PT1751176E - Derivados ciclopeptídicos que possuem actividade anti-integrina - Google Patents
Derivados ciclopeptídicos que possuem actividade anti-integrina Download PDFInfo
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- PT1751176E PT1751176E PT05742999T PT05742999T PT1751176E PT 1751176 E PT1751176 E PT 1751176E PT 05742999 T PT05742999 T PT 05742999T PT 05742999 T PT05742999 T PT 05742999T PT 1751176 E PT1751176 E PT 1751176E
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Classifications
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- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
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- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
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- A—HUMAN NECESSITIES
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- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/64—Cyclic peptides containing only normal peptide links
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
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- Oncology (AREA)
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- Urology & Nephrology (AREA)
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- Gastroenterology & Hepatology (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT000239A ITRM20040239A1 (it) | 2004-05-13 | 2004-05-13 | Derivati ciclopeptidici ad attivita' antintegrine. |
Publications (1)
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|---|---|
| PT1751176E true PT1751176E (pt) | 2010-05-12 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT05742999T PT1751176E (pt) | 2004-05-13 | 2005-05-04 | Derivados ciclopeptídicos que possuem actividade anti-integrina |
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| Country | Link |
|---|---|
| US (1) | US20070178045A1 (enExample) |
| EP (1) | EP1751176B1 (enExample) |
| JP (1) | JP2008500971A (enExample) |
| KR (1) | KR20070012524A (enExample) |
| CN (1) | CN1953990A (enExample) |
| AR (1) | AR048957A1 (enExample) |
| AT (1) | ATE460426T1 (enExample) |
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| BR (1) | BRPI0510985A (enExample) |
| CA (1) | CA2562576A1 (enExample) |
| CY (1) | CY1110039T1 (enExample) |
| DE (1) | DE602005019876D1 (enExample) |
| DK (1) | DK1751176T3 (enExample) |
| ES (1) | ES2340862T3 (enExample) |
| HR (1) | HRP20100301T1 (enExample) |
| IT (1) | ITRM20040239A1 (enExample) |
| MX (1) | MXPA06012887A (enExample) |
| PL (1) | PL1751176T3 (enExample) |
| PT (1) | PT1751176E (enExample) |
| RS (1) | RS51300B (enExample) |
| SI (1) | SI1751176T1 (enExample) |
| TW (1) | TW200606178A (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| ES2436109T3 (es) * | 2006-02-09 | 2013-12-27 | Belrose Pharma Inc. | Conjugados poliméricos de múltiples brazos de 7-etil-10-hidroxicamptotecina para el tratamiento del cáncer de mama, del cáncer colorrectal, del cáncer de páncreas, de ovario y de pulmón |
| EP1961759A1 (en) * | 2007-02-21 | 2008-08-27 | Universita'degli Studi Di Milano | Integrin targeted cyclopeptide ligands, their preparation and use |
| TWI474819B (zh) | 2012-05-15 | 2015-03-01 | 國立成功大學 | 調控物及含有該調控物之醫藥組合物 |
| JP2016515120A (ja) * | 2013-03-15 | 2016-05-26 | バイオジェン・エムエイ・インコーポレイテッドＢｉｏｇｅｎ ＭＡ Ｉｎｃ． | 抗アルファｖベータ５抗体を用いた急性腎損傷の治療及び予防 |
| CN103588863B (zh) * | 2013-11-15 | 2016-08-17 | 苏州强耀生物科技有限公司 | Rgd环肽合成制备工艺 |
| WO2022183360A1 (en) * | 2021-03-02 | 2022-09-09 | Tsao Yeou Ping | Short synthetic peptide and their uses for treating dry eye disease |
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| DE4310643A1 (de) * | 1993-04-01 | 1994-10-06 | Merck Patent Gmbh | Cyclische Adhäsionsinhibitoren |
| US5449761A (en) * | 1993-09-28 | 1995-09-12 | Cytogen Corporation | Metal-binding targeted polypeptide constructs |
| US6027711A (en) * | 1995-06-07 | 2000-02-22 | Rhomed Incorporated | Structurally determined metallo-constructs and applications |
| DE19725368A1 (de) * | 1997-06-16 | 1998-12-17 | Merck Patent Gmbh | Cyclische Adhäsionsinhibitoren und deren Verwendung für bildgebende Verfahren |
| ITRM20040240A1 (it) * | 2004-05-13 | 2004-08-13 | Ist Naz Stud Cura Dei Tumori | Camptotecine coniugate in posizione 7 con antagonisti delle integrine. |
| ITRM20040242A1 (it) * | 2004-05-13 | 2004-08-13 | Ist Naz Stud Cura Dei Tumori | "7-t-butossiimminometilcamptotecina coniugata in posizione 20 con antagonisti delle integrine. |
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2004
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2005
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- 2005-05-04 DE DE602005019876T patent/DE602005019876D1/de not_active Expired - Lifetime
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- 2005-05-04 KR KR1020067025228A patent/KR20070012524A/ko not_active Ceased
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- 2005-05-04 JP JP2007512736A patent/JP2008500971A/ja not_active Withdrawn
- 2005-05-04 RS RSP-2010/0231A patent/RS51300B/sr unknown
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- 2005-05-04 AT AT05742999T patent/ATE460426T1/de not_active IP Right Cessation
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2010
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Also Published As
| Publication number | Publication date |
|---|---|
| RS51300B (sr) | 2010-12-31 |
| HRP20100301T1 (hr) | 2010-06-30 |
| ES2340862T3 (es) | 2010-06-10 |
| WO2005111064A8 (en) | 2006-02-09 |
| JP2008500971A (ja) | 2008-01-17 |
| SI1751176T1 (sl) | 2010-06-30 |
| PL1751176T3 (pl) | 2010-08-31 |
| KR20070012524A (ko) | 2007-01-25 |
| EP1751176A1 (en) | 2007-02-14 |
| CY1110039T1 (el) | 2012-05-23 |
| TW200606178A (en) | 2006-02-16 |
| AR048957A1 (es) | 2006-06-14 |
| ATE460426T1 (de) | 2010-03-15 |
| CN1953990A (zh) | 2007-04-25 |
| US20070178045A1 (en) | 2007-08-02 |
| EP1751176B1 (en) | 2010-03-10 |
| DK1751176T3 (da) | 2010-06-14 |
| ITRM20040239A1 (it) | 2004-08-13 |
| MXPA06012887A (es) | 2007-02-15 |
| BRPI0510985A (pt) | 2007-12-04 |
| CA2562576A1 (en) | 2005-11-24 |
| DE602005019876D1 (de) | 2010-04-22 |
| WO2005111064A1 (en) | 2005-11-24 |
| AU2005243418A1 (en) | 2005-11-24 |
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