JP2006509748A5 - - Google Patents

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Publication number
JP2006509748A5
JP2006509748A5 JP2004552660A JP2004552660A JP2006509748A5 JP 2006509748 A5 JP2006509748 A5 JP 2006509748A5 JP 2004552660 A JP2004552660 A JP 2004552660A JP 2004552660 A JP2004552660 A JP 2004552660A JP 2006509748 A5 JP2006509748 A5 JP 2006509748A5
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JP
Japan
Prior art keywords
alkyl
aryl
heteroaryl
heterocyclyl
oxo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2004552660A
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English (en)
Japanese (ja)
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JP2006509748A (ja
Filing date
Publication date
Priority claimed from FR0214443A external-priority patent/FR2847253B1/fr
Application filed filed Critical
Publication of JP2006509748A publication Critical patent/JP2006509748A/ja
Publication of JP2006509748A5 publication Critical patent/JP2006509748A5/ja
Pending legal-status Critical Current

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JP2004552660A 2002-11-19 2003-11-19 Gsk−3ベータ阻害剤としてのピリダジノン誘導体 Pending JP2006509748A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0214443A FR2847253B1 (fr) 2002-11-19 2002-11-19 Nouveaux derives de pyridazinones a titre de medicaments et compositions pharmaceutiques les renfermant
PCT/EP2003/012950 WO2004046117A1 (en) 2002-11-19 2003-11-19 Pyridazinone derivatives as gsk-3beta inhibitors

Publications (2)

Publication Number Publication Date
JP2006509748A JP2006509748A (ja) 2006-03-23
JP2006509748A5 true JP2006509748A5 (enExample) 2006-12-28

Family

ID=32187711

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004552660A Pending JP2006509748A (ja) 2002-11-19 2003-11-19 Gsk−3ベータ阻害剤としてのピリダジノン誘導体

Country Status (19)

Country Link
EP (2) EP1581505B1 (enExample)
JP (1) JP2006509748A (enExample)
KR (1) KR20050083918A (enExample)
CN (1) CN1741999A (enExample)
AR (2) AR042202A1 (enExample)
AT (2) ATE368651T1 (enExample)
AU (2) AU2003296586A1 (enExample)
BR (1) BR0316720A (enExample)
CA (2) CA2506022A1 (enExample)
CO (1) CO5700722A2 (enExample)
DE (2) DE60315354T2 (enExample)
FR (1) FR2847253B1 (enExample)
MA (1) MA27814A1 (enExample)
MX (1) MXPA05005270A (enExample)
NO (1) NO20052887L (enExample)
PL (1) PL376129A1 (enExample)
RU (1) RU2005119151A (enExample)
TW (2) TW200418478A (enExample)
WO (2) WO2004046130A1 (enExample)

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US9212146B2 (en) 2008-03-18 2015-12-15 Shanghai Institute Of Materia Medica, Chinese Academy Of Sciences Substituted pyridazinones for the treatment of tumors
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US8933024B2 (en) 2010-06-18 2015-01-13 Sanofi Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
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TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
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TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
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US8871758B2 (en) 2011-03-08 2014-10-28 Sanofi Tetrasubstituted oxathiazine derivatives, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
EP2683702B1 (de) 2011-03-08 2014-12-24 Sanofi Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
US8895547B2 (en) 2011-03-08 2014-11-25 Sanofi Substituted phenyl-oxathiazine derivatives, method for producing them, drugs containing said compounds and the use thereof
EP2683701B1 (de) 2011-03-08 2014-12-24 Sanofi Mit benzyl- oder heteromethylengruppen substituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2766349B1 (de) 2011-03-08 2016-06-01 Sanofi Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
WO2012120055A1 (de) 2011-03-08 2012-09-13 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
US8828994B2 (en) 2011-03-08 2014-09-09 Sanofi Di- and tri-substituted oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013045413A1 (en) 2011-09-27 2013-04-04 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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WO2019101642A1 (en) * 2017-11-21 2019-05-31 Bayer Aktiengesellschaft Sulphur substituted 3-oxo-2,3-dihydropyridazine-4-carboxamides
CN111533697B (zh) * 2020-05-07 2023-03-31 成都大学 4-氨基哒嗪酮类化合物及其制备方法
CN111533735A (zh) * 2020-05-08 2020-08-14 张建蒙 氧代二氢哒嗪噻唑类衍生物及其在抗肿瘤药物中的应用
CN111393374A (zh) * 2020-05-08 2020-07-10 张建蒙 氧代二氢哒嗪类衍生物及其在抗肿瘤药物中的应用
AR124154A1 (es) 2020-11-27 2023-02-22 Rhizen Pharmaceuticals Ag Inhibidores de cdk
WO2022149057A1 (en) 2021-01-05 2022-07-14 Rhizen Pharmaceuticals Ag Cdk inhibitors
CN117715904A (zh) 2021-05-07 2024-03-15 凯麦拉医疗公司 Cdk2降解剂和其用途

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