US3314970A
(en)
|
|
1967-04-18 |
|
Pykrolidino ketones |
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(en)
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1941-05-01 |
1942-05-12 |
Us Rubber Co |
Parasiticide
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(en)
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1948-10-19 |
1953-08-18 |
Burroughs Wellcome Co |
Process for the preparation of amino ketones
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(en)
|
1952-09-10 |
1957-01-22 |
Merck & Co Inc |
Deamination process
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US2771391A
(en)
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1953-08-20 |
1956-11-20 |
Allied Lab Inc |
Physiologically active p-alkoxy-beta-piperidinopropiophenones causing cns depressantand anesthetic effects in animals
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(en)
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1955-07-01 |
1961-08-22 |
Endo Lab |
1, 1-diphenyl-1-hydroxy-4-(pyrrolidyl)-butanone-2
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BE561320A
(nl)
|
1956-10-04 |
1960-05-20 |
Lab Pharmaceutica Nv |
Werkwijze voor de bereiding van nieuwe 4-carbalkoxy-4-fenyl piperidine derivaten.
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US3080372A
(en)
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1960-03-25 |
1963-03-05 |
Res Lab Dr C Janssen |
1-aroylalkyl-4-arylpiperidine derivatives
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CH402859A
(de)
|
1960-05-24 |
1965-11-30 |
Wander Ag Dr A |
Verfahren zur Herstellung von a-Pyrrolidino-valerophenonen
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US3252996A
(en)
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1962-10-02 |
1966-05-24 |
Ciba Geigy Corp |
Alpha-pyrrolidinomethyl valero and caprophenones
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US3151124A
(en)
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1961-11-20 |
1964-09-29 |
Ciba Geigy Corp |
Alpha oxy-beta alkyl-gamma tertiary amino-alpha phenyl propanes
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BE633437A
(ja)
|
1962-06-11 |
|
|
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(en)
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1962-10-11 |
1965-08-31 |
Ciba Geigy Corp |
Alpha-phenyl-beta pyrrolidino-propiophenones
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US3310566A
(en)
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1963-11-18 |
1967-03-21 |
American Home Prod |
Substituted 4-piperidino-butyrophenone oximes
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US3284453A
(en)
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1964-09-29 |
1966-11-08 |
American Cyanamid Co |
4-(2-aroylethyl)-1-piperazinecarboxylic acid esters
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US3364210A
(en)
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1964-10-05 |
1968-01-16 |
American Cyanamid Co |
Substituted 3-aminoacrylophenones and method of preparing the same
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NL143925C
(ja)
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1965-03-09 |
|
|
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US3816433A
(en)
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1965-03-24 |
1974-06-11 |
Ferrosan Ab |
4-fluoro-ypsilon-(4-methylpiperidino)-butyrophenone and its pharmaceutically acceptable salts
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GB1079520A
(en)
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1965-07-19 |
1967-08-16 |
Roche Products Ltd |
Novel tetrahydro-isoquinoline derivatives and a process for the manufacture thereof
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US3317538A
(en)
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1965-10-22 |
1967-05-02 |
American Home Prod |
4, 4'-diamino-butyrophenones
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US3417087A
(en)
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1965-12-27 |
1968-12-17 |
Research Corp |
3(aminopropionyl)benzothiophenes
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US3364120A
(en)
*
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1966-01-24 |
1968-01-16 |
Babcock & Wilcox Co |
Nuclear control rod actuator
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US3637704A
(en)
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1967-10-18 |
1972-01-25 |
Dainippon Pharmaceutical Co |
1gamma-(p-fluorobenzoyl)propyl-4-phenylalkyl piperazine
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GB1186495A
(en)
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1968-02-20 |
1970-04-02 |
Delalande Sa |
0-[3-(4-Fluorobenzoyl) Proplyl]-4-Substituted Piperazines, their Acid Addition Salts and their method of preparation
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GB1196721A
(en)
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1968-02-23 |
1970-07-01 |
Ici Ltd |
Piperazine Derivatives
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CH502336A
(de)
|
1968-04-29 |
1971-01-31 |
Ciba Geigy Ag |
Verfahren zur Herstellung von neuen Estern substituierter Phenylessigsäuren
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US3465080A
(en)
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1968-10-07 |
1969-09-02 |
American Cyanamid Co |
Therapeutic compositions containing morpholinoalkylene - indoles and methods of administering such in the treatment of depression
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FR2035749A1
(ja)
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1969-02-06 |
1970-12-24 |
Bellon Labor Sa Roger |
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US3536809A
(en)
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1969-02-17 |
1970-10-27 |
Alza Corp |
Medication method
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GB1262965A
(en)
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1969-03-21 |
1972-02-09 |
Ferrosan As |
Butyrophenones
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US3598123A
(en)
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1969-04-01 |
1971-08-10 |
Alza Corp |
Bandage for administering drugs
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US3651085A
(en)
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1969-04-14 |
1972-03-21 |
Robins Co Inc A H |
1-(omega-benzoylalkyl)-3-substituted pyrrolidines
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US3703527A
(en)
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1969-06-04 |
1972-11-21 |
Hoffmann La Roche |
Preparation of mannich-bases
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US3907812A
(en)
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1969-07-16 |
1975-09-23 |
Sumitomo Chemical Co |
Butyrophenone derivatives
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US3936468A
(en)
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1969-10-27 |
1976-02-03 |
Sumitomo Chemical Company, Ltd. |
Phenylbutanol derivatives
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US3799932A
(en)
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1970-03-20 |
1974-03-26 |
Sumitomo Chemical Co |
Gamma-piperidinobutyrophenones
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US3651067A
(en)
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1970-04-15 |
1972-03-21 |
Usv Pharma Corp |
Styrene ethers of amino alcohols
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DE2021470A1
(de)
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1970-05-02 |
1971-11-25 |
Cassella Farbwerke Mainkur Ag |
Piperazinderivate
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FR2092133B1
(ja)
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1970-05-06 |
1974-03-22 |
Orsymonde |
|
US4029801A
(en)
|
1970-09-03 |
1977-06-14 |
John Wyeth & Brother Limited |
Pharmaceutical compositions and methods of treating hypertension
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US4148796A
(en)
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1971-03-15 |
1979-04-10 |
Sumitomo Chemical Company, Limited |
γ-Piperidinobutyrophenones
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US3794677A
(en)
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1971-07-01 |
1974-02-26 |
American Home Prod |
Di(lower)alkylamino-and heteroamino-(lower)alkyl-alpha,alpha,alpha-trifluoro-m-toluic acid esters and derivatives
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US3969356A
(en)
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1971-09-13 |
1976-07-13 |
Kali-Chemie Aktiengesellschaft |
N-[3-(p-f-benzoyl)-propyl]-N'-[2.(nitro,nitro-el, or methoxyphenyl)-ethyl]-p
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US3850935A
(en)
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1971-10-16 |
1974-11-26 |
Sumitomo Chemical Co |
Process for producing piperidine derivatives by degrading quaternary piperidinium salts
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JPS4948957B2
(ja)
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1971-10-26 |
1974-12-24 |
|
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US3806526A
(en)
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1972-01-28 |
1974-04-23 |
Richardson Merrell Inc |
1-aroylalkyl-4-diphenylmethyl piperidines
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BE795671A
(fr)
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1972-02-21 |
1973-08-20 |
Ugine Kuhlmann |
Nouveaux medicaments antiuriques
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US3951978A
(en)
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1972-04-22 |
1976-04-20 |
Istituto Luso Farmaco D'italia S.R.L. |
1,3-Disubstituted 3-aroylpropanes and process for the preparation thereof
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US3845770A
(en)
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1972-06-05 |
1974-11-05 |
Alza Corp |
Osmatic dispensing device for releasing beneficial agent
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(en)
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1972-06-28 |
1975-11-25 |
Sumitomo Chemical Co |
Aryl ketones and production thereof
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US3900478A
(en)
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1973-01-29 |
1975-08-19 |
Squibb & Sons Inc |
2-methyl-2-piperidino-3'-(trifluoromethyl) propiophenone
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CH602687A5
(ja)
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1973-03-12 |
1978-07-31 |
Kali Chemie Ag |
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US3916899A
(en)
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1973-04-25 |
1975-11-04 |
Alza Corp |
Osmotic dispensing device with maximum and minimum sizes for the passageway
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US3873539A
(en)
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1973-10-03 |
1975-03-25 |
Sandoz Ag |
Substituted-4-aminoacetyl alkanoylphenones
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US4054570A
(en)
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1973-10-18 |
1977-10-18 |
Ciba-Geigy Corporation |
4-Piperidinobutyrophenones
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US3992546A
(en)
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1973-10-18 |
1976-11-16 |
Ciba-Geigy Corporation |
4-Piperidinobutyrophenones as neuroleptics
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US3944064A
(en)
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1973-10-26 |
1976-03-16 |
Alza Corporation |
Self-monitored device for releasing agent at functional rate
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US4181803A
(en)
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1973-12-14 |
1980-01-01 |
Eisai Co., Ltd. |
Propiophenone derivatives and preparation thereof
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US3995047A
(en)
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1973-12-14 |
1976-11-30 |
Eisai Co., Ltd. |
Propiophenone derivatives in the treatment of pathological muscular conditions
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US3912755A
(en)
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1974-01-30 |
1975-10-14 |
Lilly Co Eli |
Preparation of pharmaceutical intermediates
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US3931197A
(en)
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1974-02-08 |
1976-01-06 |
Richardson-Merrell Inc. |
Substituted piperidine derivatives
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US4069331A
(en)
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1974-05-16 |
1978-01-17 |
Boehringer Ingelheim Gmbh |
N-(p-fluorobenzoyl-n-propyl)-4-piperidylamides and salts thereof
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IL48319A0
(en)
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1974-10-26 |
1975-12-31 |
Merck Patent Gmbh |
Araliphatic nitrogen compounds and a process for their preparation
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US4028366A
(en)
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1975-01-20 |
1977-06-07 |
Sterling Drug Inc. |
2-Naphthyl-lower-alkanoylamines
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US4169892A
(en)
*
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1975-04-03 |
1979-10-02 |
Innothera |
1-(benzothien-2'-yl)-3-morpholino propanones and therapeutic compositions containing same
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GB1498884A
(en)
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1975-04-15 |
1978-01-25 |
Wyeth John & Brother Ltd |
Aminoacetamide-pyridyl-tetrahydropyridyl and-piperidyl derivatives
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FR2316939A1
(fr)
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1975-07-08 |
1977-02-04 |
Troponwerke Dinklage & Co |
Derives de 2-benzopyranone et leur application comme medicaments
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FI60559C
(fi)
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1975-07-17 |
1982-02-10 |
Sumitomo Chemical Co |
Foerfarande foer framstaellning av ny-(tertiaer amino)-orto-aminobutyrofenonfoereningar
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FR2325379A1
(fr)
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1975-09-29 |
1977-04-22 |
Cerm Cent Europ Rech Mauvernay |
Nouveaux derives de 2-(2-hydroxyethyl)tetrahydro-1,4 oxazines substituees et leur application comme medicaments antispasmodique
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DE2557341A1
(de)
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1975-12-19 |
1977-06-30 |
Hoechst Ag |
Basisch substituierte indolderivate und verfahren zu ihrer herstellung
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US4333941A
(en)
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1975-12-22 |
1982-06-08 |
The Dow Chemical Company |
Inhibition of enveloped viruses with phenyl ketones
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US4008719A
(en)
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1976-02-02 |
1977-02-22 |
Alza Corporation |
Osmotic system having laminar arrangement for programming delivery of active agent
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FR2361883A2
(fr)
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1976-04-09 |
1978-03-17 |
Fabre Sa Pierre |
Amides de la pyrrolidino ethyl amine utilisables en therapeutique pulmonaire
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DE2718405A1
(de)
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1977-04-26 |
1978-11-02 |
Boehringer Sohn Ingelheim |
Neue n- eckige klammer auf 1-(3-benzoylpropyl)-4-piperidyl eckige klammer zu -sulfonsaeureamide und verfahren zu deren herstellung
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JPS54125630A
(en)
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1978-02-22 |
1979-09-29 |
Nippon Zoki Pharmaceutical Co |
Novel propanone derivative*its manufacture and medical composition containing it as active component
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DE2933636A1
(de)
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1978-08-30 |
1980-03-20 |
Sandoz Ag |
Neue n-phenylindolinderivate, ihre herstellung und pharmazeutische praeparate, welche diese verbindungen enthalten
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FR2443246A1
(fr)
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1978-12-05 |
1980-07-04 |
Pharmindustrie |
Nouveaux medicaments a base de derives de la phenyl-1 (piperidyl-4)-3 propanone-1
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US4293561A
(en)
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1979-03-09 |
1981-10-06 |
Syntex (U.S.A.) Inc. |
1-(Naphthyl-n-propyl)imidazole derivatives
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US4283404A
(en)
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1979-09-04 |
1981-08-11 |
Richardson-Merrell Inc. |
Aroylethenylpiperidinobutyrophenone antipsychotic agents
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DE2939292A1
(de)
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1979-09-28 |
1981-04-09 |
Boehringer Mannheim Gmbh, 6800 Mannheim |
N-phenoxyalkylpiperidin-derivate, verfahrenn zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
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DE3041199A1
(de)
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1979-11-14 |
1981-05-21 |
Sandoz-Patent-GmbH, 7850 Lörrach |
Neue stilbenverbindungen, deren herstellung und verwendung
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FR2473518A1
(fr)
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1980-01-16 |
1981-07-17 |
Unicler |
Derives du phenyl-1 morpholino-4 butene-1 ol-3, leur preparation et leur application en therapeutique
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DE3019497A1
(de)
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1980-05-22 |
1981-11-26 |
Bayer Ag, 5090 Leverkusen |
Aminopropiophenon-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide
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DE3019496A1
(de)
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1980-05-22 |
1981-11-26 |
Bayer Ag, 5090 Leverkusen |
Aminopropanol-derivate, verfahren zu ihrer herstellung und ihre verwendung als fungizide
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US4400380A
(en)
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1980-07-02 |
1983-08-23 |
Merrell Dow Pharmaceuticals Inc. |
Antiviral 1-aryl-5-amino-1-penten-3-ones
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(en)
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1981-10-07 |
1983-08-09 |
Sandoz, Inc. |
Isoxazolyl indolamines
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JPS5944371A
(ja)
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1982-09-07 |
1984-03-12 |
Dainippon Pharmaceut Co Ltd |
1―フエニル―2―メチル―3―(1―ピロリジニル)―1―プロパノン誘導体
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FR2534912B1
(fr)
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1982-10-26 |
1985-06-28 |
Lafon Labor |
Nouveaux derives de (2,4,6-trimethoxyphenyl) - (3-piperidinopropyl) -cetone, utilisation en therapeutique et procede de preparation
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US4559371A
(en)
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1983-02-18 |
1985-12-17 |
Ciba Geigy Corporation |
Photocurable colored compositions employing alpha-amino phenone initiator
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US4515793A
(en)
*
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1983-07-27 |
1985-05-07 |
Edna Mcconnell Clark Foundation |
Phenylpiperazines which are useful in the treatment of schistosomiasis
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EP0138754B1
(de)
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1983-08-15 |
1988-05-25 |
Ciba-Geigy Ag |
Photohärtbare Gemische
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HU33131A
(ja)
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1984-01-26 |
1984-10-29 |
|
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FR2560873B1
(fr)
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1984-03-09 |
1986-09-26 |
Rhone Poulenc Sante |
Medicaments a base de derives de la piperidine, nouveaux derives de la piperidine et leurs procedes de preparation
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DE3413897A1
(de)
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1984-04-13 |
1985-10-17 |
Bayer Ag, 5090 Leverkusen |
(beta)-naphthylalkylamine
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1984-05-07 |
1985-10-01 |
Sandoz, Inc. |
Indolamine derivatives as anti-fertility agents
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DE3436450A1
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1984-10-05 |
1986-04-10 |
Bayer Ag, 5090 Leverkusen |
Verfahren zur herstellung von p-aminoethylketonen
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1985-04-11 |
1991-10-15 |
Nippon Kayaku Kabushiki Kaisha |
Derivatives of an aminoketone
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FR2584715B1
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1985-07-10 |
1987-10-09 |
Lafon Labor |
Phenyl-(3-hexamethyleneiminopropyl)-cetone, procede de preparation et utilisation en therapeutique
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1985-10-09 |
1994-02-17 |
Shell Int Research |
Neue Acrylsäureamide.
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DE3602016A1
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1985-12-05 |
1987-06-11 |
Bayer Ag |
Pyri(mi)dyl-oxy- und thio-benzoesaeure-derivate
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FR2597864B1
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1986-04-28 |
1990-11-16 |
Lafon Labor |
Nouveaux derives de la n-((trimethoxy-2,4,6-benzoyl)-3 propyl) piperidine, leurs procedes de preparation et leur application en therapeutique
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KR910006138B1
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1986-09-30 |
1991-08-16 |
에자이 가부시끼가이샤 |
환상아민 유도체
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1986-12-22 |
1988-08-23 |
Ortho Pharmaceutical Corporation |
6-benzoxazinyl- and 6-benzothiazinyl-2,3,4,5-tetrahydropyridazin-3-ones and pharmaceutical use
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JPH0637389B2
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1986-12-26 |
1994-05-18 |
北陸製薬株式会社 |
頻尿治療剤
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ATE82282T1
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1987-01-20 |
1992-11-15 |
Dainippon Pharmaceutical Co |
Aromatische heterozyklische karbonsaeureamidabkoemmlinge, verfahren zur herstellung und arzneimittel, die diese enthalten.
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1987-02-11 |
1989-06-20 |
Sterling Drug Inc. |
4-arylcarbonyl-1-[(4-morpholinyl)-lower-alkyl]-1H-indoles
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1987-02-11 |
1989-10-17 |
Sterling Drug Inc. |
4-arylcarbonyl-1-[(4-morpholinyl)-lower-alkyl]-1H-indoles
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ATE89262T1
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1987-03-26 |
1993-05-15 |
Ciba Geigy Ag |
Neue alpha-aminoacetophenone als photoinitiatoren.
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1987-11-24 |
1989-09-26 |
Merrell Dow Pharmaceuticals Inc. |
1,4-Disubstituted-piperidinyl compounds useful as analgesics and muscle relaxants
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1987-11-27 |
1993-03-23 |
Eisai Co., Ltd. |
Piperidine compounds useful to treat cerebrovascular diseases
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1988-01-25 |
1988-12-13 |
Minnesota Mining And Manufacturing Company |
Photosensitizers and polymerizable compositions with mannich bases and iodonium salts
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IT1231260B
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1988-11-16 |
1991-11-28 |
Sergio Bertini Curri |
Farmaco e metodo per aumentare volume e velocita' del flusso microcircolatorio capillare a livello cutaneo
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JPH0660141B2
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1989-09-12 |
1994-08-10 |
三井東圧化学株式会社 |
ジヒドロカフェイン酸誘導体およびそれを有効成分として含有する治療剤
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1990-01-26 |
1993-01-26 |
Taiho Pharmaceutical Co., Ltd. |
Piperazine compounds, processes for preparation thereof and medical uses thereof
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1990-03-08 |
1991-05-07 |
Sterling Drug Inc. |
3-Arylcarbonyl-1H-indole-containing compounds
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1990-07-26 |
1994-01-04 |
Novo Nordisk A/S |
1,4-disubstituted piperazines
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1993-09-28 |
1998-05-12 |
Pfizer |
Benzisoxazole and benzisothizole derivatives as cholinesterase inhibitors
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FR2680366B1
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1991-08-13 |
1995-01-20 |
Adir |
Nouveaux derives d'arylethylamines, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent.
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JP3157882B2
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1991-11-15 |
2001-04-16 |
帝国臓器製薬株式会社 |
新規なベンゾチオフエン誘導体
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1992-06-22 |
1997-07-01 |
Boehringer Ingelheim Kg |
Anellated dihydropyridines and the use thereof for the production of pharmaceutical preparation
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1992-10-08 |
1996-09-24 |
Warner Lambert Co |
Apparatus for multiple simultaneous synthesis
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GB9301660D0
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1993-01-28 |
1993-03-17 |
Smithkline Beecham Plc |
Pharmaceuticals
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1993-02-01 |
2000-10-03 |
Smithkline Beecham P.L.C. |
Benzopyran, benzothiopyran and benzofuran derivatives as 5-HT4 antagonists
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1993-02-23 |
1997-04-16 |
Hoechst Ag |
Bencenosulfonil-ureas y -tioureas sustituidas, procedimiento para su preparacion y su utilizacion como agentes farmaceuticos.
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1993-04-07 |
1997-08-12 |
Otsuka Pharmaceutical Co., Ltd. |
Peripheral vasodilating agent containing piperidine derivative as active ingredient
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1993-08-18 |
1994-09-27 |
Warner-Lambert Company |
3-thio or amino substituted-benzo[b]thiophene-2-carboxamides and 3-oxygen, thio, or amino substituted-benzofuran-2-carboxamides as inhibitors of cell adhesion
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GB9324018D0
(en)
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1993-11-23 |
1994-01-12 |
Merck Sharp & Dohme |
Therapeutic agents
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FR2713637B1
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1993-12-15 |
1996-01-05 |
Cird Galderma |
Nouveaux composés bi-aromatiques dérivés d'amide, compositions pharmaceutiques et cosmétiques les contenant et utilisations.
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DK139593D0
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1993-12-16 |
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Lundbeck & Co As H |
Compounds
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CN1138324A
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1993-12-21 |
1996-12-18 |
贝林格尔·英格海姆公司 |
增环的二氢吡啶及其在制备药物制剂中的应用
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GB9408185D0
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1994-04-25 |
1994-06-15 |
Fujisawa Pharmaceutical Co |
New benzamide derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same
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