NO20052887L - Pyridazinonderivater som GSK-3Beta inhibitorer. - Google Patents

Pyridazinonderivater som GSK-3Beta inhibitorer.

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Publication number
NO20052887L
NO20052887L NO20052887A NO20052887A NO20052887L NO 20052887 L NO20052887 L NO 20052887L NO 20052887 A NO20052887 A NO 20052887A NO 20052887 A NO20052887 A NO 20052887A NO 20052887 L NO20052887 L NO 20052887L
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NO
Norway
Prior art keywords
gsk
pyridazinone derivatives
alkyl
aryl
3beta inhibitors
Prior art date
Application number
NO20052887A
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English (en)
Other versions
NO20052887D0 (no
Inventor
Hans Matter
Karl Schoenafinger
David William Will
Bernard Baudoin
Gilles Tiraboschi
Dominique Le Suisse
Thomas Rooney
Franck Halley
Guenter Mueller
Swen Hoelder
Thorsten Naumann
Original Assignee
Aventis Pharma Gmbh
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Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of NO20052887D0 publication Critical patent/NO20052887D0/no
Publication of NO20052887L publication Critical patent/NO20052887L/no

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    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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Abstract

Foreliggende oppfinnelse angår nye pyridazinonderivater med generell formel (I) hvori A er lik Al eller A2; R er usubstituert eller minst monosubstituert Ci-Cio-alkyI, aryl, aryl(C]-Ci(ralkyl)-, heteroaryl, heteoraryl-(Ci-Cio-alkyl)-, heterosyklyl, heterosyklyl- (Ci-Cio-alkyl)-, Cs-Cio-sykloalkyl, polysykloalkyl, Ci-Cio-alkenyl eller Q-Cio-alkinyl og Ar er usubstituert eller minst monosubstituert aryl eller heteioaryl.
NO20052887A 2002-11-19 2005-06-14 Pyridazinonderivater som GSK-3Beta inhibitorer. NO20052887L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0214443A FR2847253B1 (fr) 2002-11-19 2002-11-19 Nouveaux derives de pyridazinones a titre de medicaments et compositions pharmaceutiques les renfermant
PCT/EP2003/012950 WO2004046117A1 (en) 2002-11-19 2003-11-19 Pyridazinone derivatives as gsk-3beta inhibitors

Publications (2)

Publication Number Publication Date
NO20052887D0 NO20052887D0 (no) 2005-06-14
NO20052887L true NO20052887L (no) 2005-07-29

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NO20052887A NO20052887L (no) 2002-11-19 2005-06-14 Pyridazinonderivater som GSK-3Beta inhibitorer.

Country Status (19)

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EP (2) EP1581505B1 (no)
JP (1) JP2006509748A (no)
KR (1) KR20050083918A (no)
CN (1) CN1741999A (no)
AR (2) AR042202A1 (no)
AT (2) ATE368651T1 (no)
AU (2) AU2003283414A1 (no)
BR (1) BR0316720A (no)
CA (2) CA2506022A1 (no)
CO (1) CO5700722A2 (no)
DE (2) DE60315354T2 (no)
FR (1) FR2847253B1 (no)
MA (1) MA27814A1 (no)
MX (1) MXPA05005270A (no)
NO (1) NO20052887L (no)
PL (1) PL376129A1 (no)
RU (1) RU2005119151A (no)
TW (2) TW200503727A (no)
WO (2) WO2004046130A1 (no)

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