IL85167A - Acids- (S) - Hydroxymethyl-6-beta-beta-luxury by the tricyclic - Google Patents

Acids- (S) - Hydroxymethyl-6-beta-beta-luxury by the tricyclic

Info

Publication number
IL85167A
IL85167A IL8516788A IL8516788A IL85167A IL 85167 A IL85167 A IL 85167A IL 8516788 A IL8516788 A IL 8516788A IL 8516788 A IL8516788 A IL 8516788A IL 85167 A IL85167 A IL 85167A
Authority
IL
Israel
Prior art keywords
product
beta
composition
added
compound
Prior art date
Application number
IL8516788A
Other languages
English (en)
Hebrew (he)
Other versions
IL85167A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL85167A0 publication Critical patent/IL85167A0/xx
Publication of IL85167A publication Critical patent/IL85167A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/86Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with only atoms other than nitrogen atoms directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL8516788A 1987-01-27 1988-01-21 Acids- (S) - Hydroxymethyl-6-beta-beta-luxury by the tricyclic IL85167A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US731987A 1987-01-27 1987-01-27

Publications (2)

Publication Number Publication Date
IL85167A0 IL85167A0 (en) 1988-07-31
IL85167A true IL85167A (en) 1994-01-25

Family

ID=21725481

Family Applications (1)

Application Number Title Priority Date Filing Date
IL8516788A IL85167A (en) 1987-01-27 1988-01-21 Acids- (S) - Hydroxymethyl-6-beta-beta-luxury by the tricyclic

Country Status (25)

Country Link
EP (1) EP0276942B1 (xx)
JP (1) JPS63246384A (xx)
KR (1) KR900005050B1 (xx)
CN (1) CN1014710B (xx)
AT (1) ATE74359T1 (xx)
AU (2) AU590142B2 (xx)
CA (1) CA1288091C (xx)
DD (1) DD279882A5 (xx)
DE (1) DE3869630D1 (xx)
DK (1) DK36788A (xx)
ES (1) ES2031589T3 (xx)
FI (1) FI880334A (xx)
GR (1) GR3004460T3 (xx)
HU (1) HU205765B (xx)
IE (1) IE60348B1 (xx)
IL (1) IL85167A (xx)
MY (1) MY102312A (xx)
NO (1) NO172493C (xx)
NZ (1) NZ223296A (xx)
PH (1) PH24478A (xx)
PL (2) PL159842B1 (xx)
PT (1) PT86613B (xx)
SU (2) SU1591812A3 (xx)
YU (2) YU46436B (xx)
ZA (1) ZA88514B (xx)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY102312A (en) * 1987-01-27 1992-05-28 Pfizer 6-beta (substituted)-c-hydroxymethyl-penicillanic acids and derivatives thereof
WO1998029114A1 (en) * 1996-12-30 1998-07-09 Bar-Ilan University Tricarboxylic acid-containing oxyalkyl esters and uses thereof
GB0128052D0 (en) * 2001-11-22 2002-01-16 Drug Discovery Lab As Compounds
US8187727B2 (en) 2005-07-22 2012-05-29 Lg Chem, Ltd. Imidazole derivatives, preparation method thereof and organic electronic device using the same

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4272439A (en) * 1978-06-02 1981-06-09 Schering Corporation 6-(Substituted-hydroxymethylene penams)
US4304779A (en) * 1979-05-09 1981-12-08 Schering Corporation 6-(Nitrogen-containing heterocyclic)hydroxymethylpenicillanic acids, compounds related thereto and processes for their preparation
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
EP0083977A1 (en) * 1982-01-11 1983-07-20 Pfizer Inc. 6-Alpha-hydroxymethylpenicillanic acid sulfone as a beta-lactamase inhibitor
SU1395144A3 (ru) * 1984-01-30 1988-05-07 Пфайзер Инк. (Фирма) Способ получени 6-замещенных метиленпенициллановых кислот,или их сложных эфиров,или их солей с щелочными металлами
DE3584015D1 (de) * 1984-01-30 1991-10-17 Pfizer 6-(substituierte) methylen-penicillansaeure und 6-(substituierte) hydroxymethyl-penicillansaeure und deren derivate.
MY102312A (en) * 1987-01-27 1992-05-28 Pfizer 6-beta (substituted)-c-hydroxymethyl-penicillanic acids and derivatives thereof

Also Published As

Publication number Publication date
NO880297L (no) 1988-07-28
YU46436B (sh) 1993-10-20
KR880009030A (ko) 1988-09-13
AU1074388A (en) 1988-07-28
AU4883290A (en) 1990-05-17
NO172493C (no) 1993-07-28
CN88100588A (zh) 1988-08-10
IE60348B1 (en) 1994-06-29
YU124389A (en) 1990-12-31
AU590142B2 (en) 1989-10-26
YU14488A (en) 1990-02-28
NZ223296A (en) 1989-10-27
SU1591812A3 (ru) 1990-09-07
PL270301A1 (en) 1988-12-08
DD279882A5 (de) 1990-06-20
PT86613A (pt) 1988-02-01
FI880334A (fi) 1988-07-28
PL159842B1 (pl) 1993-01-29
DK36788A (da) 1988-09-23
CN1014710B (zh) 1991-11-13
FI880334A0 (fi) 1988-01-26
ZA88514B (en) 1989-09-27
YU47020B (sh) 1994-11-15
DE3869630D1 (de) 1992-05-07
HUT47118A (en) 1989-01-30
ES2031589T3 (es) 1992-12-16
PT86613B (pt) 1991-12-31
KR900005050B1 (en) 1990-07-19
IE880197L (en) 1988-07-27
PH24478A (en) 1990-07-18
ATE74359T1 (de) 1992-04-15
MY102312A (en) 1992-05-28
AU613821B2 (en) 1991-08-08
PL161601B1 (pl) 1993-07-30
NO172493B (no) 1993-04-19
NO880297D0 (no) 1988-01-25
GR3004460T3 (xx) 1993-03-31
EP0276942B1 (en) 1992-04-01
HU205765B (en) 1992-06-29
EP0276942A1 (en) 1988-08-03
IL85167A0 (en) 1988-07-31
CA1288091C (en) 1991-08-27
SU1681730A3 (ru) 1991-09-30
DK36788D0 (da) 1988-01-26
JPS63246384A (ja) 1988-10-13

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