JP2000500479A - ピラゾール誘導体、その製造方法、および該誘導体を含む医薬組成物 - Google Patents

ピラゾール誘導体、その製造方法、および該誘導体を含む医薬組成物

Info

Publication number
JP2000500479A
JP2000500479A JP9519454A JP51945497A JP2000500479A JP 2000500479 A JP2000500479 A JP 2000500479A JP 9519454 A JP9519454 A JP 9519454A JP 51945497 A JP51945497 A JP 51945497A JP 2000500479 A JP2000500479 A JP 2000500479A
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JP
Japan
Prior art keywords
formula
compound
alkyl
alkoxy
resulting
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP9519454A
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English (en)
Japanese (ja)
Other versions
JP2000500479A5 (enExample
Inventor
バルト，フランシス
コンジー，クリスティアン
マルティネ，セルジュ
リナルディ，ミュリエル
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi SA
Original Assignee
Sanofi SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi SA filed Critical Sanofi SA
Publication of JP2000500479A publication Critical patent/JP2000500479A/ja
Publication of JP2000500479A5 publication Critical patent/JP2000500479A5/ja
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP9519454A 1995-11-23 1996-11-21 ピラゾール誘導体、その製造方法、および該誘導体を含む医薬組成物 Pending JP2000500479A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9513956A FR2741621B1 (fr) 1995-11-23 1995-11-23 Nouveaux derives de pyrazole, procede pour leur preparation et compositions pharmaceutiques en contenant
FR95/13956 1995-11-23
PCT/FR1996/001847 WO1997019063A1 (fr) 1995-11-23 1996-11-21 Derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant

Publications (2)

Publication Number Publication Date
JP2000500479A true JP2000500479A (ja) 2000-01-18
JP2000500479A5 JP2000500479A5 (enExample) 2004-10-21

Family

ID=9484869

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9519454A Pending JP2000500479A (ja) 1995-11-23 1996-11-21 ピラゾール誘導体、その製造方法、および該誘導体を含む医薬組成物

Country Status (16)

Country Link
US (1) US6028084A (enExample)
EP (1) EP0876350B1 (enExample)
JP (1) JP2000500479A (enExample)
AT (1) ATE203015T1 (enExample)
AU (1) AU7698596A (enExample)
BR (1) BR9611618A (enExample)
CA (1) CA2238430C (enExample)
DE (1) DE69613860T2 (enExample)
DK (1) DK0876350T3 (enExample)
ES (1) ES2161382T3 (enExample)
FR (1) FR2741621B1 (enExample)
GR (1) GR3036830T3 (enExample)
MX (1) MX9803891A (enExample)
NO (1) NO310508B1 (enExample)
PT (1) PT876350E (enExample)
WO (1) WO1997019063A1 (enExample)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2006501275A (ja) * 2002-09-19 2006-01-12 ソルベイ・フアーマシユーチカルズ・ベー・ブイ カンナビノイド−ｃｂ１レセプターリガンドとしての１ｈ−１，２，４−トリアゾール−３−カルボキシアミド誘導体
JP2007514638A (ja) * 2003-06-26 2007-06-07 サノフィ−アベンティス ジフェニルピリジン誘導体、その製造法および治療用途
JP2008526887A (ja) * 2005-01-10 2008-07-24 ユニバーシティ オブ コネチカット カンナビノイド受容体に作用する新規なヘテロピロール類似体
JP2011506410A (ja) * 2007-12-10 2011-03-03 ７ティーエム ファーマ エイ／エス カンナビノイド受容体モジュレーター
JP2013500296A (ja) * 2009-07-29 2013-01-07 シーメンス アクティエンゲゼルシャフト 活性成分および活性成分を検査するための方法
JP2014507425A (ja) * 2011-09-30 2014-03-27 ナショナル ヘルス リサーチ インスティテュートス ピラゾール化合物

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US6028084A (en) 2000-02-22
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AU7698596A (en) 1997-06-11
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CA2238430A1 (en) 1997-05-29
DE69613860T2 (de) 2002-04-04
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EP0876350A1 (fr) 1998-11-11
ES2161382T3 (es) 2001-12-01
PT876350E (pt) 2001-12-28

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