JP2007511487A - ジペプチジルペプチダーゼｉｖ阻害剤の使用 - Google Patents
ジペプチジルペプチダーゼｉｖ阻害剤の使用 Download PDFInfo
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Landscapes
- Health & Medical Sciences (AREA)
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- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
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- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pyrrole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
Applications Claiming Priority (5)
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| US52056303P | 2003-11-17 | 2003-11-17 | |
| US52056203P | 2003-11-17 | 2003-11-17 | |
| US54719104P | 2004-02-24 | 2004-02-24 | |
| US54719204P | 2004-02-24 | 2004-02-24 | |
| PCT/EP2004/012990 WO2005049022A2 (en) | 2003-11-17 | 2004-11-16 | Use of dipeptidyl peptidase iv inhibitors |
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| JP2012123284A Division JP2012211146A (ja) | 2003-11-17 | 2012-05-30 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
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| JP2012123284A Withdrawn JP2012211146A (ja) | 2003-11-17 | 2012-05-30 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2014075331A Expired - Fee Related JP6312502B2 (ja) | 2003-11-17 | 2014-04-01 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2016123464A Withdrawn JP2016222677A (ja) | 2003-11-17 | 2016-06-22 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2017188912A Withdrawn JP2018039816A (ja) | 2003-11-17 | 2017-09-28 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2020119890A Pending JP2020183412A (ja) | 2003-11-17 | 2020-07-13 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
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| JP2012123284A Withdrawn JP2012211146A (ja) | 2003-11-17 | 2012-05-30 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2014075331A Expired - Fee Related JP6312502B2 (ja) | 2003-11-17 | 2014-04-01 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2016123464A Withdrawn JP2016222677A (ja) | 2003-11-17 | 2016-06-22 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2017188912A Withdrawn JP2018039816A (ja) | 2003-11-17 | 2017-09-28 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2020119890A Pending JP2020183412A (ja) | 2003-11-17 | 2020-07-13 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
Country Status (9)
| Country | Link |
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| EP (2) | EP2839832A3 (https=) |
| JP (6) | JP2007511487A (https=) |
| KR (10) | KR20120008093A (https=) |
| CN (1) | CN1905876B (https=) |
| AU (2) | AU2004290897B2 (https=) |
| BR (1) | BRPI0416628A (https=) |
| CA (1) | CA2545641A1 (https=) |
| MX (1) | MXPA06005518A (https=) |
| WO (1) | WO2005049022A2 (https=) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2011516410A (ja) * | 2008-02-27 | 2011-05-26 | ユリウス・マクシミリアンス−ウニヴェルジテート・ヴュルツブルク | 診断および治療のためのミクロＲＮＡ（ｍｉＲＮＡ）および下流標的 |
| JP2012522015A (ja) * | 2009-03-27 | 2012-09-20 | ブリストル−マイヤーズ スクイブ カンパニー | Ｄｐｐ−ｉｖ阻害剤を用いて主要有害心血管事象を予防する方法 |
| JP2016526555A (ja) * | 2013-06-26 | 2016-09-05 | ドン−ア エスティ カンパニー リミテッド | Ｄｐｐ−ｉｖ阻害剤を含有する腎疾患予防または治療用組成物 |
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| US7407955B2 (en) | 2002-08-21 | 2008-08-05 | Boehringer Ingelheim Pharma Gmbh & Co., Kg | 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
| US7420079B2 (en) | 2002-12-09 | 2008-09-02 | Bristol-Myers Squibb Company | Methods and compounds for producing dipeptidyl peptidase IV inhibitors and intermediates thereof |
| US7501426B2 (en) | 2004-02-18 | 2009-03-10 | Boehringer Ingelheim International Gmbh | 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions |
| EP1805676A1 (en) * | 2004-09-22 | 2007-07-11 | Tripath Imaging, Inc. | Methods and computer program products for analysis and optimization of marker candidates for cancer prognosis |
| DE102004054054A1 (de) | 2004-11-05 | 2006-05-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine |
| DOP2006000008A (es) | 2005-01-10 | 2006-08-31 | Arena Pharm Inc | Terapia combinada para el tratamiento de la diabetes y afecciones relacionadas y para el tratamiento de afecciones que mejoran mediante un incremento de la concentración sanguínea de glp-1 |
| AU2006239929B2 (en) | 2005-04-22 | 2011-11-03 | Alantos Pharmaceuticals Holding, Inc. | Dipeptidyl peptidase-IV inhibitors |
| DE102005035891A1 (de) | 2005-07-30 | 2007-02-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
| PE20071221A1 (es) | 2006-04-11 | 2007-12-14 | Arena Pharm Inc | Agonistas del receptor gpr119 en metodos para aumentar la masa osea y para tratar la osteoporosis y otras afecciones caracterizadas por masa osea baja, y la terapia combinada relacionada a estos agonistas |
| ES2654251T3 (es) * | 2006-04-19 | 2018-02-12 | Ludwig-Maximilians-Universität München | Hormona paratiroidea (PTH) para su utilización en el tratamiento de la isquemia |
| PE20110235A1 (es) | 2006-05-04 | 2011-04-14 | Boehringer Ingelheim Int | Combinaciones farmaceuticas que comprenden linagliptina y metmorfina |
| KR101452915B1 (ko) | 2006-05-04 | 2014-10-21 | 베링거 인겔하임 인터내셔날 게엠베하 | 다형태 |
| EP1852108A1 (en) | 2006-05-04 | 2007-11-07 | Boehringer Ingelheim Pharma GmbH & Co.KG | DPP IV inhibitor formulations |
| US20100247491A1 (en) * | 2007-02-01 | 2010-09-30 | Christof Westenfelder | Potentiation of Stem Cell Homing and Treatment of Organ Dysfunction or Organ Failure |
| PE20090938A1 (es) * | 2007-08-16 | 2009-08-08 | Boehringer Ingelheim Int | Composicion farmaceutica que comprende un derivado de benceno sustituido con glucopiranosilo |
| BRPI0815405A2 (pt) * | 2007-08-17 | 2015-02-03 | Boehringer Ingelheim Int | Compostos derivados de purina, processo para a preparação de uma composição farmacêutica e uso dos mesmos |
| PE20091730A1 (es) | 2008-04-03 | 2009-12-10 | Boehringer Ingelheim Int | Formulaciones que comprenden un inhibidor de dpp4 |
| EP2108960A1 (en) | 2008-04-07 | 2009-10-14 | Arena Pharmaceuticals, Inc. | Methods of using A G protein-coupled receptor to identify peptide YY (PYY) secretagogues and compounds useful in the treatment of conditons modulated by PYY |
| KR20190016601A (ko) | 2008-08-06 | 2019-02-18 | 베링거 인겔하임 인터내셔날 게엠베하 | 메트포르민 요법이 부적합한 환자에서의 당뇨병 치료 |
| UY32030A (es) | 2008-08-06 | 2010-03-26 | Boehringer Ingelheim Int | "tratamiento para diabetes en pacientes inapropiados para terapia con metformina" |
| CA2736421A1 (en) | 2008-09-10 | 2010-03-18 | Boehringer Ingelheim International Gmbh | Combination therapy for the treatment of diabetes and related conditions |
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| TW201036975A (en) | 2009-01-07 | 2010-10-16 | Boehringer Ingelheim Int | Treatment for diabetes in patients with inadequate glycemic control despite metformin therapy |
| AP2011005795A0 (en) | 2009-02-13 | 2011-08-31 | Boehringer Ingelheim Int | SGLT-2 inhibitor for treating type 1 diabetes mellitus, type 2 diabetes mellitus, impaired glucose tolerance or hyperglycemia. |
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| JP2011516410A (ja) * | 2008-02-27 | 2011-05-26 | ユリウス・マクシミリアンス−ウニヴェルジテート・ヴュルツブルク | 診断および治療のためのミクロＲＮＡ（ｍｉＲＮＡ）および下流標的 |
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| JP2012522015A (ja) * | 2009-03-27 | 2012-09-20 | ブリストル−マイヤーズ スクイブ カンパニー | Ｄｐｐ−ｉｖ阻害剤を用いて主要有害心血管事象を予防する方法 |
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| KR20060109911A (ko) | 2006-10-23 |
| JP2020183412A (ja) | 2020-11-12 |
| CN1905876A (zh) | 2007-01-31 |
| KR20120126133A (ko) | 2012-11-20 |
| WO2005049022A3 (en) | 2005-07-21 |
| EP1686994A2 (en) | 2006-08-09 |
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| JP2012211146A (ja) | 2012-11-01 |
| JP2014159436A (ja) | 2014-09-04 |
| AU2004290897A1 (en) | 2005-06-02 |
| BRPI0416628A (pt) | 2007-01-16 |
| EP2839832A3 (en) | 2015-06-24 |
| CN1905876B (zh) | 2010-06-09 |
| KR20150132601A (ko) | 2015-11-25 |
| EP2839832A2 (en) | 2015-02-25 |
| KR20130105741A (ko) | 2013-09-25 |
| AU2009202080A1 (en) | 2009-06-18 |
| CA2545641A1 (en) | 2005-06-02 |
| KR20120008093A (ko) | 2012-01-25 |
| WO2005049022A2 (en) | 2005-06-02 |
| KR20150028829A (ko) | 2015-03-16 |
| MXPA06005518A (es) | 2006-08-17 |
| JP2018039816A (ja) | 2018-03-15 |
| JP6312502B2 (ja) | 2018-04-18 |
| JP2016222677A (ja) | 2016-12-28 |
| KR20140089408A (ko) | 2014-07-14 |
| KR20170104639A (ko) | 2017-09-15 |
| KR20180050427A (ko) | 2018-05-14 |
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