IL85167A - חומצות-)s(- הידרוקסימתיל- פניצילאניות 6-בטא-מותרות ע" י הטרוציקליל - Google Patents

חומצות-)s(- הידרוקסימתיל- פניצילאניות 6-בטא-מותרות ע" י הטרוציקליל

Info

Publication number
IL85167A
IL85167A IL8516788A IL8516788A IL85167A IL 85167 A IL85167 A IL 85167A IL 8516788 A IL8516788 A IL 8516788A IL 8516788 A IL8516788 A IL 8516788A IL 85167 A IL85167 A IL 85167A
Authority
IL
Israel
Prior art keywords
product
beta
composition
added
compound
Prior art date
Application number
IL8516788A
Other languages
English (en)
Other versions
IL85167A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL85167A0 publication Critical patent/IL85167A0/xx
Publication of IL85167A publication Critical patent/IL85167A/he

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/86—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with only atoms other than nitrogen atoms directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL8516788A 1987-01-27 1988-01-21 חומצות-)s(- הידרוקסימתיל- פניצילאניות 6-בטא-מותרות ע" י הטרוציקליל IL85167A (he)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US731987A 1987-01-27 1987-01-27

Publications (2)

Publication Number Publication Date
IL85167A0 IL85167A0 (en) 1988-07-31
IL85167A true IL85167A (he) 1994-01-25

Family

ID=21725481

Family Applications (1)

Application Number Title Priority Date Filing Date
IL8516788A IL85167A (he) 1987-01-27 1988-01-21 חומצות-)s(- הידרוקסימתיל- פניצילאניות 6-בטא-מותרות ע" י הטרוציקליל

Country Status (25)

Country Link
EP (1) EP0276942B1 (he)
JP (1) JPS63246384A (he)
KR (1) KR900005050B1 (he)
CN (1) CN1014710B (he)
AT (1) ATE74359T1 (he)
AU (2) AU590142B2 (he)
CA (1) CA1288091C (he)
DD (1) DD279882A5 (he)
DE (1) DE3869630D1 (he)
DK (1) DK36788A (he)
ES (1) ES2031589T3 (he)
FI (1) FI880334A (he)
GR (1) GR3004460T3 (he)
HU (1) HU205765B (he)
IE (1) IE60348B1 (he)
IL (1) IL85167A (he)
MY (1) MY102312A (he)
NO (1) NO172493C (he)
NZ (1) NZ223296A (he)
PH (1) PH24478A (he)
PL (2) PL159842B1 (he)
PT (1) PT86613B (he)
SU (2) SU1591812A3 (he)
YU (2) YU46436B (he)
ZA (1) ZA88514B (he)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3869630D1 (de) * 1987-01-27 1992-05-07 Pfizer 6-beta(substituierte)-(s)-hydroxymethylpenicillansaeure und deren derivate.
EP0961614A4 (en) * 1996-12-30 2002-07-24 Univ Bar Ilan OXYALKYLESTERS CONTAINING TRICARBOXYLIC ACID AND USES THEREOF
GB0128052D0 (en) * 2001-11-22 2002-01-16 Drug Discovery Lab As Compounds
US8187727B2 (en) 2005-07-22 2012-05-29 Lg Chem, Ltd. Imidazole derivatives, preparation method thereof and organic electronic device using the same

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4272439A (en) * 1978-06-02 1981-06-09 Schering Corporation 6-(Substituted-hydroxymethylene penams)
US4304779A (en) * 1979-05-09 1981-12-08 Schering Corporation 6-(Nitrogen-containing heterocyclic)hydroxymethylpenicillanic acids, compounds related thereto and processes for their preparation
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
GR77151B (he) * 1982-01-11 1984-09-07 Prizer
DD247677A5 (de) * 1984-01-30 1987-07-15 ������@���Kk�� Verfahren zur herstellung von 6-(subst.)-methylenpenicillan- und 6-(subst.)-hydroxymehtylpenicillansaeure und deren derivaten
EP0150984B1 (en) * 1984-01-30 1991-09-11 Pfizer Inc. 6-(substituted) methylenepenicillanic and 6-(substituted) hydroxymethylpenicillanic acids and derivatives thereof
DE3869630D1 (de) * 1987-01-27 1992-05-07 Pfizer 6-beta(substituierte)-(s)-hydroxymethylpenicillansaeure und deren derivate.

Also Published As

Publication number Publication date
PT86613B (pt) 1991-12-31
HUT47118A (en) 1989-01-30
DK36788D0 (da) 1988-01-26
AU4883290A (en) 1990-05-17
SU1591812A3 (ru) 1990-09-07
AU613821B2 (en) 1991-08-08
IL85167A0 (en) 1988-07-31
CA1288091C (en) 1991-08-27
PH24478A (en) 1990-07-18
AU590142B2 (en) 1989-10-26
YU14488A (en) 1990-02-28
ES2031589T3 (es) 1992-12-16
CN88100588A (zh) 1988-08-10
PL161601B1 (pl) 1993-07-30
DK36788A (da) 1988-09-23
PL159842B1 (pl) 1993-01-29
MY102312A (en) 1992-05-28
KR880009030A (ko) 1988-09-13
PL270301A1 (en) 1988-12-08
YU46436B (sh) 1993-10-20
JPS63246384A (ja) 1988-10-13
HU205765B (en) 1992-06-29
IE60348B1 (en) 1994-06-29
FI880334A (fi) 1988-07-28
FI880334A0 (fi) 1988-01-26
EP0276942A1 (en) 1988-08-03
ZA88514B (en) 1989-09-27
NO880297L (no) 1988-07-28
DE3869630D1 (de) 1992-05-07
YU47020B (sh) 1994-11-15
SU1681730A3 (ru) 1991-09-30
DD279882A5 (de) 1990-06-20
YU124389A (en) 1990-12-31
CN1014710B (zh) 1991-11-13
GR3004460T3 (he) 1993-03-31
EP0276942B1 (en) 1992-04-01
IE880197L (en) 1988-07-27
NZ223296A (en) 1989-10-27
AU1074388A (en) 1988-07-28
KR900005050B1 (en) 1990-07-19
NO172493C (no) 1993-07-28
PT86613A (pt) 1988-02-01
ATE74359T1 (de) 1992-04-15
NO172493B (no) 1993-04-19
NO880297D0 (no) 1988-01-25

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