JP2005534715A - カンナビノイドレセプタ配位子 - Google Patents
カンナビノイドレセプタ配位子 Download PDFInfo
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- JP2005534715A JP2005534715A JP2004527741A JP2004527741A JP2005534715A JP 2005534715 A JP2005534715 A JP 2005534715A JP 2004527741 A JP2004527741 A JP 2004527741A JP 2004527741 A JP2004527741 A JP 2004527741A JP 2005534715 A JP2005534715 A JP 2005534715A
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- 0 *Cc(cc1)ccc1Oc(c(Br)c1)ccc1Cl Chemical compound *Cc(cc1)ccc1Oc(c(Br)c1)ccc1Cl 0.000 description 7
- BDJKPIJIQAZEMV-ZDUSSCGKSA-N C[C@@H](c(cc1)ccc1S(c1ccc(C(F)(F)F)cc1S(c(cccc1)c1F)(=O)=O)(=O)=O)N Chemical compound C[C@@H](c(cc1)ccc1S(c1ccc(C(F)(F)F)cc1S(c(cccc1)c1F)(=O)=O)(=O)=O)N BDJKPIJIQAZEMV-ZDUSSCGKSA-N 0.000 description 1
- TZWKENIGHNSLHO-INIZCTEOSA-N C[C@@H](c(cc1)ccc1Sc(ccc(OC)c1)c1Sc(cc1)ccc1OC)NS(C)(=O)=O Chemical compound C[C@@H](c(cc1)ccc1Sc(ccc(OC)c1)c1Sc(cc1)ccc1OC)NS(C)(=O)=O TZWKENIGHNSLHO-INIZCTEOSA-N 0.000 description 1
- OXAWWBKQUDXTSJ-UHFFFAOYSA-N O=C(c(cc1)ccc1Sc(ccc(Cl)c1)c1S(c1ccccc1F)(=O)=O)Oc(c(F)c(c(F)c1F)F)c1F Chemical compound O=C(c(cc1)ccc1Sc(ccc(Cl)c1)c1S(c1ccccc1F)(=O)=O)Oc(c(F)c(c(F)c1F)F)c1F OXAWWBKQUDXTSJ-UHFFFAOYSA-N 0.000 description 1
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/64—Sulfur atoms
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- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
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- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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| JP2009544755A (ja) * | 2006-07-28 | 2009-12-17 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Cb2受容体を変調する化合物 |
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2003
- 2003-08-05 WO PCT/US2003/024398 patent/WO2004014825A1/en not_active Ceased
- 2003-08-05 JP JP2004527741A patent/JP2005534715A/ja active Pending
- 2003-08-05 EP EP03784905A patent/EP1539662A1/en not_active Withdrawn
- 2003-08-05 MX MXPA05001433A patent/MXPA05001433A/es active IP Right Grant
- 2003-08-05 CA CA002494827A patent/CA2494827A1/en not_active Abandoned
- 2003-08-05 AU AU2003257172A patent/AU2003257172A1/en not_active Abandoned
- 2003-08-05 PE PE2003000774A patent/PE20040754A1/es not_active Application Discontinuation
- 2003-08-06 TW TW092121502A patent/TW200413298A/zh unknown
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2009
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| JP2009544755A (ja) * | 2006-07-28 | 2009-12-17 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Cb2受容体を変調する化合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2010024251A (ja) | 2010-02-04 |
| AU2003257172A1 (en) | 2004-02-25 |
| AR040803A1 (es) | 2005-04-20 |
| TW200413298A (en) | 2004-08-01 |
| US20030232859A1 (en) | 2003-12-18 |
| US7067539B2 (en) | 2006-06-27 |
| MXPA05001433A (es) | 2005-06-06 |
| PE20040754A1 (es) | 2004-11-20 |
| CA2494827A1 (en) | 2004-02-19 |
| EP1539662A1 (en) | 2005-06-15 |
| WO2004014825A1 (en) | 2004-02-19 |
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