JP2009528284A5 - - Google Patents
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- Publication number
- JP2009528284A5 JP2009528284A5 JP2008555763A JP2008555763A JP2009528284A5 JP 2009528284 A5 JP2009528284 A5 JP 2009528284A5 JP 2008555763 A JP2008555763 A JP 2008555763A JP 2008555763 A JP2008555763 A JP 2008555763A JP 2009528284 A5 JP2009528284 A5 JP 2009528284A5
- Authority
- JP
- Japan
- Prior art keywords
- phenyl
- benzimidazol
- carboxylic acid
- thiazole
- dimethoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 CC(C=C1)(C=Cc(nc2)c1[n]2-c1nc(*)c(*)[s]1)N Chemical compound CC(C=C1)(C=Cc(nc2)c1[n]2-c1nc(*)c(*)[s]1)N 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US77696406P | 2006-02-27 | 2006-02-27 | |
| PCT/EP2007/051541 WO2007096315A1 (en) | 2006-02-27 | 2007-02-19 | 4-phenyl-thiazole-5-carboxylic acids and 4-phenyl-thiazole-5-carboxylic acid amides as plk1 inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009528284A JP2009528284A (ja) | 2009-08-06 |
| JP2009528284A5 true JP2009528284A5 (enExample) | 2012-06-07 |
Family
ID=38051896
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008555763A Pending JP2009528284A (ja) | 2006-02-27 | 2007-02-19 | Ｐｌｋ１阻害剤としての４−フェニル−チアゾール−５−カルボン酸及び４−フェニル−チアゾール−５−カルボン酸アミド |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US7504513B2 (enExample) |
| EP (1) | EP1991543A1 (enExample) |
| JP (1) | JP2009528284A (enExample) |
| KR (1) | KR101060539B1 (enExample) |
| CN (1) | CN101415704A (enExample) |
| AR (1) | AR059621A1 (enExample) |
| AU (1) | AU2007217575A1 (enExample) |
| BR (1) | BRPI0710473A2 (enExample) |
| CA (1) | CA2642921A1 (enExample) |
| CR (1) | CR10206A (enExample) |
| EC (1) | ECSP088700A (enExample) |
| IL (1) | IL193481A0 (enExample) |
| MA (1) | MA30260B1 (enExample) |
| MX (1) | MX2008010884A (enExample) |
| NO (1) | NO20083708L (enExample) |
| RU (1) | RU2008138163A (enExample) |
| TW (1) | TW200745097A (enExample) |
| WO (1) | WO2007096315A1 (enExample) |
| ZA (1) | ZA200807074B (enExample) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008149784A1 (ja) * | 2007-06-08 | 2008-12-11 | Nec Corporation | 半導体集積回路及びフィルタ制御方法 |
| WO2009094224A1 (en) | 2008-01-25 | 2009-07-30 | Millennium Pharmaceuticals, Inc. | Thiophenes and their use as phosphatidylinositol 3-kinase (pi3k) inhibitors |
| US8962614B2 (en) * | 2008-04-17 | 2015-02-24 | The Johns Hopkins University | ON01910.Na enhances chemotherapeutic agent activity in drug-resistant tumors |
| CN102150210B (zh) * | 2008-09-10 | 2013-04-10 | 数据激光有限公司 | 数据存储介质 |
| WO2010077295A1 (en) * | 2008-12-09 | 2010-07-08 | King Faisal Specialist Hospital & Research Centre | Substituted tricyclic heterocycles and uses to treat tumors and proliferative disorders |
| JP2012512223A (ja) * | 2008-12-18 | 2012-05-31 | エフ．ホフマン−ラ ロシュ アーゲー | チアゾリル−ベンズイミダゾール類 |
| US9090601B2 (en) * | 2009-01-30 | 2015-07-28 | Millennium Pharmaceuticals, Inc. | Thiazole derivatives |
| US8796314B2 (en) | 2009-01-30 | 2014-08-05 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
| CA2750935A1 (en) | 2009-01-30 | 2010-08-12 | Millennium Pharmaceuticals, Inc. | Heteroaryls and their use as pi3k inhibitors |
| PH12013500274A1 (en) | 2010-08-11 | 2013-03-04 | Millennium Pharm Inc | Heteroaryls and uses thereof |
| JP2013533318A (ja) | 2010-08-11 | 2013-08-22 | ミレニアム ファーマシューティカルズ， インコーポレイテッド | ヘテロアリールおよびその使用 |
| WO2012021611A1 (en) | 2010-08-11 | 2012-02-16 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
| CA2814688A1 (en) | 2010-10-13 | 2012-04-19 | Millennium Pharmaceuticals, Inc. | Heteroaryls and uses thereof |
Family Cites Families (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4322429A (en) * | 1980-09-16 | 1982-03-30 | Eli Lilly And Company | Isoxazolylbenzamides as insecticides |
| US4818270A (en) * | 1986-08-28 | 1989-04-04 | Monsanto Company | 2-(Heteroamino)-4,5-substituted-oxazole/thiazole compounds as herbicide antidotes, compositions and use |
| US6194447B1 (en) * | 1998-07-02 | 2001-02-27 | Neurosearch A/S | Bis (benzimidazole) derivatives serving as potassium blocking agents |
| KR100904157B1 (ko) | 2000-08-10 | 2009-06-23 | 파마시아 이탈리아 에스.피.에이. | 키나제 억제제로서 활성인 비사이클로-피라졸, 이의제조방법 및 이를 포함하는 약제학적 조성물 |
| GB0102687D0 (en) | 2001-02-02 | 2001-03-21 | Pharmacia & Upjohn Spa | Oxazolyl-pyrazole derivatives active as kinase inhibitors,process for their preparation and pharmaceutical compositions comprising them |
| EP1476552A2 (en) | 2002-02-22 | 2004-11-17 | Strebhardt, Klaus, Prof. Dr. | Agent for inhibiting development or progress of proliferative diseases and especially cancer diseases and pharmaceutical composition containing said agent |
| EP1486490A1 (en) * | 2002-02-28 | 2004-12-15 | Takeda Chemical Industries, Ltd. | Azole compounds |
| AU2003213660C1 (en) | 2002-02-28 | 2010-10-28 | Onconova Therapeutics, Inc. | Amino-substituted (E)-2,6-dialkoxystyryl 4-substituted benzylsulfones for treating proliferative disorders |
| JP2003321460A (ja) * | 2002-02-28 | 2003-11-11 | Takeda Chem Ind Ltd | アゾール化合物 |
| EP1501794A1 (de) | 2002-05-03 | 2005-02-02 | Schering Aktiengesellschaft | Thiazolidinone und ihre verwendung als polo like kinase inhibitoren |
| US6906186B1 (en) | 2002-07-30 | 2005-06-14 | Isis Pharmaceuticals, Inc. | Antisense modulation of polo-like kinase expression |
| BR0313160A (pt) * | 2002-08-08 | 2005-07-12 | Smithkline Beecham Corp | Composto, composição farmacêutica, métodos para tratar uma condição e um neoplasmo suscetìvel em um animal em um animal, processo para preparar um composto e uso de um composto |
| EP1576128A4 (en) | 2002-11-14 | 2008-02-13 | Massachusetts Inst Technology | PRODUCTS AND METHODS FOR MODULATING INTERACTIONS BETWEEN PEPTIDE PEPTIDE BINDING DOMAINS |
| WO2004043936A1 (ja) | 2002-11-14 | 2004-05-27 | Kyowa Hakko Kogyo Co., Ltd. | Ｐｌｋ阻害剤 |
| WO2004054186A1 (ja) | 2002-12-12 | 2004-06-24 | Fujitsu Limited | データ中継装置、連想メモリデバイス、および連想メモリデバイス利用情報検索方法 |
| GB0302220D0 (en) | 2003-01-30 | 2003-03-05 | Cyclacel Ltd | Use |
| US7514446B2 (en) | 2003-02-20 | 2009-04-07 | Smithkline Beecham Corporation | Pyrimidine compounds |
| ES2326808T3 (es) | 2003-04-01 | 2009-10-20 | Smithkline Beecham Corporation | Compuestos de imidazotriazina para el tratamiento de enfermedades cancerosas. |
| NZ571898A (en) | 2003-06-24 | 2010-01-29 | Pfizer Prod Inc | Reaction of 2-chloro-8-benzyloxyquinoline with 2-nitrophenylamine in the presence of 1,2-bis(diphenylphosphino)ethane (dppe), palladium catalyst and a base |
| WO2005019193A2 (en) | 2003-08-20 | 2005-03-03 | Smithkline Beecham Corporation | Phenylurea derivatives useful in the treatment of conditions mediated by polo-like kinases (plk) |
| JP5164380B2 (ja) | 2003-10-21 | 2013-03-21 | サイクラセル リミテッド | ピリミジン−４−イル−３，４−チオン化合物及び治療におけるその使用 |
| DE10351744A1 (de) | 2003-10-31 | 2005-06-16 | Schering Ag | Thiazolidinone, deren Herstellung und Verwendung als Arzneimittel |
| JP2007519720A (ja) | 2004-01-28 | 2007-07-19 | スミスクライン ビーチャム コーポレーション | チアゾール化合物 |
-
2007
- 2007-02-07 US US11/703,306 patent/US7504513B2/en not_active Expired - Fee Related
- 2007-02-19 RU RU2008138163/04A patent/RU2008138163A/ru not_active Application Discontinuation
- 2007-02-19 AU AU2007217575A patent/AU2007217575A1/en not_active Abandoned
- 2007-02-19 EP EP07712233A patent/EP1991543A1/en not_active Withdrawn
- 2007-02-19 JP JP2008555763A patent/JP2009528284A/ja active Pending
- 2007-02-19 CN CNA2007800068055A patent/CN101415704A/zh active Pending
- 2007-02-19 WO PCT/EP2007/051541 patent/WO2007096315A1/en not_active Ceased
- 2007-02-19 KR KR1020087021067A patent/KR101060539B1/ko not_active Expired - Fee Related
- 2007-02-19 CA CA002642921A patent/CA2642921A1/en not_active Abandoned
- 2007-02-19 MX MX2008010884A patent/MX2008010884A/es not_active Application Discontinuation
- 2007-02-19 BR BRPI0710473-1A patent/BRPI0710473A2/pt not_active IP Right Cessation
- 2007-02-23 AR ARP070100768A patent/AR059621A1/es unknown
- 2007-02-26 TW TW096106341A patent/TW200745097A/zh unknown
-
2008
- 2008-08-14 CR CR10206A patent/CR10206A/es not_active Application Discontinuation
- 2008-08-14 IL IL193481A patent/IL193481A0/en unknown
- 2008-08-15 ZA ZA200807074A patent/ZA200807074B/xx unknown
- 2008-08-26 EC EC2008008700A patent/ECSP088700A/es unknown
- 2008-08-28 NO NO20083708A patent/NO20083708L/no not_active Application Discontinuation
- 2008-09-04 MA MA31208A patent/MA30260B1/fr unknown
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