571420A1 (en) 2004-06-25 2006-01-05 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
AR058584A1 (es) 2005-12-22 2008-02-13 Takeda Pharmaceutical Derivados de metastina y uso de los mismos
US20090099334A1 (en) * 2005-12-22 2009-04-16 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
US8404643B2 (en) 2005-12-22 2013-03-26 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
US20090093615A1 (en) * 2005-12-22 2009-04-09 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
WO2007125619A1 (ja) * 2006-04-26 2007-11-08 Kyoto University Gpr54アゴニスト活性を有する新規化合物
JO3048B1 (ar) 2006-10-25 2016-09-05 Takeda Pharmaceuticals Co مشتقات متاستين واستخدامها
US8110639B2 (en) * 2006-11-17 2012-02-07 Solvay Advanced Polymers, L.L.C. Transparent and flame retardant polysulfone compositions
EP2277900A4 (en) * 2008-04-24 2011-08-03 Takeda Pharmaceutical METASTINE DERIVATIVE AND ITS USE
EP2275433B1 (en) * 2008-04-30 2017-06-07 Kyoto University Metastin derivative and use thereof
LT2314609T (lt) * 2008-07-30 2017-04-10 Takeda Pharmaceutical Company Limited Metastino darinys ir jo panaudojimas
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