JP2005531526A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2005531526A5 JP2005531526A5 JP2003580307A JP2003580307A JP2005531526A5 JP 2005531526 A5 JP2005531526 A5 JP 2005531526A5 JP 2003580307 A JP2003580307 A JP 2003580307A JP 2003580307 A JP2003580307 A JP 2003580307A JP 2005531526 A5 JP2005531526 A5 JP 2005531526A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- formula
- compound
- alkyl
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 0 CCCCC1=SC(N(*)N=C)=C(*)*1 Chemical compound CCCCC1=SC(N(*)N=C)=C(*)*1 0.000 description 2
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02290788A EP1348701A1 (en) | 2002-03-28 | 2002-03-28 | (2,4-disubstituted-thiazol-5-yl) amine compounds as PDE7 inhibitors |
| PCT/EP2003/002287 WO2003082839A1 (en) | 2002-03-28 | 2003-03-06 | (4,2-disubstituted-thiazol-5-yl)amine compounds as pde7 inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005531526A JP2005531526A (ja) | 2005-10-20 |
| JP2005531526A5 true JP2005531526A5 (https=) | 2006-04-20 |
Family
ID=27798934
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003580307A Withdrawn JP2005531526A (ja) | 2002-03-28 | 2003-03-06 | Ｐｄｅ７阻害剤としての（４，２−２置換−チアゾール−５−イル）アミン化合物 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US6753340B2 (https=) |
| EP (2) | EP1348701A1 (https=) |
| JP (1) | JP2005531526A (https=) |
| AU (1) | AU2003212310A1 (https=) |
| BR (1) | BR0308765A (https=) |
| CA (1) | CA2480679A1 (https=) |
| MX (1) | MXPA04009476A (https=) |
| WO (1) | WO2003082839A1 (https=) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2004044235A1 (en) * | 2002-11-13 | 2004-05-27 | Bayer Healthcare Ag | DIAGNOSTICS AND THERAPEUTICS FOR DISEASES ASSOCIATED WITH HUMAN PHOSPHODIESTERASE 7A1 (PDE7a1) |
| ES2217956B1 (es) * | 2003-01-23 | 2006-04-01 | Almirall Prodesfarma, S.A. | Nuevos derivados de 4-aminotieno(2,3-d)pirimidin-6-carbonitrilo. |
| KR100783255B1 (ko) | 2004-02-13 | 2007-12-06 | 워너-램버트 캄파니 엘엘씨 | 안드로젠 수용체 조절제 |
| JP2007532621A (ja) | 2004-04-13 | 2007-11-15 | ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー | アンドロゲンモジュレータ |
| WO2005102990A1 (en) | 2004-04-22 | 2005-11-03 | Warner-Lambert Company Llc | Androgen modulators |
| TW200724139A (en) | 2005-05-05 | 2007-07-01 | Warner Lambert Co | Androgen modulators |
| WO2007056457A2 (en) | 2005-11-09 | 2007-05-18 | Combinatorx, Incorporated | Methods, compositions, and kits for the treatment of medical conditions |
| GB0701426D0 (en) * | 2007-01-25 | 2007-03-07 | Univ Sheffield | Compounds and their use |
| US8637528B2 (en) | 2007-03-27 | 2014-01-28 | Omeros Corporation | Use of PDE7 inhibitors for the treatment of movement disorders |
| WO2008119057A2 (en) * | 2007-03-27 | 2008-10-02 | Omeros Corporation | The use of pde7 inhibitors for the treatment of movement disorders |
| FR2943673B1 (fr) | 2009-03-27 | 2013-03-29 | Sanofi Aventis | Applications therapeutiques de derives de quinazolinedione |
| NZ628054A (en) | 2010-11-08 | 2016-03-31 | Omeros Corp | Treatment of addiction and impulse-control disorders using pde7 inhibitors |
| US9220715B2 (en) | 2010-11-08 | 2015-12-29 | Omeros Corporation | Treatment of addiction and impulse-control disorders using PDE7 inhibitors |
| US20130184280A1 (en) * | 2011-12-21 | 2013-07-18 | Telik, Inc. | Substituted thiazoles as vegfr2 kinase inhibitors |
| KR102494647B1 (ko) | 2016-07-14 | 2023-01-31 | 브리스톨-마이어스 스큅 컴퍼니 | 비시클릭 헤테로아릴 치환된 화합물 |
| CN109689664B (zh) | 2016-07-14 | 2022-04-15 | 百时美施贵宝公司 | 作为par4抑制剂的三环杂芳基取代的喹啉和氮杂喹啉化合物 |
| US20190292176A1 (en) | 2016-07-14 | 2019-09-26 | Bistol-Myers Squibb Company | Bicyclic heteroaryl substituted compounds |
| US11987981B2 (en) | 2016-07-28 | 2024-05-21 | Carboshield, Inc. | Structural element reinforcement systems and methods |
| US12195987B2 (en) | 2016-07-28 | 2025-01-14 | Carboshield, Inc. | Structural element reinforcement systems and methods |
| IL318817A (en) | 2022-08-18 | 2025-04-01 | Mitodicure Gmbh | Use of a therapeutic agent with PHOSPHODIESTERASE-7 inhibitory activity for the treatment and prevention of diseases associated with chronic fatigue, exhaustion and/or exercise intolerance |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0772606A1 (en) * | 1994-07-27 | 1997-05-14 | G.D. SEARLE & CO. | Substituted thiazoles for the treatment of inflammation |
| WO1998008844A1 (de) * | 1996-08-26 | 1998-03-05 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Thiazol-derivate als selektive inhibitoren der pde-iv |
| US6313156B1 (en) * | 1999-12-23 | 2001-11-06 | Icos Corporation | Thiazole compounds as cyclic-AMP-specific phosphodiesterase inhibitors |
| AU2001237401B2 (en) * | 2000-03-01 | 2006-11-09 | Janssen Pharmaceutica N.V. | 2,4-disubstituted thiazolyl derivatives |
-
2002
- 2002-03-28 EP EP02290788A patent/EP1348701A1/en not_active Withdrawn
-
2003
- 2003-03-06 JP JP2003580307A patent/JP2005531526A/ja not_active Withdrawn
- 2003-03-06 EP EP03708184A patent/EP1492778A1/en not_active Withdrawn
- 2003-03-06 WO PCT/EP2003/002287 patent/WO2003082839A1/en not_active Ceased
- 2003-03-06 AU AU2003212310A patent/AU2003212310A1/en not_active Abandoned
- 2003-03-06 BR BR0308765-4A patent/BR0308765A/pt not_active IP Right Cessation
- 2003-03-06 CA CA002480679A patent/CA2480679A1/en not_active Abandoned
- 2003-03-06 MX MXPA04009476A patent/MXPA04009476A/es active IP Right Grant
- 2003-03-27 US US10/401,392 patent/US6753340B2/en not_active Expired - Fee Related
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2005531526A5 (https=) | ||
| EP3209656B1 (en) | Indole carboxamides compounds useful as kinase inhibitors | |
| JP4881433B2 (ja) | 治療薬の薬物動態の調整 | |
| JP2006514626A5 (https=) | ||
| JP7044392B2 (ja) | マラリアの治療のための化合物及び方法 | |
| JP2009542696A5 (https=) | ||
| CA2521158A1 (fr) | Derives de 2-acylamino-4-phenylthiazole, leur preparation et leur application en therapeutique | |
| TW201002703A (en) | Quinazolinedione derivatives as TRPA1 modulators | |
| US20210179577A1 (en) | Aromatic sulfonamide derivatives for the treatment of ischemic stroke | |
| JP2000505451A (ja) | キノロン類およびこれらの治療的使用 | |
| RU2002133220A (ru) | Замещенные 1-аминоалкиллактамы и их применение в качестве антагонистов мускариновых рецепторов | |
| JP2000505450A (ja) | キノロン類およびこれらの治療的使用 | |
| JP2005531526A (ja) | Ｐｄｅ７阻害剤としての（４，２−２置換−チアゾール−５−イル）アミン化合物 | |
| JP2006507355A5 (https=) | ||
| HUP9903797A2 (hu) | Benzofurán-karboxamidok és -szulfonamidok, alkalmazásuk gyógyszerkészítmények előállítására és ezek a gyógyszerkészítmények | |
| JP2004525183A5 (https=) | ||
| JP2005528367A5 (https=) | ||
| JP2006503857A5 (https=) | ||
| JP4306804B2 (ja) | タキキニンアンタゴニスト | |
| JPH09509957A (ja) | 免疫調節剤としてのキノリン誘導体 | |
| FR3050732B1 (fr) | Nouveaux derives de phosphinolactones et leurs utilisations pharmaceutiques | |
| JP2006500372A5 (https=) | ||
| MX2014012634A (es) | Compuesto heterociclico aromatico biciclico nitrogenado. | |
| CN103827100B (zh) | 用于降低血清尿酸的[1,2,4]噻二嗪1,1-二氧化物化合物 | |
| JP2005535648A (ja) | キナゾリン誘導体 |