JP2008500971A5 - - Google Patents

Download PDF

Info

Publication number
JP2008500971A5
JP2008500971A5 JP2007512736A JP2007512736A JP2008500971A5 JP 2008500971 A5 JP2008500971 A5 JP 2008500971A5 JP 2007512736 A JP2007512736 A JP 2007512736A JP 2007512736 A JP2007512736 A JP 2007512736A JP 2008500971 A5 JP2008500971 A5 JP 2008500971A5
Authority
JP
Japan
Prior art keywords
phe
gly
asp
arg
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2007512736A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008500971A (ja
Filing date
Publication date
Priority claimed from IT000239A external-priority patent/ITRM20040239A1/it
Application filed filed Critical
Publication of JP2008500971A publication Critical patent/JP2008500971A/ja
Publication of JP2008500971A5 publication Critical patent/JP2008500971A5/ja
Withdrawn legal-status Critical Current

Links

JP2007512736A 2004-05-13 2005-05-04 抗−インテグリン活性を有するシクロペプチド誘導体 Withdrawn JP2008500971A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT000239A ITRM20040239A1 (it) 2004-05-13 2004-05-13 Derivati ciclopeptidici ad attivita' antintegrine.
PCT/IT2005/000262 WO2005111064A1 (en) 2004-05-13 2005-05-04 Cyclopeptide derivatives with anti-integrin activity

Publications (2)

Publication Number Publication Date
JP2008500971A JP2008500971A (ja) 2008-01-17
JP2008500971A5 true JP2008500971A5 (enExample) 2008-06-26

Family

ID=34968013

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007512736A Withdrawn JP2008500971A (ja) 2004-05-13 2005-05-04 抗−インテグリン活性を有するシクロペプチド誘導体

Country Status (23)

Country Link
US (1) US20070178045A1 (enExample)
EP (1) EP1751176B1 (enExample)
JP (1) JP2008500971A (enExample)
KR (1) KR20070012524A (enExample)
CN (1) CN1953990A (enExample)
AR (1) AR048957A1 (enExample)
AT (1) ATE460426T1 (enExample)
AU (1) AU2005243418A1 (enExample)
BR (1) BRPI0510985A (enExample)
CA (1) CA2562576A1 (enExample)
CY (1) CY1110039T1 (enExample)
DE (1) DE602005019876D1 (enExample)
DK (1) DK1751176T3 (enExample)
ES (1) ES2340862T3 (enExample)
HR (1) HRP20100301T1 (enExample)
IT (1) ITRM20040239A1 (enExample)
MX (1) MXPA06012887A (enExample)
PL (1) PL1751176T3 (enExample)
PT (1) PT1751176E (enExample)
RS (1) RS51300B (enExample)
SI (1) SI1751176T1 (enExample)
TW (1) TW200606178A (enExample)
WO (1) WO2005111064A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2436109T3 (es) * 2006-02-09 2013-12-27 Belrose Pharma Inc. Conjugados poliméricos de múltiples brazos de 7-etil-10-hidroxicamptotecina para el tratamiento del cáncer de mama, del cáncer colorrectal, del cáncer de páncreas, de ovario y de pulmón
EP1961759A1 (en) * 2007-02-21 2008-08-27 Universita'degli Studi Di Milano Integrin targeted cyclopeptide ligands, their preparation and use
TWI474819B (zh) 2012-05-15 2015-03-01 國立成功大學 調控物及含有該調控物之醫藥組合物
JP2016515120A (ja) * 2013-03-15 2016-05-26 バイオジェン・エムエイ・インコーポレイテッドBiogen MA Inc. 抗アルファvベータ5抗体を用いた急性腎損傷の治療及び予防
CN103588863B (zh) * 2013-11-15 2016-08-17 苏州强耀生物科技有限公司 Rgd环肽合成制备工艺
WO2022183360A1 (en) * 2021-03-02 2022-09-09 Tsao Yeou Ping Short synthetic peptide and their uses for treating dry eye disease

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4310643A1 (de) * 1993-04-01 1994-10-06 Merck Patent Gmbh Cyclische Adhäsionsinhibitoren
US5449761A (en) * 1993-09-28 1995-09-12 Cytogen Corporation Metal-binding targeted polypeptide constructs
US6027711A (en) * 1995-06-07 2000-02-22 Rhomed Incorporated Structurally determined metallo-constructs and applications
DE19725368A1 (de) * 1997-06-16 1998-12-17 Merck Patent Gmbh Cyclische Adhäsionsinhibitoren und deren Verwendung für bildgebende Verfahren
ITRM20040240A1 (it) * 2004-05-13 2004-08-13 Ist Naz Stud Cura Dei Tumori Camptotecine coniugate in posizione 7 con antagonisti delle integrine.
ITRM20040242A1 (it) * 2004-05-13 2004-08-13 Ist Naz Stud Cura Dei Tumori "7-t-butossiimminometilcamptotecina coniugata in posizione 20 con antagonisti delle integrine.

Similar Documents

Publication Publication Date Title
CN104586859B (zh) 喹硫平的氨基酸缀合物、其制备和使用方法
ES2892954T3 (es) Derivados fluorados del ácido 3-(2-oxo-3-(3-(5,6,7,8-tetrahidro-1,8-naftiridin-2-il)propil)imidazolidin-1-il)propanoico y usos de los mismos
KR20120089806A (ko) 구안파신의 전구 약물
JP2011523412A5 (enExample)
RU2003137593A (ru) Соединения на основе пептидов для направленной доставки к рецепторам интегринов
KR20170141757A (ko) 테트라하이드로나프티리디닐 프로피온산 유도체 및 이의 용도
EP3442990A1 (en) Chiral peptides
EP4072561A1 (en) Methods of treating cancer
CN118679146A (zh) 色胺前药
RU2608388C2 (ru) Сложные эфиры пентамидин-амидоксим кислот как пролекарства и их применение в качестве лекарственных средств
JP7229482B2 (ja) 新規アミド系化合物、並びにそれを用いたPin1阻害剤、炎症性疾患の治療剤及び癌の治療剤
JP6952911B2 (ja) 2−(αヒドロキシペンチル)安息香酸の有機アミンエステル誘導体薬物
CN110662540A (zh) 用于治疗癌症的瑞格菲尼和pd-1/pd-l1(2)抑制剂的组合产品
JP5253155B2 (ja) 肥満治療に有用なmao−b阻害剤
US8598180B2 (en) Tetrahydroindolone derivatives for treatment of neurological conditions
HRP20100301T1 (hr) Ciklopeptidni derivati sa anti-integrinskom aktivnošću
ES2553891T3 (es) Derivados de piridina como moduladores NET/SERT
JP2002212070A (ja) アスパラギン酸誘導体を有効成分として含有するスフィンゴシン−1−リン酸拮抗剤
KR20240142499A (ko) Ntsr1-표적화 방사성제약 및 dna 손상 반응 억제제 조합 요법
WO2021002481A1 (ja) 生分解性に優れる腎ターゲティング型薬物送達用担体
JP6429399B2 (ja) 抗プリオン化合物のマレイン酸塩及びその製造方法、並びにその医薬組成物
US20130116298A1 (en) Antitumor agent or postoperative adjuvant chemotherapeutic agent for hepatocellular carcinoma treatment
RU2692078C2 (ru) Конъюгат, содержащий фолиевую кислоту и индол-3-карбинол, для медицинского применения
KR20170016822A (ko) 소수성 약물 전달용 신규한 폴리머계 하이드로트로프
WO2015192052A1 (en) Egfr targeting compounds and methods of use thereof