JP2007523072A5 - - Google Patents

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Publication number
JP2007523072A5
JP2007523072A5 JP2006551898A JP2006551898A JP2007523072A5 JP 2007523072 A5 JP2007523072 A5 JP 2007523072A5 JP 2006551898 A JP2006551898 A JP 2006551898A JP 2006551898 A JP2006551898 A JP 2006551898A JP 2007523072 A5 JP2007523072 A5 JP 2007523072A5
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JP
Japan
Prior art keywords
alkyl
amino
group
formula
methyl
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2006551898A
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English (en)
Japanese (ja)
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JP2007523072A (ja
JP5032851B2 (ja
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Priority claimed from PCT/GB2005/000237 external-priority patent/WO2005075439A1/en
Publication of JP2007523072A publication Critical patent/JP2007523072A/ja
Publication of JP2007523072A5 publication Critical patent/JP2007523072A5/ja
Application granted granted Critical
Publication of JP5032851B2 publication Critical patent/JP5032851B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2006551898A 2004-02-03 2005-01-31 キナゾリン誘導体 Expired - Fee Related JP5032851B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP04290274 2004-02-03
EP04290274.2 2004-02-03
PCT/GB2005/000237 WO2005075439A1 (en) 2004-02-03 2005-01-31 Quinazoline derivatives

Publications (3)

Publication Number Publication Date
JP2007523072A JP2007523072A (ja) 2007-08-16
JP2007523072A5 true JP2007523072A5 (https=) 2008-03-21
JP5032851B2 JP5032851B2 (ja) 2012-09-26

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ID=34833782

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006551898A Expired - Fee Related JP5032851B2 (ja) 2004-02-03 2005-01-31 キナゾリン誘導体

Country Status (11)

Country Link
US (1) US7632840B2 (https=)
EP (1) EP1713781B1 (https=)
JP (1) JP5032851B2 (https=)
CN (1) CN1914182B (https=)
AR (1) AR047703A1 (https=)
AT (1) ATE413389T1 (https=)
DE (1) DE602005010824D1 (https=)
ES (1) ES2315834T3 (https=)
TW (1) TW200529851A (https=)
UY (1) UY28736A1 (https=)
WO (1) WO2005075439A1 (https=)

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GB0126433D0 (en) * 2001-11-03 2002-01-02 Astrazeneca Ab Compounds
JP2005515176A (ja) * 2001-11-03 2005-05-26 アストラゼネカ アクチボラグ 抗腫瘍剤としてのキナゾリン誘導体
GB0309009D0 (en) * 2003-04-22 2003-05-28 Astrazeneca Ab Quinazoline derivatives
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AU2004272346A1 (en) * 2003-09-16 2005-03-24 Astrazeneca Ab Quinazoline derivatives
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JP2009508917A (ja) * 2005-09-20 2009-03-05 アストラゼネカ アクチボラグ 抗癌剤としてのキナゾリン誘導体
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JP2009517451A (ja) * 2005-12-02 2009-04-30 アストラゼネカ アクチボラグ Erbbチロシンキナーゼの阻害剤として使用されるキナゾリン誘導体
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GB201604329D0 (en) * 2016-03-14 2016-04-27 Univ Strathclyde Methods and systems for improving stability of a ship
CN111777620A (zh) * 2019-04-04 2020-10-16 山东轩竹医药科技有限公司 酪氨酸激酶抑制剂的新用途

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GB0326459D0 (en) 2003-11-13 2003-12-17 Astrazeneca Ab Quinazoline derivatives
AU2005250224A1 (en) 2004-06-04 2005-12-15 Astrazeneca Ab Quinazoline derivatives as ERBB receptor tyrosine kinases
EP1838712B8 (en) 2004-12-14 2011-10-12 AstraZeneca AB Pyrazolopyrimidine compounds as antitumor agents
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GB0504475D0 (en) 2005-03-04 2005-04-13 Astrazeneca Ab Chemical compounds
GB0504474D0 (en) 2005-03-04 2005-04-13 Astrazeneca Ab Chemical compounds
GB0508717D0 (en) 2005-04-29 2005-06-08 Astrazeneca Ab Chemical compounds
GB0508715D0 (en) 2005-04-29 2005-06-08 Astrazeneca Ab Chemical compounds
WO2007034144A1 (en) 2005-09-20 2007-03-29 Astrazeneca Ab 4- (ih-indazol-s-yl-amino)-quinazoline compounds as erbb receptor tyrosine kinase inhibitors for the treatment of cancer
JP2009508917A (ja) 2005-09-20 2009-03-05 アストラゼネカ アクチボラグ 抗癌剤としてのキナゾリン誘導体
JP2009517450A (ja) 2005-12-02 2009-04-30 アストラゼネカ アクチボラグ チロシンキナーゼ阻害薬としての4−アニリノ置換キナゾリン誘導体
JP2009517451A (ja) 2005-12-02 2009-04-30 アストラゼネカ アクチボラグ Erbbチロシンキナーゼの阻害剤として使用されるキナゾリン誘導体

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