|
ATE430565T1
(de)
|
2001-02-28 |
2009-05-15 |
Merck & Co Inc |
Acylierte piperidinderivate als melanocortin-4- rezeptoragonisten
|
|
DE60215132T2
(de)
*
|
2001-02-28 |
2007-08-23 |
Merck & Co., Inc. |
Acylierte piperidin-derivate als melanocortin-4-rezeptor-agonisten
|
|
US6911447B2
(en)
|
2001-04-25 |
2005-06-28 |
The Procter & Gamble Company |
Melanocortin receptor ligands
|
|
JP4336196B2
(ja)
|
2001-07-18 |
2009-09-30 |
メルク エンド カムパニー インコーポレーテッド |
メラノコルチン受容体作動薬としての架橋ピペリジン誘導体
|
|
US7115607B2
(en)
|
2001-07-25 |
2006-10-03 |
Amgen Inc. |
Substituted piperazinyl amides and methods of use
|
|
US6977264B2
(en)
|
2001-07-25 |
2005-12-20 |
Amgen Inc. |
Substituted piperidines and methods of use
|
|
US7456184B2
(en)
|
2003-05-01 |
2008-11-25 |
Palatin Technologies Inc. |
Melanocortin receptor-specific compounds
|
|
US7354923B2
(en)
|
2001-08-10 |
2008-04-08 |
Palatin Technologies, Inc. |
Piperazine melanocortin-specific compounds
|
|
NZ534757A
(en)
|
2002-03-12 |
2006-07-28 |
Merck & Co Inc |
Substituted amides
|
|
US7026335B2
(en)
|
2002-04-30 |
2006-04-11 |
The Procter & Gamble Co. |
Melanocortin receptor ligands
|
|
US7105526B2
(en)
|
2002-06-28 |
2006-09-12 |
Banyu Pharmaceuticals Co., Ltd. |
Benzimidazole derivatives
|
|
AU2003268493A1
(en)
|
2002-09-11 |
2004-04-30 |
Merck & Co., Inc. |
Piperazine urea derivatives as melanocortin-4 receptor agonists
|
|
TW200504033A
(en)
|
2002-10-23 |
2005-02-01 |
Procter & Gamble |
Melanocortin receptor ligands
|
|
MY134457A
(en)
*
|
2002-11-22 |
2007-12-31 |
Merck & Co Inc |
Substituted amides
|
|
US7772188B2
(en)
|
2003-01-28 |
2010-08-10 |
Ironwood Pharmaceuticals, Inc. |
Methods and compositions for the treatment of gastrointestinal disorders
|
|
WO2004078717A1
(en)
*
|
2003-03-03 |
2004-09-16 |
Merck & Co., Inc. |
Acylated piperazine derivatives as melanocortin-4 receptor agonists
|
|
US6998488B2
(en)
|
2003-03-10 |
2006-02-14 |
Merck & Co., Inc. |
Process and intermediates for the preparation of 4-aryl piperidines
|
|
CA2519939A1
(en)
|
2003-03-26 |
2004-10-14 |
Merck & Co., Inc. |
Bicyclic piperidine derivatives as melanocortin-4 receptor agonists
|
|
GB0308333D0
(en)
*
|
2003-04-10 |
2003-05-14 |
Glaxo Group Ltd |
Novel compounds
|
|
AR044510A1
(es)
*
|
2003-04-14 |
2005-09-14 |
Merck & Co Inc |
Procedimiento e intermedios para preparar acidos carboxilicos de pirrolidina
|
|
US7049323B2
(en)
|
2003-04-25 |
2006-05-23 |
Bristol-Myers Squibb Company |
Amidoheterocycles as modulators of the melanocortin-4 receptor
|
|
EP1648457A2
(en)
|
2003-07-22 |
2006-04-26 |
Merck & Co., Inc. |
Piperidine derivatives as melanocortin-4 receptor agonists
|
|
AU2004274309B2
(en)
|
2003-09-22 |
2010-04-08 |
Msd K.K. |
Novel piperidine derivative
|
|
US20050192286A1
(en)
*
|
2003-10-22 |
2005-09-01 |
Neurocrine Biosciences, Inc. |
Ligands of melanocortin receptors and compositions and methods related thereto
|
|
US7989634B2
(en)
|
2003-11-12 |
2011-08-02 |
Lg Life Sciences Ltd. |
Melanocortin receptor agonists
|
|
GB0402492D0
(en)
*
|
2004-02-04 |
2004-03-10 |
Pfizer Ltd |
Pharmaceutically active compounds
|
|
US7649002B2
(en)
|
2004-02-04 |
2010-01-19 |
Pfizer Inc |
(3,5-dimethylpiperidin-1yl)(4-phenylpyrrolidin-3-yl)methanone derivatives as MCR4 agonists
|
|
AU2005230864A1
(en)
|
2004-03-29 |
2005-10-20 |
Merck Sharp & Dohme Corp. |
Diaryltriazoles as inhibitors of 11-beta-hydroxysteroid dehydrogenase-1
|
|
US20080125403A1
(en)
|
2004-04-02 |
2008-05-29 |
Merck & Co., Inc. |
Method of Treating Men with Metabolic and Anthropometric Disorders
|
|
JP2008506696A
(ja)
*
|
2004-07-16 |
2008-03-06 |
メルク エンド カムパニー インコーポレーテッド |
メラノコルチン−４受容体作用薬としてのアシル化ピペリジン誘導体
|
|
EP1773338B1
(en)
|
2004-07-19 |
2010-01-06 |
Merck & Co., Inc. |
Acylated piperidine derivatives as melanocortin-4 receptor agonists
|
|
CN1993320A
(zh)
|
2004-08-06 |
2007-07-04 |
默克公司 |
作为11－β－羟基类固醇脱氢酶－1的抑制剂的磺酰化合物
|
|
WO2006028631A2
(en)
*
|
2004-08-13 |
2006-03-16 |
Merck & Co., Inc. |
Inhibition of voluntary ethanol consumption with non-peptidyl melanocortin 4-receptor agonists
|
|
EP1804798A4
(en)
*
|
2004-10-05 |
2008-01-23 |
Merck & Co Inc |
METHOD FOR THE TREATMENT OF SUBSTANCE ABUSE AND SEARCH
|
|
TW200630337A
(en)
|
2004-10-14 |
2006-09-01 |
Euro Celtique Sa |
Piperidinyl compounds and the use thereof
|
|
US20080200376A1
(en)
*
|
2004-10-29 |
2008-08-21 |
Maccoss Malcolm |
Compositions and Methods For the Treatment Of Obesity and Sexual Dysfunction
|
|
EP2286840A3
(en)
|
2004-11-01 |
2013-09-04 |
Amylin Pharmaceuticals, LLC |
Treatment of obesity and related diseases
|
|
WO2006057904A1
(en)
*
|
2004-11-23 |
2006-06-01 |
Merck & Co., Inc. |
Stereoselective preparation of 4-aryl piperidine amides by asymmetric hydrogenation of a prochiral enamide and intermediates of this process
|
|
GB0428514D0
(en)
*
|
2004-12-31 |
2005-02-09 |
Prosidion Ltd |
Compounds
|
|
CA2609388C
(en)
|
2005-05-30 |
2013-08-06 |
Banyu Pharmaceutical Co., Ltd. |
Novel piperidine derivative
|
|
US8129413B2
(en)
|
2005-06-27 |
2012-03-06 |
Merck Sharp & Dohme Corp. |
Crystalline forms of MC4R agonist and process for synthesis
|
|
AU2006275702A1
(en)
|
2005-07-29 |
2007-02-08 |
Concert Pharmaceuticals Inc. |
Novel pharmaceutical compounds
|
|
WO2007015162A1
(en)
*
|
2005-08-04 |
2007-02-08 |
Pfizer Limited |
Piperidinoyl-pyrrolidine and piperidinoyl-piperidine compounds
|
|
JPWO2007018248A1
(ja)
|
2005-08-10 |
2009-02-19 |
萬有製薬株式会社 |
ピリドン化合物
|
|
BRPI0614649A2
(pt)
|
2005-08-11 |
2011-04-12 |
Amylin Pharmaceuticals Inc |
polipeptìdeos hìbridos com propriedades selecionáveis
|
|
EP2330124B1
(en)
|
2005-08-11 |
2015-02-25 |
Amylin Pharmaceuticals, LLC |
Hybrid polypeptides with selectable properties
|
|
EP1921065B1
(en)
|
2005-08-24 |
2010-10-20 |
Banyu Pharmaceutical Co., Ltd. |
Phenylpyridone derivative
|
|
WO2007029847A1
(ja)
|
2005-09-07 |
2007-03-15 |
Banyu Pharmaceutical Co., Ltd. |
二環性芳香族置換ピリドン誘導体
|
|
BRPI0616463A2
(pt)
|
2005-09-29 |
2011-06-21 |
Merck & Co Inc |
composto, composição farmacêutica, e, uso de um composto
|
|
AU2006297452A1
(en)
*
|
2005-09-30 |
2007-04-12 |
Merck Sharp & Dohme Corp. |
Acylated piperidine derivatives as melanocortin-4 receptor agonists
|
|
EP1940401B1
(en)
|
2005-10-18 |
2012-07-11 |
Merck Sharp & Dohme Corp. |
Acylated spiropiperidine derivatives as melanocortin-4 receptor modulators
|
|
WO2007048027A2
(en)
|
2005-10-21 |
2007-04-26 |
Novartis Ag |
Combination of a renin-inhibitor and an anti-dyslipidemic agent and/or an antiobesity agent
|
|
AU2006307046A1
(en)
|
2005-10-27 |
2007-05-03 |
Msd K.K. |
Novel benzoxathiin derivative
|
|
US8158791B2
(en)
|
2005-11-10 |
2012-04-17 |
Msd K.K. |
Aza-substituted spiro derivatives
|
|
EP1801098A1
(en)
|
2005-12-16 |
2007-06-27 |
Merck Sante |
2-Adamantylurea derivatives as selective 11B-HSD1 inhibitors
|
|
CN101426782B
(zh)
*
|
2006-02-23 |
2012-10-31 |
辉瑞股份有限公司 |
黑皮质素4型受体激动剂哌啶羰基吡咯烷
|
|
ES2402581T3
(es)
|
2006-02-23 |
2013-05-06 |
Pfizer Limited |
Piperidinoilpirrolidinas como agonistas del receptor de melanocortina tipo 4
|
|
WO2007110449A1
(en)
|
2006-03-29 |
2007-10-04 |
Euro-Celtique S.A. |
Benzenesulfonamide compounds and their use
|
|
US8937181B2
(en)
|
2006-04-13 |
2015-01-20 |
Purdue Pharma L.P. |
Benzenesulfonamide compounds and the use thereof
|
|
TW200815353A
(en)
|
2006-04-13 |
2008-04-01 |
Euro Celtique Sa |
Benzenesulfonamide compounds and their use
|
|
US20080027072A1
(en)
*
|
2006-04-20 |
2008-01-31 |
Ampla Pharmaceuticals, Inc. |
Potentiation of MC4 receptor activity
|
|
TWI332501B
(en)
*
|
2006-07-14 |
2010-11-01 |
Lg Life Sciences Ltd |
Melanocortin receptor agonists
|
|
WO2008026563A1
(en)
*
|
2006-08-30 |
2008-03-06 |
Shionogi & Co., Ltd. |
Hydrazine amide derivative
|
|
JP5489333B2
(ja)
|
2006-09-22 |
2014-05-14 |
メルク・シャープ・アンド・ドーム・コーポレーション |
脂肪酸合成阻害剤を用いた治療の方法
|
|
AU2007301126A1
(en)
|
2006-09-28 |
2008-04-03 |
Banyu Pharmaceutical Co., Ltd. |
Diaryl ketimine derivative
|
|
EP2121659B1
(en)
*
|
2006-12-18 |
2013-05-15 |
7TM Pharma A/S |
Modulators of cb1 receptors
|
|
EP1935420A1
(en)
|
2006-12-21 |
2008-06-25 |
Merck Sante |
2-Adamantyl-butyramide derivatives as selective 11beta-HSD1 inhibitors
|
|
CA2682727C
(en)
|
2007-04-02 |
2016-03-22 |
Banyu Pharmaceutical Co., Ltd. |
Indoledione derivative
|
|
US8399486B2
(en)
*
|
2007-04-09 |
2013-03-19 |
Purdue Pharma L.P. |
Benzenesulfonyl compounds and the use thereof
|
|
US8969514B2
(en)
|
2007-06-04 |
2015-03-03 |
Synergy Pharmaceuticals, Inc. |
Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
|
|
EP2527360B1
(en)
|
2007-06-04 |
2015-10-28 |
Synergy Pharmaceuticals Inc. |
Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
|
|
US8765736B2
(en)
|
2007-09-28 |
2014-07-01 |
Purdue Pharma L.P. |
Benzenesulfonamide compounds and the use thereof
|
|
US20110015181A1
(en)
|
2008-03-06 |
2011-01-20 |
Makoto Ando |
Alkylaminopyridine derivative
|
|
EP2272841A1
(en)
|
2008-03-28 |
2011-01-12 |
Banyu Pharmaceutical Co., Ltd. |
Diarylmethylamide derivative having antagonistic activity on melanin-concentrating hormone receptor
|
|
EP2110374A1
(en)
|
2008-04-18 |
2009-10-21 |
Merck Sante |
Benzofurane, benzothiophene, benzothiazol derivatives as FXR modulators
|
|
AU2009261248A1
(en)
|
2008-06-19 |
2009-12-23 |
Banyu Pharmaceutical Co., Ltd. |
Spirodiamine-diarylketoxime derivative
|
|
EP3241839B1
(en)
|
2008-07-16 |
2019-09-04 |
Bausch Health Ireland Limited |
Agonists of guanylate cyclase useful for the treatment of gastrointestinal, inflammation, cancer and other disorders
|
|
WO2010013595A1
(ja)
|
2008-07-30 |
2010-02-04 |
萬有製薬株式会社 |
５員－５員又は５員－６員縮環シクロアルキルアミン誘導体
|
|
JP5530438B2
(ja)
|
2008-08-06 |
2014-06-25 |
ファイザー・リミテッド |
Ｍｃ４作動薬としてのジアゼピンおよびジアゾカン化合物
|
|
WO2010047982A1
(en)
|
2008-10-22 |
2010-04-29 |
Merck Sharp & Dohme Corp. |
Novel cyclic benzimidazole derivatives useful anti-diabetic agents
|
|
JP5557845B2
(ja)
|
2008-10-31 |
2014-07-23 |
メルク・シャープ・アンド・ドーム・コーポレーション |
糖尿病用剤として有用な新規環状ベンゾイミダゾール誘導体
|
|
UA99555C2
(en)
|
2008-11-12 |
2012-08-27 |
Элджи Лайф Саенсез Лтд. |
Melanocortin receptor agonists
|
|
JP5514831B2
(ja)
|
2008-11-17 |
2014-06-04 |
メルク・シャープ・アンド・ドーム・コーポレーション |
糖尿病の治療のための置換二環式アミン
|
|
WO2010067233A1
(en)
|
2008-12-08 |
2010-06-17 |
Pfizer Inc. |
1,2,4 triazolo [4, 3 -a] [1,5] benzodiazepin-5 (6h) -ones as agonists of the cholecystokinin-1 receptor (cck-ir)
|
|
CN102245570A
(zh)
*
|
2008-12-16 |
2011-11-16 |
弗·哈夫曼-拉罗切有限公司 |
制备吡咯烷-3-甲酸类的方法
|
|
WO2010084428A1
(en)
|
2009-01-20 |
2010-07-29 |
Pfizer Inc. |
Substituted pyrazinone amides
|
|
WO2010086820A1
(en)
|
2009-02-02 |
2010-08-05 |
Pfizer Inc. |
4-amino-5-oxo-7, 8-dihydropyrimido [5,4-f] [1,4] oxazepin-6 (5h) -yl) phenyl derivatives, pharmaceutical compositions and uses thereof
|
|
WO2010089685A1
(en)
|
2009-02-03 |
2010-08-12 |
Pfizer Inc. |
4-amino-7,8-dihydropyrido[4,3-d]pyrimidin-5(6h)-one derivatives
|
|
JP2012516885A
(ja)
|
2009-02-04 |
2012-07-26 |
ファイザー・インク |
４−アミノ−７，８−ジヒドロピリド［４，３−ｄ］ピリミジン−５（６Ｈ）−オン誘導体
|
|
JP5642661B2
(ja)
*
|
2009-03-05 |
2014-12-17 |
塩野義製薬株式会社 |
Ｎｐｙｙ５受容体拮抗作用を有するピペリジンおよびピロリジン誘導体
|
|
US20110319379A1
(en)
|
2009-03-11 |
2011-12-29 |
Corbett Jeffrey W |
Substituted Indazole Amides And Their Use As Glucokinase Activators
|
|
MY151246A
(en)
|
2009-03-11 |
2014-04-30 |
Pfizer |
Benzofuranyl derivatives
|
|
WO2010106457A2
(en)
|
2009-03-20 |
2010-09-23 |
Pfizer Inc. |
3-oxa-7-azabicyclo[3.3.1]nonanes
|
|
NZ596467A
(en)
|
2009-06-05 |
2014-01-31 |
Pfizer |
L- ( piperidin-4-yl) -pyrazole derivatives as gpr 119 modulators
|
|
WO2011011506A1
(en)
|
2009-07-23 |
2011-01-27 |
Schering Corporation |
Spirocyclic oxazepine compounds as stearoyl-coenzyme a delta-9 desaturase inhibitors
|
|
CA2768577A1
(en)
|
2009-07-23 |
2011-01-27 |
Schering Corporation |
Benzo-fused oxazepine compounds as stearoyl-coenzyme a delta-9 desaturase inhibitors
|
|
US20130072427A1
(en)
|
2009-09-23 |
2013-03-21 |
Pfizer Inc. |
Gpr 119 modulators
|
|
EA021983B1
(ru)
|
2009-11-02 |
2015-10-30 |
Пфайзер Инк. |
Производные диоксабицикло[3.2.1]октан-2,3,4-триола
|
|
WO2011058474A1
(en)
|
2009-11-10 |
2011-05-19 |
Pfizer Inc. |
N1-pyrazolospiroketone acetyl-coa carboxylase inhibitors
|
|
EP2499140A1
(en)
|
2009-11-10 |
2012-09-19 |
Pfizer Inc. |
N2-pyrazolospiroketone acetyl-coa carboxylase inhibitors
|
|
AU2010317842A1
(en)
|
2009-11-16 |
2012-07-12 |
Mellitech |
[1,5]-diazocin derivatives
|
|
EP2504342A1
(en)
|
2009-11-23 |
2012-10-03 |
Pfizer Inc. |
Imidazo-pyrazoles as gpr119 inhibitors
|
|
CN103664873B
(zh)
|
2009-12-30 |
2016-06-15 |
深圳信立泰药业股份有限公司 |
作为二肽基肽酶iv(dpp-iv)抑制剂的3-(3-氨基哌啶-1-基)-5-氧代-1,2,4-三嗪衍生物
|
|
US9044606B2
(en)
|
2010-01-22 |
2015-06-02 |
Ethicon Endo-Surgery, Inc. |
Methods and devices for activating brown adipose tissue using electrical energy
|
|
US8476227B2
(en)
|
2010-01-22 |
2013-07-02 |
Ethicon Endo-Surgery, Inc. |
Methods of activating a melanocortin-4 receptor pathway in obese subjects
|
|
US8895596B2
(en)
|
2010-02-25 |
2014-11-25 |
Merck Sharp & Dohme Corp |
Cyclic benzimidazole derivatives useful as anti-diabetic agents
|
|
CA2792234C
(en)
|
2010-03-19 |
2014-05-27 |
Pfizer Inc. |
2,3 dihydro-1h-inden-1-yl-2,7-diazaspiro [3.5] nonane derivatives and their use as antagonists or inverse agonists of the ghrelin receptor
|
|
EP2563764B1
(en)
|
2010-04-26 |
2015-02-25 |
Merck Sharp & Dohme Corp. |
Novel spiropiperidine prolylcarboxypeptidase inhibitors
|
|
US9365539B2
(en)
|
2010-05-11 |
2016-06-14 |
Merck Sharp & Dohme Corp. |
Prolylcarboxypeptidase inhibitors
|
|
US9006268B2
(en)
|
2010-06-11 |
2015-04-14 |
Merck Sharp & Dohme Corp. |
Prolylcarboxypeptidase inhibitors
|
|
WO2011158149A1
(en)
|
2010-06-18 |
2011-12-22 |
Pfizer Inc. |
2-(3,5-disubstitutedphenyl)pyrimidin-4(3h)-one derivatives
|
|
US9616097B2
(en)
|
2010-09-15 |
2017-04-11 |
Synergy Pharmaceuticals, Inc. |
Formulations of guanylate cyclase C agonists and methods of use
|
|
HRP20161178T1
(hr)
|
2010-09-30 |
2016-11-04 |
Pfizer Inc. |
N1-PIRAZOLOSPIROKETONSKI INHIBITORI ACETIL-CoA-KARBOKSILAZE
|
|
BR112013010310A2
(pt)
|
2010-10-29 |
2016-11-29 |
Pfizer |
inibidores de acetil-coa carboxilase de lactama n1/n2
|
|
MX2013006768A
(es)
|
2010-12-23 |
2013-07-22 |
Pfizer |
Moduladores de receptor de glucagon.
|
|
HRP20161177T1
(hr)
|
2011-02-08 |
2016-11-04 |
Pfizer Inc. |
Modulator glukagonskog receptora
|
|
BR112013021236B1
(pt)
|
2011-02-25 |
2021-05-25 |
Merck Sharp & Dohme Corp |
composto derivado de benzimidazol, e, composição
|
|
MY162167A
(en)
|
2011-04-22 |
2017-05-31 |
Pfizer |
Substituted acetyl-coa carboxylase inhibitors
|
|
CA2841757A1
(en)
|
2011-07-15 |
2013-01-24 |
Etzer Darout |
Gpr 119 modulators
|
|
AU2012288493B2
(en)
|
2011-07-22 |
2015-08-06 |
Pfizer Inc. |
Quinolinyl glucagon receptor modulators
|
|
JP2015515472A
(ja)
|
2012-04-06 |
2015-05-28 |
ファイザー・インク |
ジアシルグリセロールアシルトランスフェラーゼ２阻害薬
|
|
US8889730B2
(en)
|
2012-04-10 |
2014-11-18 |
Pfizer Inc. |
Indole and indazole compounds that activate AMPK
|
|
ES2585262T3
(es)
|
2012-05-04 |
2016-10-04 |
Pfizer Inc |
Compuestos heterocíclicos de hexahidropiran[3,4-d][1,3]tiazin-2-amina sustituidos como inhibidores de PPA, BACE1 y BACE2
|
|
US9527875B2
(en)
|
2012-08-02 |
2016-12-27 |
Merck Sharp & Dohme Corp. |
Antidiabetic tricyclic compounds
|
|
CA2882389A1
(en)
|
2012-09-20 |
2014-03-27 |
Pfizer Inc. |
Alkyl-substituted hexahydropyrano[3,4-d][1,3]thiazin-2-amine compounds
|
|
WO2014091352A1
(en)
|
2012-12-11 |
2014-06-19 |
Pfizer Inc. |
Hexahydropyrano [3,4-d][1,3]thiazin-2-amine compounds as inhibitors of bace1
|
|
CA2893333C
(en)
|
2012-12-19 |
2017-10-24 |
Pfizer Inc. |
Carbocyclic-and heterocyclic-substituted hexahydropyrano[3,4-d][1,3]thiazin-2-amine compounds
|
|
WO2014125394A1
(en)
|
2013-02-13 |
2014-08-21 |
Pfizer Inc. |
HETEROARYL-SUBSTITUTED HEXAHYDROPYRANO [3,4-d][1,3] THIAZIN-2-AMINE COMPOUNDS
|
|
US9233981B1
(en)
|
2013-02-15 |
2016-01-12 |
Pfizer Inc. |
Substituted phenyl hexahydropyrano[3,4-d][1,3]thiazin-2-amine compounds
|
|
RU2015140066A
(ru)
|
2013-02-22 |
2017-03-30 |
Мерк Шарп И Доум Корп. |
Противодиабетические бициклические соединения
|
|
WO2014139388A1
(en)
|
2013-03-14 |
2014-09-18 |
Merck Sharp & Dohme Corp. |
Novel indole derivatives useful as anti-diabetic agents
|
|
CA2905435A1
(en)
|
2013-03-15 |
2014-09-25 |
Synergy Pharmaceuticals Inc. |
Compositions useful for the treatment of gastrointestinal disorders
|
|
CA2905438A1
(en)
|
2013-03-15 |
2014-09-25 |
Synergy Pharmaceuticals Inc. |
Agonists of guanylate cyclase and their uses
|
|
SI3004138T1
(sl)
|
2013-06-05 |
2024-07-31 |
Bausch Health Ireland Limited |
Ultra čisti agonisti gvanilat ciklaze C, postopek za njihovo pripravo in uporabo
|
|
WO2015051496A1
(en)
|
2013-10-08 |
2015-04-16 |
Merck Sharp & Dohme Corp. |
Antidiabetic tricyclic compounds
|
|
ES2665153T3
(es)
|
2013-10-09 |
2018-04-24 |
Pfizer Inc. |
Antagonistas del receptor EP3 de prostaglandina
|
|
LT3119757T
(lt)
|
2014-03-17 |
2018-07-10 |
Pfizer Inc. |
Diacilglicerolio aciltransferazės 2 inhibitoriai, skirti panaudoti metabolinių ir susijusių ligų gydyme
|
|
PE20170327A1
(es)
|
2014-04-10 |
2017-04-21 |
Pfizer |
2-AMINO-6-METIL-4,4a,5,6-TETRAHIDROPIRANO[3,4d] [1,3] TIAZIN-8a(8H)-IL-1,3-TIAZOL-4-ILAMIDAS
|
|
SG11201609864UA
(en)
*
|
2014-05-29 |
2016-12-29 |
Mitsubishi Tanabe Pharma Corp |
Novel pyrrolidine compound and application as melanocortin receptor agonist
|
|
KR102431436B1
(ko)
|
2014-08-29 |
2022-08-10 |
테스 파마 에스.알.엘. |
α-아미노-β-카복시뮤콘산 세미알데히드 데카복실라제의 억제제
|
|
WO2016092413A1
(en)
|
2014-12-10 |
2016-06-16 |
Pfizer Inc. |
Indole and indazole compounds that activate ampk
|
|
WO2016103097A1
(en)
|
2014-12-22 |
2016-06-30 |
Pfizer Inc. |
Antagonists of prostaglandin ep3 receptor
|
|
US10092738B2
(en)
|
2014-12-29 |
2018-10-09 |
Ethicon Llc |
Methods and devices for inhibiting nerves when activating brown adipose tissue
|
|
US10080884B2
(en)
|
2014-12-29 |
2018-09-25 |
Ethicon Llc |
Methods and devices for activating brown adipose tissue using electrical energy
|
|
EP3766885B1
(en)
|
2015-06-17 |
2022-05-25 |
Pfizer Inc. |
Tricyclic compounds and their use as phosphodiesterase inhibitors
|
|
WO2017051294A1
(en)
|
2015-09-24 |
2017-03-30 |
Pfizer Inc. |
N-[2-(3-amino-2,5-dimethyl-1,1-dioxido-5,6-dihydro-2h-1,2,4-thiadiazin-5-yl)-1,3-thiazol-4-yl] amides useful as bace inhibitors
|
|
EP3353182A1
(en)
|
2015-09-24 |
2018-08-01 |
Pfizer Inc |
Tetrahydropyrano[3,4-d][1,3]oxazin derivatives and their use as bace inhibitors
|
|
WO2017051276A1
(en)
|
2015-09-24 |
2017-03-30 |
Pfizer Inc. |
N-[2-(2-amino-6,6-disubstituted-4, 4a, 5, 6-tetrahydropyrano [3,4-d][1,3] thiazin-8a (8h)-yl) -1, 3-thiazol-4-yl] amides
|
|
SI3397631T1
(sl)
|
2015-12-29 |
2022-01-31 |
Pfizer Inc. |
Substituirani 3-azabiciklo(3.1.0)heksani kot zaviralci ketoheksokinaze
|
|
AR109179A1
(es)
|
2016-08-19 |
2018-11-07 |
Pfizer |
Inhibidores de diacilglicerol aciltransferasa 2
|
|
AR109950A1
(es)
|
2016-10-14 |
2019-02-06 |
Tes Pharma S R L |
INHIBIDORES DE LA ÁCIDO a-AMINO-b-CARBOXIMUCÓNICO SEMIALDEHÍDO DESCARBOXILASA
|
|
US11072602B2
(en)
|
2016-12-06 |
2021-07-27 |
Merck Sharp & Dohme Corp. |
Antidiabetic heterocyclic compounds
|
|
WO2018118670A1
(en)
|
2016-12-20 |
2018-06-28 |
Merck Sharp & Dohme Corp. |
Antidiabetic spirochroman compounds
|
|
CR20210110A
(es)
|
2018-08-31 |
2021-05-13 |
Pfizer |
Combinaciones para tratamiento de ehna/ehgna y enfermedades relacionadas
|
|
AR117122A1
(es)
|
2018-11-20 |
2021-07-14 |
Tes Pharma S R L |
INHIBIDORES DE LA ÁCIDO a-AMINO-b-CARBOXIMUCÓNICO SEMIALDEHÍDO DESCARBOXILASA
|
|
WO2020234726A1
(en)
|
2019-05-20 |
2020-11-26 |
Pfizer Inc. |
Combinations comprising benzodioxol as glp-1r agonists for use in the treatment of nash/nafld and related diseases
|
|
EP3953327B1
(en)
*
|
2019-11-07 |
2023-12-27 |
Lg Chem, Ltd. |
Melanocortin-4 receptor agonists
|
|
WO2022139441A1
(ko)
*
|
2020-12-22 |
2022-06-30 |
주식회사 엘지화학 |
무정형의 멜라노코르틴 수용체 작용제 및 이의 제조방법
|
|
US20250066337A1
(en)
|
2021-08-26 |
2025-02-27 |
Pfizer Inc. |
Amorphous Form of (S)-2-(5-((3-Ethoxypyridin-2-YL)Oxy)Pyridin-3-YL)-N-(Tetrahydrofuran-3-YL)Pyrimidine-5-Carboxamide
|
|
WO2024118524A1
(en)
|
2022-11-28 |
2024-06-06 |
Cerevel Therapeutics, Llc |
Azaindole compounds and their use as phosphodiesterase inhibitors
|