JP2008503473A - Ｃ−ｋｉｔ活性を調節する化合物 - Google Patents
Ｃ−ｋｉｔ活性を調節する化合物 Download PDFInfo
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Classifications
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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- A—HUMAN NECESSITIES
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Landscapes
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- Otolaryngology (AREA)
- Physical Education & Sports Medicine (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
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| US58089804P | 2004-06-17 | 2004-06-17 | |
| US68207605P | 2005-05-17 | 2005-05-17 | |
| US68205805P | 2005-05-17 | 2005-05-17 | |
| PCT/US2005/021231 WO2006009755A2 (en) | 2004-06-17 | 2005-06-16 | Azaindoles modulating c-kit activity and uses therefor |
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| JP2008503473A true JP2008503473A (ja) | 2008-02-07 |
| JP2008503473A5 JP2008503473A5 (enExample) | 2008-07-31 |
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| JP2007516717A Pending JP2008503473A (ja) | 2004-06-17 | 2005-06-16 | Ｃ−ｋｉｔ活性を調節する化合物 |
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| Country | Link |
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| US (1) | US20060058339A1 (enExample) |
| EP (1) | EP1755597A2 (enExample) |
| JP (1) | JP2008503473A (enExample) |
| AU (1) | AU2005265017A1 (enExample) |
| CA (1) | CA2570817A1 (enExample) |
| PA (1) | PA8637601A1 (enExample) |
| SV (1) | SV2005002148A (enExample) |
| TW (1) | TW200616632A (enExample) |
| WO (2) | WO2006009755A2 (enExample) |
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2008545652A (ja) * | 2005-05-17 | 2008-12-18 | プレキシコン，インコーポレーテッド | ｃ−ｋｉｔおよびｃ−ｆｍｓ活性を調節する化合物およびその用途 |
| JP2008546797A (ja) * | 2005-06-22 | 2008-12-25 | プレキシコン，インコーポレーテッド | キナーゼ調節のための化合物および方法，およびその適応症 |
| JP2012517465A (ja) * | 2009-02-12 | 2012-08-02 | オリバーズ・ファルマ | プロテインキナーゼａｂｌおよびｓｒｃの阻害剤としてのアザインドール誘導体 |
| JP2013510166A (ja) * | 2009-11-06 | 2013-03-21 | プレキシコン インコーポレーテッド | キナーゼ調節のための化合物、方法およびその適用 |
| JP2018524381A (ja) * | 2015-07-20 | 2018-08-30 | ジェンザイム・コーポレーション | コロニー刺激因子−１受容体（ｃｓｆ−１ｒ）阻害剤 |
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| JP2016106090A (ja) * | 2009-11-06 | 2016-06-16 | プレキシコン インコーポレーテッドＰｌｅｘｘｉｋｏｎ Ｉｎｃ． | キナーゼ調節のための化合物、方法およびその適用 |
| JP2018524381A (ja) * | 2015-07-20 | 2018-08-30 | ジェンザイム・コーポレーション | コロニー刺激因子−１受容体（ｃｓｆ−１ｒ）阻害剤 |
| US11274108B2 (en) | 2015-07-20 | 2022-03-15 | Genzyme Corporation | Colony stimulating factor-1 receptor (CSF-1R) inhibitors |
| JP2025094019A (ja) * | 2015-07-20 | 2025-06-24 | ジェンザイム・コーポレーション | コロニー刺激因子－１受容体（ｃｓｆ－１ｒ）阻害剤 |
| US12503477B2 (en) | 2015-07-20 | 2025-12-23 | Genzyme Corporation | Colony stimulating factor-1 receptor (CSF-1R) inhibitors |
| US11530216B2 (en) | 2020-12-23 | 2022-12-20 | Genzyme Corporation | Deuterated colony stimulating factor-1 receptor (CSF-1R) inhibitors |
Also Published As
| Publication number | Publication date |
|---|---|
| PA8637601A1 (es) | 2006-06-02 |
| CA2570817A1 (en) | 2006-01-26 |
| SV2005002148A (es) | 2005-12-09 |
| WO2006009755A3 (en) | 2006-04-20 |
| WO2006009797A1 (en) | 2006-01-26 |
| WO2006009755A2 (en) | 2006-01-26 |
| US20060058339A1 (en) | 2006-03-16 |
| AU2005265017A1 (en) | 2006-01-26 |
| TW200616632A (en) | 2006-06-01 |
| EP1755597A2 (en) | 2007-02-28 |
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