JP2007511487A5 - - Google Patents
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- JP2007511487A5 JP2007511487A5 JP2006538825A JP2006538825A JP2007511487A5 JP 2007511487 A5 JP2007511487 A5 JP 2007511487A5 JP 2006538825 A JP2006538825 A JP 2006538825A JP 2006538825 A JP2006538825 A JP 2006538825A JP 2007511487 A5 JP2007511487 A5 JP 2007511487A5
- Authority
- JP
- Japan
- Prior art keywords
- injury
- heart failure
- drug
- dpp
- disease
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US52056303P | 2003-11-17 | 2003-11-17 | |
| US52056203P | 2003-11-17 | 2003-11-17 | |
| US54719204P | 2004-02-24 | 2004-02-24 | |
| US54719104P | 2004-02-24 | 2004-02-24 | |
| PCT/EP2004/012990 WO2005049022A2 (en) | 2003-11-17 | 2004-11-16 | Use of dipeptidyl peptidase iv inhibitors |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012123284A Division JP2012211146A (ja) | 2003-11-17 | 2012-05-30 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2007511487A JP2007511487A (ja) | 2007-05-10 |
| JP2007511487A5 true JP2007511487A5 (https=) | 2008-02-07 |
Family
ID=34623985
Family Applications (6)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006538825A Withdrawn JP2007511487A (ja) | 2003-11-17 | 2004-11-16 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2012123284A Withdrawn JP2012211146A (ja) | 2003-11-17 | 2012-05-30 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2014075331A Expired - Fee Related JP6312502B2 (ja) | 2003-11-17 | 2014-04-01 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2016123464A Withdrawn JP2016222677A (ja) | 2003-11-17 | 2016-06-22 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2017188912A Withdrawn JP2018039816A (ja) | 2003-11-17 | 2017-09-28 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2020119890A Pending JP2020183412A (ja) | 2003-11-17 | 2020-07-13 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
Family Applications After (5)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012123284A Withdrawn JP2012211146A (ja) | 2003-11-17 | 2012-05-30 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2014075331A Expired - Fee Related JP6312502B2 (ja) | 2003-11-17 | 2014-04-01 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2016123464A Withdrawn JP2016222677A (ja) | 2003-11-17 | 2016-06-22 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2017188912A Withdrawn JP2018039816A (ja) | 2003-11-17 | 2017-09-28 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
| JP2020119890A Pending JP2020183412A (ja) | 2003-11-17 | 2020-07-13 | ジペプチジルペプチダーゼｉｖ阻害剤の使用 |
Country Status (9)
| Country | Link |
|---|---|
| EP (2) | EP1686994A2 (https=) |
| JP (6) | JP2007511487A (https=) |
| KR (10) | KR20170104639A (https=) |
| CN (1) | CN1905876B (https=) |
| AU (2) | AU2004290897B2 (https=) |
| BR (1) | BRPI0416628A (https=) |
| CA (1) | CA2545641A1 (https=) |
| MX (1) | MXPA06005518A (https=) |
| WO (1) | WO2005049022A2 (https=) |
Families Citing this family (63)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7407955B2 (en) | 2002-08-21 | 2008-08-05 | Boehringer Ingelheim Pharma Gmbh & Co., Kg | 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
| US7420079B2 (en) | 2002-12-09 | 2008-09-02 | Bristol-Myers Squibb Company | Methods and compounds for producing dipeptidyl peptidase IV inhibitors and intermediates thereof |
| US7501426B2 (en) | 2004-02-18 | 2009-03-10 | Boehringer Ingelheim International Gmbh | 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions |
| CA2580795A1 (en) * | 2004-09-22 | 2006-04-06 | Tripath Imaging, Inc. | Methods and compositions for evaluating breast cancer prognosis |
| DE102004054054A1 (de) | 2004-11-05 | 2006-05-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine |
| DOP2006000008A (es) | 2005-01-10 | 2006-08-31 | Arena Pharm Inc | Terapia combinada para el tratamiento de la diabetes y afecciones relacionadas y para el tratamiento de afecciones que mejoran mediante un incremento de la concentración sanguínea de glp-1 |
| KR20080000665A (ko) | 2005-04-22 | 2008-01-02 | 알란토스 파마슈티컬즈 홀딩, 인코포레이티드 | 디펩티딜 펩티다아제-ⅳ 억제제 |
| DE102005035891A1 (de) | 2005-07-30 | 2007-02-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
| PE20071221A1 (es) | 2006-04-11 | 2007-12-14 | Arena Pharm Inc | Agonistas del receptor gpr119 en metodos para aumentar la masa osea y para tratar la osteoporosis y otras afecciones caracterizadas por masa osea baja, y la terapia combinada relacionada a estos agonistas |
| PL2007416T3 (pl) * | 2006-04-19 | 2018-05-30 | Ludwig-Maximilians-Universität München | Parathormon (PTH) do zastosowania w leczeniu niedokrwienia |
| PE20080251A1 (es) | 2006-05-04 | 2008-04-25 | Boehringer Ingelheim Int | Usos de inhibidores de dpp iv |
| EP1852108A1 (en) | 2006-05-04 | 2007-11-07 | Boehringer Ingelheim Pharma GmbH & Co.KG | DPP IV inhibitor formulations |
| EP2540725A1 (de) | 2006-05-04 | 2013-01-02 | Boehringer Ingelheim International GmbH | Polymorphe von 1-((4-Methyl-chinazolin-2-yl)methyl)-3-methyl-7-(2-butin-1-yl)-8-(3-(R)-amino-piperidin-1-yl)xanthin |
| AU2008210988B2 (en) * | 2007-02-01 | 2012-09-06 | Allocure, Inc. | Potentiation of stem cell homing and treatment of organ dysfunction or organ failure |
| CL2008002427A1 (es) * | 2007-08-16 | 2009-09-11 | Boehringer Ingelheim Int | Composicion farmaceutica que comprende 1-cloro-4-(b-d-glucopiranos-1-il)-2-[4-((s)-tetrahidrofurano-3-iloxi)bencil]-benceno combinado con 1-[(4-metilquinazolin-2-il)metil]-3-metil-7-(2-butin-1-il)-8-(3-(r)-aminopiperidin-1-il)xantina; y su uso para tratar diabetes mellitus tipo 2. |
| WO2009024542A2 (en) * | 2007-08-17 | 2009-02-26 | Boehringer Ingelheim International Gmbh | Purin derivatives for use in the treatment of fab-related diseases |
| EP2096171A1 (en) * | 2008-02-27 | 2009-09-02 | Julius-Maximilians-Universität Würzburg | MicroRNA (miRNA) and down-stream targets for diagnostic and therapeutic purposes |
| PE20091730A1 (es) | 2008-04-03 | 2009-12-10 | Boehringer Ingelheim Int | Formulaciones que comprenden un inhibidor de dpp4 |
| EP2108960A1 (en) | 2008-04-07 | 2009-10-14 | Arena Pharmaceuticals, Inc. | Methods of using A G protein-coupled receptor to identify peptide YY (PYY) secretagogues and compounds useful in the treatment of conditons modulated by PYY |
| UY32030A (es) | 2008-08-06 | 2010-03-26 | Boehringer Ingelheim Int | "tratamiento para diabetes en pacientes inapropiados para terapia con metformina" |
| BRPI0916997A2 (pt) | 2008-08-06 | 2020-12-15 | Boehringer Ingelheim International Gmbh | Inibidor de dpp-4 e seu uso |
| CN102149407A (zh) | 2008-09-10 | 2011-08-10 | 贝林格尔.英格海姆国际有限公司 | 治疗糖尿病和相关病症的组合疗法 |
| US20200155558A1 (en) | 2018-11-20 | 2020-05-21 | Boehringer Ingelheim International Gmbh | Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug |
| CN102256976A (zh) | 2008-12-23 | 2011-11-23 | 贝林格尔.英格海姆国际有限公司 | 有机化合物的盐形式 |
| AR074990A1 (es) | 2009-01-07 | 2011-03-02 | Boehringer Ingelheim Int | Tratamiento de diabetes en pacientes con un control glucemico inadecuado a pesar de la terapia con metformina |
| DK2396005T3 (da) | 2009-02-13 | 2026-02-09 | Boehringer Ingelheim Int | Sglt2 hæmmer til at forbedre glykæmisk kontrol |
| JP5685550B2 (ja) | 2009-02-13 | 2015-03-18 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Ｓｇｌｔ２阻害剤、ｄｐｐ−ｉｖ阻害剤、更に必要により抗糖尿病薬を含む医薬組成物及びその使用 |
| MX2011009852A (es) * | 2009-03-27 | 2011-09-29 | Bristol Myers Squibb Co | Metodos para prevenir episodios cardiovasculares adversos mayores con inhibidores de dipeptidil peptidasa iv. |
| AR077642A1 (es) | 2009-07-09 | 2011-09-14 | Arena Pharm Inc | Moduladores del metabolismo y el tratamiento de trastornos relacionados con el mismo |
| UY32919A (es) | 2009-10-02 | 2011-04-29 | Boehringer Ingelheim Int | Composición farmacéutica, forma de dosificación farmacéutica, procedimiento para su preparación, mé todos para su tratamiento y sus usos |
| KR20240090632A (ko) | 2009-11-27 | 2024-06-21 | 베링거 인겔하임 인터내셔날 게엠베하 | 리나글립틴과 같은 ｄｐｐ－ｉｖ 억제제를 사용한 유전자형 검사된 당뇨병 환자의 치료 |
| CA2795513A1 (en) | 2010-04-06 | 2011-10-13 | Arena Pharmaceuticals, Inc. | Modulators of the gpr119 receptor and the treatment of disorders related thereto |
| CN102946875A (zh) | 2010-05-05 | 2013-02-27 | 贝林格尔.英格海姆国际有限公司 | 组合疗法 |
| WO2011161161A1 (en) | 2010-06-24 | 2011-12-29 | Boehringer Ingelheim International Gmbh | Diabetes therapy |
| EP3323818A1 (en) | 2010-09-22 | 2018-05-23 | Arena Pharmaceuticals, Inc. | Modulators of the gpr119 receptor and the treatment of disorders related thereto |
| AR083878A1 (es) | 2010-11-15 | 2013-03-27 | Boehringer Ingelheim Int | Terapia antidiabetica vasoprotectora y cardioprotectora, linagliptina, metodo de tratamiento |
| AR085689A1 (es) | 2011-03-07 | 2013-10-23 | Boehringer Ingelheim Int | Composiciones farmaceuticas de metformina, linagliptina y un inhibidor de sglt-2 |
| US20140018371A1 (en) | 2011-04-01 | 2014-01-16 | Arena Pharmaceuticals, Inc. | Modulators Of The GPR119 Receptor And The Treatment Of Disorders Related Thereto |
| WO2012145361A1 (en) | 2011-04-19 | 2012-10-26 | Arena Pharmaceuticals, Inc. | Modulators of the gpr119 receptor and the treatment of disorders related thereto |
| US20140038889A1 (en) | 2011-04-22 | 2014-02-06 | Arena Pharmaceuticals, Inc. | Modulators Of The GPR119 Receptor And The Treatment Of Disorders Related Thereto |
| US20140051714A1 (en) | 2011-04-22 | 2014-02-20 | Arena Pharmaceuticals, Inc. | Modulators Of The GPR119 Receptor And The Treatment Of Disorders Related Thereto |
| WO2012170702A1 (en) | 2011-06-08 | 2012-12-13 | Arena Pharmaceuticals, Inc. | Modulators of the gpr119 receptor and the treatment of disorders related thereto |
| US8883800B2 (en) | 2011-07-15 | 2014-11-11 | Boehringer Ingelheim International Gmbh | Substituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions |
| WO2013055910A1 (en) | 2011-10-12 | 2013-04-18 | Arena Pharmaceuticals, Inc. | Modulators of the gpr119 receptor and the treatment of disorders related thereto |
| US9555001B2 (en) | 2012-03-07 | 2017-01-31 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition and uses thereof |
| JP6224084B2 (ja) | 2012-05-14 | 2017-11-01 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 糸球体上皮細胞関連障害及び／又はネフローゼ症候群の治療に用いるｄｐｐ−４阻害薬としてのキサンチン誘導体 |
| JP6218811B2 (ja) | 2012-05-14 | 2017-10-25 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Ｓｉｒｓ及び／又は敗血症の治療に用いるｄｐｐ−４阻害薬としてのキサンチン誘導体 |
| WO2013174767A1 (en) | 2012-05-24 | 2013-11-28 | Boehringer Ingelheim International Gmbh | A xanthine derivative as dpp -4 inhibitor for use in modifying food intake and regulating food preference |
| WO2014074668A1 (en) | 2012-11-08 | 2014-05-15 | Arena Pharmaceuticals, Inc. | Modulators of gpr119 and the treatment of disorders related thereto |
| HK1213818A1 (zh) | 2013-04-05 | 2016-07-15 | 勃林格殷格翰国际有限公司 | 依帕列净的治疗用途 |
| TR201901110T4 (tr) | 2013-04-05 | 2019-02-21 | Boehringer Ingelheim Int | Empagliflozinin terapötik kullanımları. |
| US11813275B2 (en) | 2013-04-05 | 2023-11-14 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition, methods for treating and uses thereof |
| CA2812519A1 (en) | 2013-04-05 | 2014-10-05 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition, methods for treating and uses thereof |
| EP4678242A3 (en) | 2013-04-18 | 2026-03-18 | Boehringer Ingelheim International GmbH | Pharmaceutical composition, methods for treating and uses thereof |
| CN105555275B (zh) * | 2013-06-26 | 2021-04-20 | 东亚St株式会社 | 含有dpp-iv抑制剂的用于预防和治疗肾脏疾病的组合物 |
| EP3110449B1 (en) | 2014-02-28 | 2023-06-28 | Boehringer Ingelheim International GmbH | Medical use of a dpp-4 inhibitor |
| EA201791982A1 (ru) | 2015-03-09 | 2020-02-17 | Интекрин Терапьютикс, Инк. | Способы лечения неалкогольной жировой болезни печени и/или липодистрофии |
| CN109310697A (zh) | 2016-06-10 | 2019-02-05 | 勃林格殷格翰国际有限公司 | 利格列汀和二甲双胍的组合 |
| KR20190084096A (ko) | 2016-11-10 | 2019-07-15 | 베링거 인겔하임 인터내셔날 게엠베하 | 약제학적 조성물, 치료 방법 및 이의 용도 |
| JP2020515639A (ja) | 2017-04-03 | 2020-05-28 | コヒラス・バイオサイエンシズ・インコーポレイテッド | 進行性核上性麻痺の処置のためのＰＰＡＲγアゴニスト |
| KR20190019542A (ko) | 2017-08-18 | 2019-02-27 | 현대자동차주식회사 | 차량용 쿨러 |
| KR102142559B1 (ko) | 2018-07-31 | 2020-08-07 | 가톨릭대학교 산학협력단 | Dpp4 억제제를 유효성분으로 포함하는 심근섬유증의 예방 또는 치료용 조성물 |
| JP2022548214A (ja) | 2019-09-17 | 2022-11-17 | ノバルティス アーゲー | ビルダグリプチンとメトホルミンとの組み合わせ療法 |
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-
2004
- 2004-11-16 WO PCT/EP2004/012990 patent/WO2005049022A2/en not_active Ceased
- 2004-11-16 KR KR1020177024680A patent/KR20170104639A/ko not_active Withdrawn
- 2004-11-16 BR BRPI0416628-0A patent/BRPI0416628A/pt not_active Application Discontinuation
- 2004-11-16 KR KR1020067009502A patent/KR20060109911A/ko not_active Withdrawn
- 2004-11-16 KR KR1020127028863A patent/KR20120126133A/ko not_active Withdrawn
- 2004-11-16 KR KR1020147014776A patent/KR20140089408A/ko not_active Withdrawn
- 2004-11-16 CA CA002545641A patent/CA2545641A1/en not_active Abandoned
- 2004-11-16 KR KR1020157032295A patent/KR20150132601A/ko not_active Ceased
- 2004-11-16 AU AU2004290897A patent/AU2004290897B2/en not_active Ceased
- 2004-11-16 KR KR20157002440A patent/KR20150028829A/ko not_active Withdrawn
- 2004-11-16 CN CN2004800405089A patent/CN1905876B/zh not_active Expired - Fee Related
- 2004-11-16 KR KR1020167036999A patent/KR20170005163A/ko not_active Withdrawn
- 2004-11-16 KR KR1020137021480A patent/KR20130105741A/ko not_active Withdrawn
- 2004-11-16 KR KR1020187012266A patent/KR20180050427A/ko not_active Ceased
- 2004-11-16 JP JP2006538825A patent/JP2007511487A/ja not_active Withdrawn
- 2004-11-16 MX MXPA06005518A patent/MXPA06005518A/es active IP Right Grant
- 2004-11-16 EP EP04797932A patent/EP1686994A2/en not_active Withdrawn
- 2004-11-16 KR KR1020127000489A patent/KR20120008093A/ko not_active Withdrawn
- 2004-11-16 EP EP14190100.9A patent/EP2839832A3/en not_active Withdrawn
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2009
- 2009-05-26 AU AU2009202080A patent/AU2009202080A1/en not_active Abandoned
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2012
- 2012-05-30 JP JP2012123284A patent/JP2012211146A/ja not_active Withdrawn
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2014
- 2014-04-01 JP JP2014075331A patent/JP6312502B2/ja not_active Expired - Fee Related
-
2016
- 2016-06-22 JP JP2016123464A patent/JP2016222677A/ja not_active Withdrawn
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2017
- 2017-09-28 JP JP2017188912A patent/JP2018039816A/ja not_active Withdrawn
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2020
- 2020-07-13 JP JP2020119890A patent/JP2020183412A/ja active Pending
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