JP2007529433A5 - - Google Patents

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Publication number
JP2007529433A5
JP2007529433A5 JP2007503195A JP2007503195A JP2007529433A5 JP 2007529433 A5 JP2007529433 A5 JP 2007529433A5 JP 2007503195 A JP2007503195 A JP 2007503195A JP 2007503195 A JP2007503195 A JP 2007503195A JP 2007529433 A5 JP2007529433 A5 JP 2007529433A5
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JP
Japan
Prior art keywords
formula
compound
compounds
calcipotriol
protecting group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2007503195A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007529433A (ja
JP4667450B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/DK2005/000161 external-priority patent/WO2005087719A1/en
Publication of JP2007529433A publication Critical patent/JP2007529433A/ja
Publication of JP2007529433A5 publication Critical patent/JP2007529433A5/ja
Application granted granted Critical
Publication of JP4667450B2 publication Critical patent/JP4667450B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP2007503195A 2004-03-18 2005-03-10 ビタミンd類似体の立体選択的合成 Expired - Fee Related JP4667450B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US55396204P 2004-03-18 2004-03-18
DKPA200400454 2004-03-22
PCT/DK2005/000161 WO2005087719A1 (en) 2004-03-18 2005-03-10 Stereoselective synthesis of vitamin d analogues

Publications (3)

Publication Number Publication Date
JP2007529433A JP2007529433A (ja) 2007-10-25
JP2007529433A5 true JP2007529433A5 (https=) 2008-05-01
JP4667450B2 JP4667450B2 (ja) 2011-04-13

Family

ID=34961016

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007503195A Expired - Fee Related JP4667450B2 (ja) 2004-03-18 2005-03-10 ビタミンd類似体の立体選択的合成

Country Status (17)

Country Link
EP (1) EP1730108B1 (https=)
JP (1) JP4667450B2 (https=)
KR (1) KR100859277B1 (https=)
CN (1) CN1934078B (https=)
AR (1) AR048274A1 (https=)
AT (1) ATE390411T1 (https=)
BR (1) BRPI0507318A (https=)
CA (1) CA2555260C (https=)
CY (1) CY1108156T1 (https=)
DE (2) DE602005005645T2 (https=)
ES (1) ES2304686T3 (https=)
IL (1) IL176718A (https=)
PL (1) PL1730108T3 (https=)
RU (1) RU2380359C2 (https=)
SI (1) SI1730108T1 (https=)
TW (1) TWI324063B (https=)
WO (1) WO2005087719A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4744507B2 (ja) * 2004-04-02 2011-08-10 レオ ファーマ アクティーゼルスカブ ビタミンd類似体の合成に有用な中間体の新規製造法
CN101400649B (zh) 2006-03-17 2012-07-04 利奥制药有限公司 药物中间体的异构化
US8013189B2 (en) 2007-09-21 2011-09-06 Basf Se Accelerated amide and ester reductions with amine boranes and additives
EP2299809B1 (en) * 2008-06-17 2018-10-17 Ben Gurion University Of The Negev R&D Authority Substituted cyclohexylidene-ethylidene-octahydro-indene compounds
CN103265528B (zh) * 2013-05-10 2015-05-06 湖南千金湘江药业股份有限公司 埃索美拉唑镁的制备方法
CN106908524B (zh) * 2015-12-23 2021-05-04 重庆华邦胜凯制药有限公司 卡泊三醇中间体l及其潜在基因毒性杂质的分离与测定方法
CN107643354B (zh) * 2016-07-22 2022-02-01 重庆华邦胜凯制药有限公司 卡泊三醇起始原料a及相关杂质的分离与测定方法
ES2945426B2 (es) * 2021-12-30 2024-01-22 Laboratorios Vinas S A Procedimiento para obtener epímeros 24S a partir de derivados de vitaminas D y procedimiento de obtención de vitaminas D relacionado

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4866048A (en) * 1985-08-02 1989-09-12 Leo Pharmaceutical Products Ltd. Novel vitamin D analogues
JPH075542B2 (ja) * 1988-09-14 1995-01-25 呉羽化学工業株式会社 ビタミンd▲下3▼誘導体及びその製造方法
US5247104A (en) * 1992-11-04 1993-09-21 Wisconsin Alumni Research Foundation Preparation of 1α, 24-dihydroxyvitamin D analogs
GB9300763D0 (en) * 1993-01-15 1993-03-03 Leo Pharm Prod Ltd Chemical compound
US5449668A (en) * 1993-06-04 1995-09-12 Duphar International Research B.V. Vitamin D compounds and method of preparing these compounds
GB9524812D0 (en) * 1995-12-05 1996-02-07 Leo Pharm Prod Ltd Chemical compounds
GB9622590D0 (en) * 1996-10-30 1997-01-08 Leo Pharm Prod Ltd Chemical compounds
US6262283B1 (en) * 1996-12-06 2001-07-17 Magainin Pharmaceuticals Inc. Stereoselective synthesis of 24-hydroxylated compounds useful for the preparation of aminosterols, vitamin D analogs, and other compounds
EP1123921A4 (en) * 1998-10-23 2003-08-20 Teijin Ltd VITAMIN D 3 DERIVATIVES? AND MEDICINES FOR INFLAMMATORY RESPIRATORY DISEASES CONTAINING THEM

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