JP2009040767A5 - - Google Patents
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- Publication number
- JP2009040767A5 JP2009040767A5 JP2008173198A JP2008173198A JP2009040767A5 JP 2009040767 A5 JP2009040767 A5 JP 2009040767A5 JP 2008173198 A JP2008173198 A JP 2008173198A JP 2008173198 A JP2008173198 A JP 2008173198A JP 2009040767 A5 JP2009040767 A5 JP 2009040767A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- pharmaceutically acceptable
- solvate
- acceptable salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- 150000001875 compounds Chemical class 0.000 claims 11
- 150000003839 salts Chemical class 0.000 claims 9
- 239000012453 solvate Substances 0.000 claims 9
- -1 4-methylpent-1-yl Chemical group 0.000 claims 7
- 125000000217 alkyl group Chemical group 0.000 claims 3
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 claims 2
- 125000004210 cyclohexylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C1([H])[H] 0.000 claims 2
- 239000003814 drug Substances 0.000 claims 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 2
- PNYZSYOQKIXTEL-QMMMGPOBSA-N (2s)-2-amino-3-cyclobutyl-2-methylpropanoic acid Chemical compound OC(=O)[C@](N)(C)CC1CCC1 PNYZSYOQKIXTEL-QMMMGPOBSA-N 0.000 claims 1
- ASDHRKWLZHKRQV-VIFPVBQESA-N (2s)-2-amino-3-cyclopentyl-2-methylpropanoic acid Chemical compound OC(=O)[C@](N)(C)CC1CCCC1 ASDHRKWLZHKRQV-VIFPVBQESA-N 0.000 claims 1
- ZIMXPVDWRPAZJL-JTQLQIEISA-N (2s)-2-amino-5-ethyl-2-methylheptanoic acid Chemical compound CCC(CC)CC[C@](C)(N)C(O)=O ZIMXPVDWRPAZJL-JTQLQIEISA-N 0.000 claims 1
- VHWJJTKKTVOZNB-APPZFPTMSA-N (2s,5r)-2-amino-2,5-dimethylheptanoic acid Chemical compound CC[C@@H](C)CC[C@](C)(N)C(O)=O VHWJJTKKTVOZNB-APPZFPTMSA-N 0.000 claims 1
- 125000004493 2-methylbut-1-yl group Chemical group CC(C*)CC 0.000 claims 1
- 125000004850 cyclobutylmethyl group Chemical group C1(CCC1)C* 0.000 claims 1
- 125000004851 cyclopentylmethyl group Chemical group C1(CCCC1)C* 0.000 claims 1
- 125000001153 fluoro group Chemical group F* 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
- 239000008194 pharmaceutical composition Substances 0.000 claims 1
- 239000000546 pharmaceutical excipient Substances 0.000 claims 1
- 229940124597 therapeutic agent Drugs 0.000 claims 1
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US67602505P | 2005-04-28 | 2005-04-28 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008508341A Division JP4173909B1 (ja) | 2005-04-28 | 2006-04-19 | アミノ酸誘導体 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009040767A JP2009040767A (ja) | 2009-02-26 |
| JP2009040767A5 true JP2009040767A5 (hr) | 2009-05-28 |
Family
ID=36677128
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008508341A Expired - Fee Related JP4173909B1 (ja) | 2005-04-28 | 2006-04-19 | アミノ酸誘導体 |
| JP2008173198A Ceased JP2009040767A (ja) | 2005-04-28 | 2008-07-02 | アミノ酸誘導体 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008508341A Expired - Fee Related JP4173909B1 (ja) | 2005-04-28 | 2006-04-19 | アミノ酸誘導体 |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US7612226B2 (hr) |
| EP (1) | EP1879567A1 (hr) |
| JP (2) | JP4173909B1 (hr) |
| KR (1) | KR100925900B1 (hr) |
| CN (1) | CN101166524B (hr) |
| AP (1) | AP2007004161A0 (hr) |
| AR (1) | AR054441A1 (hr) |
| AU (1) | AU2006238933B2 (hr) |
| BR (1) | BRPI0609879A2 (hr) |
| CA (1) | CA2606353C (hr) |
| CR (1) | CR9472A (hr) |
| DO (1) | DOP2006000095A (hr) |
| EA (1) | EA200701852A1 (hr) |
| GT (1) | GT200600178A (hr) |
| HK (1) | HK1116417A1 (hr) |
| IL (1) | IL185790A0 (hr) |
| MA (1) | MA29408B1 (hr) |
| MX (1) | MX2007010978A (hr) |
| NL (1) | NL1031705C2 (hr) |
| NO (1) | NO20076000L (hr) |
| PE (1) | PE20061435A1 (hr) |
| SV (1) | SV2008002512A (hr) |
| TN (1) | TNSN07400A1 (hr) |
| TW (1) | TW200719889A (hr) |
| UY (1) | UY29498A1 (hr) |
| WO (1) | WO2006114707A1 (hr) |
| ZA (1) | ZA200707678B (hr) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL126999A (en) | 1996-07-24 | 2002-03-10 | Warner Lambert Co | Pharmaceutical preparations containing isobutylgaba and its history for use in the treatment of pain |
| AP2007004161A0 (en) * | 2005-04-28 | 2007-10-31 | Pfizer Ltd | Amino acid derivatives |
| US20090227680A1 (en) * | 2005-11-17 | 2009-09-10 | Pfizer, Inc. | Amino Acid Derivatives |
| US8278355B2 (en) | 2006-09-12 | 2012-10-02 | Therexcell Pharma Inc. | Isovaline for treatment of pain |
| CN101195583B (zh) * | 2006-12-04 | 2012-07-04 | 四川抗菌素工业研究所有限公司 | 一种光学纯米那普仑及其盐的制备方法 |
| PL2334638T3 (pl) * | 2008-09-09 | 2019-04-30 | Hoffmann La Roche | Polimorfy acylosulfonoamidów |
| JP2012176902A (ja) * | 2011-02-25 | 2012-09-13 | Tosoh F-Tech Inc | 新規な光学活性含フッ素化合物、その製造方法及びそれを用いた光学活性３，３，３−トリフルオロアラニンの製造方法 |
| AT514349B1 (de) * | 2013-06-12 | 2018-05-15 | Red Bull Gmbh | Alpha-alkylierte Aminosäuren (AAAAs) |
Family Cites Families (60)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB504209A (en) | 1937-12-14 | 1939-04-21 | Pirelli General Cable Works | Improvements in or relating to electric cables |
| BR6239521D0 (pt) * | 1961-08-09 | 1973-06-14 | Merck & Co Inc | Processo de preparacao de novos amino acidos |
| FR2586562B1 (fr) | 1985-09-02 | 1989-03-10 | Inst Nat Sante Rech Med | Composition pharmaceutique contenant de l'a-methylhistamine |
| DE3811256A1 (de) | 1988-04-02 | 1989-10-19 | Hoechst Ag | (alpha)-trifluormethylaminosaeure-derivate, verfahren zur herstellung von (alpha)-trifluormethylaminosaeure-derivaten und ihre verwendung als arzneimittel |
| EP0484437A4 (en) | 1989-07-27 | 1994-06-01 | Searle & Co | Renal-selective prodrugs for the treatment of hypertension |
| FR2681067B1 (fr) * | 1991-09-10 | 1993-12-17 | Elf Sanofi | Derives heterocycliques n-substitues, leur preparation, les compositions pharmaceutiques en contenant. |
| JPH042899A (ja) | 1990-04-16 | 1992-01-07 | Arakawa Chem Ind Co Ltd | 紙用サイズ剤および該サイズ剤を用いる紙サイジング方法 |
| FR2661909B1 (fr) | 1990-05-09 | 1997-08-14 | Inst Nat Sante Rech Med | Nouveaux composes agonistes du recepteur h3 de l'histamine a usage therapeutique, compositions pharmaceutiques agissant comme agonistes dudit recepteur et procede de preparation. |
| JPH051002A (ja) | 1991-02-15 | 1993-01-08 | Nikko Kyodo Co Ltd | α−アミノ酸の製造方法 |
| CA2068038A1 (en) | 1991-05-08 | 1992-11-09 | Christopher Yee | Enzymatic resolution of .alpha.-tertiary carboxylic acid esters |
| US5993775A (en) | 1991-11-27 | 1999-11-30 | Diatide, Inc. | Radioactively labeled peptides comprising a single thiol moiety |
| GB9200210D0 (en) | 1992-01-07 | 1992-02-26 | British Bio Technology | Compounds |
| US5786373A (en) | 1992-10-14 | 1998-07-28 | Merck & Co., Inc. | Fibrinogen receptor antagonists |
| US5362747A (en) | 1992-11-25 | 1994-11-08 | Abbott Laboratories | 2-nitroaryl and 2-cyanoaryl compounds as regulators of nitric oxide synthase |
| GB9325360D0 (en) | 1993-12-10 | 1994-02-16 | Univ Bristol | Organic compounds |
| GB9325368D0 (en) | 1993-12-10 | 1994-02-16 | Univ Bristol | Organic compounds |
| IS4261A (is) | 1994-02-21 | 1995-08-22 | Astra Aktiebolag | Nýir peptíð-ópíóíðar til meðhöndlunar á verkjum og notkun þeirra |
| DE19533617A1 (de) | 1995-09-11 | 1997-03-13 | Degussa | Neues Verfahren zur Herstellung von optisch aktiven alpha-Aminosäuren und alpha-Aminosäure-Derivaten |
| DE69624081T2 (de) | 1995-12-20 | 2003-06-12 | Hoffmann La Roche | Matrix-metalloprotease Inhibitoren |
| WO1998014208A1 (en) | 1996-09-30 | 1998-04-09 | President And Fellows Of Harvard College | Reactive ligands and covalent ligand-protein complexes |
| US5962523A (en) | 1996-10-25 | 1999-10-05 | Discovery Laboratories, Inc. | Methods of using butyric acid derivatives to protect against hair loss |
| JPH10333511A (ja) | 1997-05-30 | 1998-12-18 | Ricoh Co Ltd | 画像除去促進液、該画像除去促進液を用いた被記録材の再生方法及び再生装置 |
| JP4205191B2 (ja) | 1997-12-26 | 2009-01-07 | ダイセル化学工業株式会社 | α−アミノニトリル誘導体及びα−アミノ酸の製造方法 |
| ES2220257T1 (es) | 1998-03-11 | 2004-12-16 | Kabushiki Kaisha Soken | Agentes normalizadores para la piel. |
| JP2002512214A (ja) * | 1998-04-17 | 2002-04-23 | ケネス カリー， | 代謝生成物産生グルタミン酸レセプターアンタゴニストとしてのキュバン誘導体およびそれらの調製プロセス |
| DK1140945T3 (da) | 1998-12-18 | 2003-09-15 | Novo Nordisk As | Kondenserede 1,2,4-thiadiazinderivater, deres fremstilling og anvendelse |
| WO2000037422A2 (en) | 1998-12-22 | 2000-06-29 | Neurosearch A/S | Ion channel modulating agents |
| FR2788271B1 (fr) | 1999-01-07 | 2001-02-09 | Rhone Poulenc Agrochimie | Nouveau procede de preparation d'aminoacides chiraux |
| JP2002535302A (ja) | 1999-01-22 | 2002-10-22 | ファーマコア，インコーポレイテッド | 化学式１の化合物およびその誘導体の合成方法 |
| KR100440643B1 (ko) | 1999-01-28 | 2004-07-21 | 쥬가이 세이야쿠 가부시키가이샤 | 치환 페네틸아민 유도체 |
| FR2791982B1 (fr) | 1999-04-06 | 2002-12-27 | Inst Nat Sante Rech Med | Inhibiteurs de lta4 hydrolase et leurs applications therapeutiques. |
| WO2001009117A1 (en) | 1999-07-29 | 2001-02-08 | Allellix Neuroscience Inc. | Tricyclic compounds as glycine transport inhibitors |
| FR2796943A1 (fr) | 1999-07-30 | 2001-02-02 | Aventis Pharma Sa | Derives de benzoxazinnes, leur procede de preparation et leur utilisation en therapeutique |
| EP1210933A4 (en) | 1999-09-07 | 2003-01-22 | Soken Kk | SKIN CARE AGENTS |
| JP4728548B2 (ja) | 1999-09-07 | 2011-07-20 | 三菱レイヨン株式会社 | 光学活性アミノアルコールの製造方法 |
| JP2001081013A (ja) | 1999-09-10 | 2001-03-27 | Soken Kk | 毛髪健全化剤 |
| US7300775B2 (en) | 1999-12-29 | 2007-11-27 | Verenium Corporation | Methods for producing α-substituted carboxylic acids using nitrilases and strecker reagents |
| US6656958B2 (en) | 2000-02-02 | 2003-12-02 | Abbott Laboratories | Substituted pyridine compounds useful for controlling chemical synaptic transmission |
| DE10121028A1 (de) | 2000-05-05 | 2002-01-31 | Basf Ag | Verfahren zur Herstellung von Aldehyden |
| DE10121026A1 (de) | 2000-05-05 | 2002-02-07 | Basf Ag | Verfahren zur Herstellung von Aldehyden |
| EP1300392B1 (en) | 2000-05-18 | 2012-09-05 | Mitsubishi Rayon Co., Ltd. | Process for producing optically active alpha-amino acid and optically active alpha-amino acid amide |
| WO2003011799A1 (en) | 2000-07-31 | 2003-02-13 | Brandeis University | Kinetic resolutions of chirat 3- and 3-substituted carboxylic acids |
| DE10048715A1 (de) | 2000-09-30 | 2004-05-19 | Grünenthal GmbH | Verwendung von Aminosäure zur Behandlung von Schmerz |
| AUPR406901A0 (en) | 2001-03-29 | 2001-04-26 | La Trobe University | Insecticide and method of controlling insects |
| JP4715058B2 (ja) | 2001-08-02 | 2011-07-06 | Ｊｓｒ株式会社 | 感放射性樹脂組成物 |
| JP2003221328A (ja) | 2002-01-29 | 2003-08-05 | Soken Kk | 皮膚健全化剤 |
| JP4414331B2 (ja) | 2002-05-15 | 2010-02-10 | ジェンザイム、コーポレーション | ベンゾニトリルおよびベンズイミデートの合成 |
| WO2004013112A1 (en) | 2002-08-01 | 2004-02-12 | Basf Aktiengesellschaft | Pesticidal fluoroalkene derivatives |
| US20060025471A1 (en) * | 2002-09-13 | 2006-02-02 | Kenneth Curry | Xanthenyl cubane analogs with activity at the metabotropic glutamate receptors |
| EP1584690A1 (en) | 2003-01-10 | 2005-10-12 | Kaneka Corporation | PROCESS FOR PRODUCING OPTICALLY ACTIVE a-METHYLCYSTEINE DERIVATIVE |
| JP2005060311A (ja) | 2003-08-13 | 2005-03-10 | Mochida Pharmaceut Co Ltd | Ｎ−（ベンゾイル）アミノ酸誘導体を有効成分とするニューロパシー性疼痛治療剤 |
| GB0322140D0 (en) * | 2003-09-22 | 2003-10-22 | Pfizer Ltd | Combinations |
| WO2005044780A1 (ja) | 2003-11-10 | 2005-05-19 | Kyorin Pharmaceutical Co., Ltd. | アミノカルボン酸誘導体とその付加塩及びｓ１ｐ受容体調節剤 |
| CA2554735A1 (en) * | 2004-01-30 | 2005-08-11 | Peplin Biolipids Pty Ltd | Therapeutic and carrier molecules |
| GB0405289D0 (en) | 2004-03-09 | 2004-04-21 | Novartis Ag | Organic compounds |
| CA2599662A1 (en) | 2005-03-01 | 2006-09-08 | Pfizer Limited | Use of pde7 inhibitors for the treatment of neuropathic pain |
| TW200642687A (en) * | 2005-03-01 | 2006-12-16 | Pfizer Ltd | Combinations comprising α-2-δ ligands |
| JP4521463B2 (ja) * | 2005-03-17 | 2010-08-11 | ファイザー株式会社 | 疼痛の治療に有用なｎ−（ｎ−スルホニルアミノメチル）シクロプロパンカルボキサミド誘導体 |
| AP2007004161A0 (en) * | 2005-04-28 | 2007-10-31 | Pfizer Ltd | Amino acid derivatives |
| JP2009517453A (ja) * | 2005-12-02 | 2009-04-30 | ファイザー・リミテッド | Ｐｄｅ７阻害剤としてのスピロ環式キナゾリン誘導体 |
-
2006
- 2006-04-19 AP AP2007004161A patent/AP2007004161A0/xx unknown
- 2006-04-19 CN CN2006800141982A patent/CN101166524B/zh not_active Expired - Fee Related
- 2006-04-19 AU AU2006238933A patent/AU2006238933B2/en not_active Ceased
- 2006-04-19 WO PCT/IB2006/001086 patent/WO2006114707A1/en active Application Filing
- 2006-04-19 KR KR1020077024860A patent/KR100925900B1/ko not_active IP Right Cessation
- 2006-04-19 MX MX2007010978A patent/MX2007010978A/es active IP Right Grant
- 2006-04-19 BR BRPI0609879-7A patent/BRPI0609879A2/pt not_active Application Discontinuation
- 2006-04-19 EP EP06727559A patent/EP1879567A1/en not_active Withdrawn
- 2006-04-19 CA CA2606353A patent/CA2606353C/en not_active Expired - Fee Related
- 2006-04-19 JP JP2008508341A patent/JP4173909B1/ja not_active Expired - Fee Related
- 2006-04-19 EA EA200701852A patent/EA200701852A1/ru unknown
- 2006-04-25 PE PE2006000431A patent/PE20061435A1/es not_active Application Discontinuation
- 2006-04-26 UY UY29498A patent/UY29498A1/es not_active Application Discontinuation
- 2006-04-26 AR ARP060101665A patent/AR054441A1/es not_active Application Discontinuation
- 2006-04-26 DO DO2006000095A patent/DOP2006000095A/es unknown
- 2006-04-27 TW TW095115092A patent/TW200719889A/zh unknown
- 2006-04-27 NL NL1031705A patent/NL1031705C2/nl not_active IP Right Cessation
- 2006-04-27 GT GT200600178A patent/GT200600178A/es unknown
- 2006-04-28 SV SV2006002512A patent/SV2008002512A/es not_active Application Discontinuation
- 2006-04-28 US US11/414,422 patent/US7612226B2/en not_active Expired - Fee Related
-
2007
- 2007-09-06 ZA ZA200707678A patent/ZA200707678B/xx unknown
- 2007-09-06 IL IL185790A patent/IL185790A0/en unknown
- 2007-10-25 CR CR9472A patent/CR9472A/es unknown
- 2007-10-26 TN TNP2007000400A patent/TNSN07400A1/fr unknown
- 2007-10-26 MA MA30323A patent/MA29408B1/fr unknown
- 2007-11-21 NO NO20076000A patent/NO20076000L/no not_active Application Discontinuation
-
2008
- 2008-06-18 HK HK08106675.1A patent/HK1116417A1/xx not_active IP Right Cessation
- 2008-07-02 JP JP2008173198A patent/JP2009040767A/ja not_active Ceased
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